REVIEW
|
doi:10.20944/preprints202203.0032.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
artificial intelligence; machine learning; drug design; covid-19; structure-based drug design; ligand-based drug design
Online: 2 March 2022 (03:00:37 CET)
REVIEW
|
doi:10.20944/preprints202007.0478.v2
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
Bioinformatics; Drug Design; Small Organic Molecule; Target identification; Web-based Server
Online: 25 July 2020 (17:50:30 CEST)
COMMUNICATION
|
doi:10.20944/preprints202406.0704.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
EphB2; monoclonal antibody; Cell-Based Immunization and Screening; flow cytometry
Online: 11 June 2024 (11:40:41 CEST)
REVIEW
|
doi:10.20944/preprints202306.0141.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
Mycobacterium tuberculosis; target identification; activity-based probes; affinity-based probes
Online: 2 June 2023 (07:39:37 CEST)
ARTICLE
|
doi:10.20944/preprints202112.0296.v1
Subject:
Medicine And Pharmacology,
Pharmacology And Toxicology
Keywords:
Plasmodium falciparum dihydroorotate dehydrogenase; fragment-based drug design; 2D-QSAR; DFT calculation; Lead optimization; Induced Fit docking
Online: 20 December 2021 (09:39:42 CET)
REVIEW
|
doi:10.20944/preprints202302.0510.v1
Subject:
Medicine And Pharmacology,
Pharmacology And Toxicology
Keywords:
Metal-Based Drugs; CuZn; Anti-Chemoresistance; Osteosarcoma Therapy; Ligand Biosensors.
Online: 28 February 2023 (06:51:00 CET)
ARTICLE
|
doi:10.20944/preprints202011.0292.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
Alzheimer's disease; BACE1; Molecular dynamics; MM/GBSA; Inhibitors; Drug likeness; Ligand efficiency, Kd.
Online: 10 November 2020 (09:10:50 CET)
REVIEW
|
doi:10.20944/preprints202304.1108.v1
Subject:
Medicine And Pharmacology,
Pharmacy
Keywords:
biopolymers; nanogels; drug delivery; polysaccharide-based nanogels; protein-based nanogels; nanotechnology
Online: 28 April 2023 (04:32:57 CEST)
REVIEW
|
doi:10.20944/preprints202405.0601.v1
Subject:
Biology And Life Sciences,
Life Sciences
Keywords:
Data science; Big data; Data mining; Bioinformatics; Chemometric; Medicinal chemistry; Targets; Knowledge discovery; Artificial intelligence, Machine learning, Deep learning; Data integration; Metadata, Database; QSAR; Collaborative drug discovery; Structure-based drug design; Ligand-based drug discovery; Clinical trials; Product development.
Online: 10 May 2024 (10:15:20 CEST)
REVIEW
|
doi:10.20944/preprints202209.0201.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
ligand-based pharmacophores; structure-based pharmacophores; virtual screening; drug design; machine learning; molecular dynamics; de novo design
Online: 14 September 2022 (09:10:58 CEST)
REVIEW
|
doi:10.20944/preprints202408.1879.v3
Subject:
Medicine And Pharmacology,
Complementary And Alternative Medicine
Keywords:
bacteriophage; phage therapy; antimicrobial resistance; intracellular pathogen; biofilm generating pathogen; phage vector; antibacterial phage capsid; phage-based vaccines; phage-based medicine.
Online: 9 September 2024 (11:38:59 CEST)
ARTICLE
|
doi:10.20944/preprints202012.0437.v1
Subject:
Medicine And Pharmacology,
Immunology And Allergy
Keywords:
malnutrition; translation; physiologically based pharmacokinetics; PBPK; pediatrics
Online: 17 December 2020 (16:03:40 CET)
ARTICLE
|
doi:10.20944/preprints202403.1433.v1
Subject:
Computer Science And Mathematics,
Artificial Intelligence And Machine Learning
Keywords:
FLT3 Inhibitors; Ligand-based Drug Design; Computer-Aided Drug Design; QSAR Modeling; AML Treatment
Online: 25 March 2024 (08:47:40 CET)
ARTICLE
|
doi:10.20944/preprints201807.0523.v1
Subject:
Social Sciences,
Education
Keywords:
game-based learning; game design; project-based teaching; informatics and society, cybersecurity
Online: 26 July 2018 (16:38:48 CEST)
ARTICLE
|
doi:10.20944/preprints202003.0150.v1
Subject:
Engineering,
Control And Systems Engineering
Keywords:
CFD; numerical optimization; CAD parametrization; cloud-based; design space exploration; SSIM
Online: 9 March 2020 (09:50:23 CET)
ARTICLE
|
doi:10.20944/preprints201709.0074.v1
Subject:
Engineering,
Electrical And Electronic Engineering
Keywords:
recommendation system; context awareness; location based services; mobile computing, cloud-based computing
Online: 18 September 2017 (08:54:04 CEST)
ARTICLE
|
doi:10.20944/preprints201907.0220.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
diversity; fragment-based drug discovery; library design; library size
Online: 19 July 2019 (07:54:41 CEST)
REVIEW
|
doi:10.20944/preprints202406.0966.v1
Subject:
Engineering,
Architecture, Building And Construction
Keywords:
mycelium-based material; mycelium composites; fungi; construction biomaterial; natural fibers; fiber-reinforced mycelium
Online: 14 June 2024 (11:26:16 CEST)
ARTICLE
|
doi:10.20944/preprints201806.0493.v1
Subject:
Engineering,
Electrical And Electronic Engineering
Keywords:
electromagnetically actuated cantilevers; nanometrology; multiobjective optimisation; active cantilevers; SOI-based prototyping
Online: 29 June 2018 (15:52:53 CEST)
ARTICLE
|
doi:10.20944/preprints202403.1552.v1
Subject:
Engineering,
Architecture, Building And Construction
Keywords:
bio‐based building products; bio‐based materials; building envelope; curtain wall faç ade; prefabrication; sustainable construction
Online: 26 March 2024 (12:01:24 CET)
REVIEW
|
doi:10.20944/preprints202308.0434.v1
Subject:
Medicine And Pharmacology,
Medicine And Pharmacology
Keywords:
In silico studies; drug discovery; SARS-CoV-2; molecular docking; virtual screening; molecular dynamics simulations; drug candidates; antiviral activity; receptor-ligand complex; drug design
Online: 4 August 2023 (11:11:21 CEST)
REVIEW
|
doi:10.20944/preprints201811.0409.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
G quadruplex, Oncogene, ligand, cancer
Online: 16 November 2018 (11:34:24 CET)
ARTICLE
Subject:
Engineering,
Automotive Engineering
Keywords:
Automotive development; Secure SDLC; Evidence-based standard; ISO/SAE 21434; UNECE cybersecurity regulation
Online: 9 December 2020 (10:59:57 CET)
REVIEW
|
doi:10.20944/preprints202306.1426.v1
Subject:
Medicine And Pharmacology,
Pharmacology And Toxicology
Keywords:
Trypanosomatids; squalene synthase; farnesyl diphosphate synthase; target-based approach; neglected tropical diseases.
Online: 20 June 2023 (10:27:48 CEST)
ARTICLE
|
doi:10.20944/preprints201912.0374.v1
Subject:
Biology And Life Sciences,
Biophysics
Keywords:
alpha-fetoprotein; estrogens; selective estrogen receptor modulators; homology-based modeling; molecular docking; protein-ligand interaction; amino acid substitutions
Online: 29 December 2019 (08:08:23 CET)
ARTICLE
|
doi:10.20944/preprints202310.0425.v1
Subject:
Biology And Life Sciences,
Virology
Keywords:
hepatitis B; antiviral; drug discovery; HBc protein; pharmacophore-based screening; drug repurposing
Online: 8 October 2023 (05:11:37 CEST)
ARTICLE
|
doi:10.20944/preprints202312.0193.v1
Subject:
Social Sciences,
Education
Keywords:
digital literacy; digital game-based assessment; ECGD; AHP; assessment model
Online: 4 December 2023 (15:12:33 CET)
ARTICLE
|
doi:10.20944/preprints202007.0121.v1
Subject:
Engineering,
Civil Engineering
Keywords:
performance-based building design; PBBD; high-rise residential.
Online: 7 July 2020 (09:46:46 CEST)
ARTICLE
|
doi:10.20944/preprints202012.0395.v1
Subject:
Engineering,
Automotive Engineering
Keywords:
Innovation; Up-scaling; NBS Nature-based solutions (NBS); Hydrometeorological hazards; PHUSICOS project; Flooding; Landslides; Avalanches; Rockfall; Europe
Online: 16 December 2020 (08:33:57 CET)
ARTICLE
|
doi:10.20944/preprints202310.1331.v1
Subject:
Arts And Humanities,
Architecture
Keywords:
inclusive park; disabilities; research-based design; research through designing
Online: 23 October 2023 (05:13:53 CEST)
ARTICLE
|
doi:10.20944/preprints202404.0199.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
follicular thyroid neoplasia; PAX8– PPARγ fusion; fusion protein; structure-based drug design
Online: 3 April 2024 (07:24:16 CEST)
REVIEW
|
doi:10.20944/preprints202211.0444.v1
Subject:
Chemistry And Materials Science,
Electrochemistry
Keywords:
Density functional theory; Descriptor; Carbon-based materials; Electrocatalysis; Low dimension
Online: 23 November 2022 (11:04:03 CET)
ARTICLE
|
doi:10.20944/preprints202312.1171.v1
Subject:
Engineering,
Industrial And Manufacturing Engineering
Keywords:
case-based reasoning; reliability centered maintenance; fuzzy logic technique; risk priority number
Online: 15 December 2023 (14:51:16 CET)
ARTICLE
|
doi:10.20944/preprints202305.1202.v1
Subject:
Engineering,
Aerospace Engineering
Keywords:
Generative model; Knowledge-Based Engineering; Design automation; Conceptual design; Aerospace Engineering; Computer Aided Design
Online: 17 May 2023 (07:14:32 CEST)
ARTICLE
|
doi:10.20944/preprints201810.0771.v2
Subject:
Social Sciences,
Education
Keywords:
scientific competence; competence-based education; educational planning; Education for Sustainable Development; evaluation of digital resources
Online: 29 November 2019 (03:17:18 CET)
ARTICLE
|
doi:10.20944/preprints202212.0157.v1
Subject:
Engineering,
Control And Systems Engineering
Keywords:
self-adaption; wireless sensors; model-based design; control engineering
Online: 8 December 2022 (10:24:09 CET)
ARTICLE
|
doi:10.20944/preprints201810.0513.v1
Subject:
Engineering,
Control And Systems Engineering
Keywords:
project based learning; human powered vehicles; sustainable transportation design
Online: 23 October 2018 (03:42:42 CEST)
ARTICLE
|
doi:10.20944/preprints202308.1098.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
Transcriptional meta-analysis; molecular docking; RT-qPCR; Bioinformatics; Structural-based virtual screening
Online: 15 August 2023 (11:47:28 CEST)
ARTICLE
|
doi:10.20944/preprints202409.0267.v1
Subject:
Chemistry And Materials Science,
Biomaterials
Keywords:
plant-based fibers; thermopressing; induction; fiberboards; mechanical properties; climate change
Online: 3 September 2024 (14:13:01 CEST)
ARTICLE
|
doi:10.20944/preprints202404.0603.v1
Subject:
Engineering,
Electrical And Electronic Engineering
Keywords:
beam diagnostics; electron beam; plasma-based accelerator; x-ray Free Electron Laser (XFEL).
Online: 9 April 2024 (08:44:39 CEST)
REVIEW
|
doi:10.20944/preprints202401.0523.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
antibodies; biologics; chemical entities; fluorine-based drugs; imaging; natural products; new chemical entities; oligonucleotides; peptides; TIDES
Online: 8 January 2024 (09:44:44 CET)
ARTICLE
|
doi:10.20944/preprints202311.1953.v1
Subject:
Chemistry And Materials Science,
Organic Chemistry
Keywords:
palladium-catalyzed; 2-pyridone ligand; tertiary aldehydes
Online: 30 November 2023 (05:45:42 CET)
ARTICLE
|
doi:10.20944/preprints202309.1323.v1
Subject:
Chemistry And Materials Science,
Inorganic And Nuclear Chemistry
Keywords:
dual emission; ruthenium; polypyridyl ligand; electrochemistry; photophysics
Online: 19 September 2023 (13:28:20 CEST)
ARTICLE
|
doi:10.20944/preprints201902.0124.v4
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
enzymes Cyclooxygenase, ligand, metabolites, antiinflammatory, Molecular Docking
Online: 29 May 2019 (11:39:02 CEST)
REVIEW
|
doi:10.20944/preprints201707.0019.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
affective disorders; alzheimer’s disease; l-Deprenyl (Selegiline); donepezil; galantamine; value; inhibitor constant; mechanism-based inhibition; multitarget-directed ligand (MTDL); rasagiline; rivastigmine
Online: 11 July 2017 (05:58:53 CEST)
ARTICLE
|
doi:10.20944/preprints202408.0957.v1
Subject:
Engineering,
Control And Systems Engineering
Keywords:
Automatic control; artificial intelligence; controller growing; neural-network based controller; disturbance rejection; robust control; DC motor
Online: 14 August 2024 (07:20:45 CEST)
ARTICLE
|
doi:10.20944/preprints201902.0024.v1
Subject:
Engineering,
Civil Engineering
Keywords:
infiltration based BMP’s; flood; infiltration; clogging; soil permeability; underdrain; soil saturation rate; drainage basin; urban drainage
Online: 3 February 2019 (03:05:39 CET)
ARTICLE
|
doi:10.20944/preprints202104.0157.v1
Subject:
Business, Economics And Management,
Accounting And Taxation
Keywords:
National Centralized Drug Procurement; "4+7" policy; drug price; interrupted time series; volume-based procurement.
Online: 6 April 2021 (08:18:10 CEST)
ARTICLE
|
doi:10.20944/preprints202403.1258.v1
Subject:
Engineering,
Mechanical Engineering
Keywords:
electromobility; additive manufacturing; spare parts supply; process comparison; powder bed fusion of metals via laser beam; metal extrusion-based additive manufacturing
Online: 21 March 2024 (09:17:13 CET)
ARTICLE
|
doi:10.20944/preprints202408.0959.v1
Subject:
Engineering,
Civil Engineering
Keywords:
seismic retrofit; dissipative bracings; design methods; direct displacement method; force-based design; behavior factor
Online: 14 August 2024 (07:10:33 CEST)
ARTICLE
|
doi:10.20944/preprints202310.1074.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
mixed-based combinatorial library; structure–activity relationships; cyclic peptide; mu-opioid receptor; delta-opioid receptor; bifunctional ligand; antinociception; opioid antagonist; opioid liabilities
Online: 17 October 2023 (11:21:32 CEST)
ARTICLE
|
doi:10.20944/preprints202407.1116.v1
Subject:
Biology And Life Sciences,
Life Sciences
Keywords:
Hepatitis C virus; MD Simulations; Covalent inhibitor; Drug resistance; Pharmacophore-based virtual screening
Online: 16 July 2024 (04:54:08 CEST)
ARTICLE
|
doi:10.20944/preprints202405.0060.v1
Subject:
Biology And Life Sciences,
Biophysics
Keywords:
Enthalpy-Entropy compensation; Protein Ligand Interactions; Thermodynamic Parameters
Online: 1 May 2024 (07:45:22 CEST)
REVIEW
|
doi:10.20944/preprints202404.0801.v1
Subject:
Biology And Life Sciences,
Immunology And Microbiology
Keywords:
malaria; ligand-receptor interaction; phage display; vaccine target
Online: 11 April 2024 (11:29:14 CEST)
BRIEF REPORT
Subject:
Biology And Life Sciences,
Cell And Developmental Biology
Keywords:
SARS-CoV2; spike; receptor–ligand docking; super infection
Online: 20 March 2020 (08:30:40 CET)
ARTICLE
|
doi:10.20944/preprints202211.0001.v1
Subject:
Computer Science And Mathematics,
Hardware And Architecture
Keywords:
smart attendance system; attendance monitoring system; students’ absenteeism; Bluetooth Low Energy technology; beacon-based application
Online: 1 November 2022 (01:07:13 CET)
ARTICLE
|
doi:10.20944/preprints202111.0125.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
artificial intelligence; de novo design; fragment-based drug discovery; HIV-1 inhibitors; pseudo natural products
Online: 8 November 2021 (09:23:49 CET)
ARTICLE
|
doi:10.20944/preprints202306.0249.v1
Subject:
Chemistry And Materials Science,
Applied Chemistry
Keywords:
Oxolinic acid; Metal-based complex; Spectroscopy; Microscopic characterization; Antimicrobial activity.
Online: 5 June 2023 (07:09:44 CEST)
ARTICLE
|
doi:10.20944/preprints202308.1376.v1
Subject:
Engineering,
Architecture, Building And Construction
Keywords:
air supply optimization; double-objective optimization; surrogate-based optimization; Kriging model; genetic algorithm
Online: 21 August 2023 (03:23:07 CEST)
ARTICLE
|
doi:10.20944/preprints202404.0469.v1
Subject:
Biology And Life Sciences,
Biophysics
Keywords:
Alzheimer’ s disease; amyloid β peptide; human serum albumin; low-molecular-weight ligand; protein-ligand interaction; surface plasmon resonance spectroscopy
Online: 7 April 2024 (10:18:10 CEST)
ARTICLE
|
doi:10.20944/preprints202302.0164.v1
Subject:
Environmental And Earth Sciences,
Environmental Science
Keywords:
coastal transformation; ecosystem services; transdisciplinarity; nature-based solutions; southern North Sea; Gute Küste Niedersachsen
Online: 9 February 2023 (11:17:26 CET)
ARTICLE
Subject:
Medicine And Pharmacology,
Immunology And Allergy
Keywords:
In vitro–In vivo Correlation; Physiologically Based Pharmacokinetic Model; BCS Class II; Rivaroxaban; Xarelto; Food Effect; Population Kinetics
Online: 25 January 2021 (09:41:41 CET)
ARTICLE
|
doi:10.20944/preprints201903.0166.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
Structure-based design; glycogen phosphorylase inhibitor; glycogen metabolism; type 2 diabetes; X-ray crystallography; N-acyl-β-D-glucopyranosylamine
Online: 15 March 2019 (14:06:06 CET)
ARTICLE
|
doi:10.20944/preprints202405.1612.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
Personalized cancer vaccines; Neoantigens; Pancreatic Ductal Adenocarcinoma; peptide based personalized cancer vaccine; MHC; HLA; TCR
Online: 24 May 2024 (05:54:00 CEST)
ARTICLE
|
doi:10.20944/preprints202310.1838.v1
Subject:
Engineering,
Mechanical Engineering
Keywords:
Particle swarm optimization algorithm; Reliability-based design and optimization; Simulated annealing algorithm; Most probable point
Online: 30 October 2023 (07:14:52 CET)
ARTICLE
|
doi:10.20944/preprints202401.1836.v1
Subject:
Medicine And Pharmacology,
Medicine And Pharmacology
Keywords:
Malaria; Virtual Screening; Molecular Dynamics Simulation; Pharmacophore; Modelling; Ligand
Online: 25 January 2024 (14:26:11 CET)
ARTICLE
|
doi:10.20944/preprints202104.0245.v1
Subject:
Chemistry And Materials Science,
Analytical Chemistry
Keywords:
bis(tetrazine); coordination; host-guest; ligand; silver; XRD structure
Online: 8 April 2021 (14:27:58 CEST)
ARTICLE
|
doi:10.20944/preprints201902.0064.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
Dopamine receptors, Molecular Docking, Molecular Dynamics, Receptor-Ligand Interactions
Online: 6 February 2019 (13:54:13 CET)
REVIEW
|
doi:10.20944/preprints201810.0312.v1
Subject:
Chemistry And Materials Science,
Nanotechnology
Keywords:
upconversion; nanoparticles; lanthanide; surface modification; functionalisation; ligand engineering; silanisation;
Online: 15 October 2018 (12:59:30 CEST)
ARTICLE
|
doi:10.20944/preprints202002.0097.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
Protein structure and dynamics; Molecular structure and modeling; Protein and macromolecules; Computational methods and bioinformatics; Computer-based teaching tools; Learning materials and teaching tools; Multimedia teaching tools
Online: 7 February 2020 (11:42:09 CET)
ARTICLE
|
doi:10.20944/preprints202306.0771.v1
Subject:
Engineering,
Metallurgy And Metallurgical Engineering
Keywords:
Solder Alloys; Mechanical Properties; Alloy Design; Sn-based Alloys; Data Science; Predictive models; Machine Learning
Online: 12 June 2023 (05:23:12 CEST)
ARTICLE
|
doi:10.20944/preprints202302.0428.v1
Subject:
Biology And Life Sciences,
Biology And Biotechnology
Keywords:
hybrid cheese; faba bean protein; insect protein; desirability-based mixture design; spreadability texture analysis; sensory analysis
Online: 27 February 2023 (01:44:30 CET)
REVIEW
|
doi:10.20944/preprints202409.1548.v1
Subject:
Environmental And Earth Sciences,
Sustainable Science And Technology
Keywords:
circular economy; urban design; adaptive reuse; green architecture; nature‐based solutions; regenerative cities; urban planning; resource loops; sustainable development
Online: 19 September 2024 (16:02:10 CEST)
ARTICLE
|
doi:10.20944/preprints202007.0606.v1
Subject:
Business, Economics And Management,
Business And Management
Keywords:
Design Thinking; hydrosocial contract; web-based prototype; household engagement; Product Service Systems; clustering; ICT; sustainable use of water; customization
Online: 25 July 2020 (11:27:24 CEST)
ARTICLE
|
doi:10.20944/preprints202409.0877.v1
Subject:
Biology And Life Sciences,
Biophysics
Keywords:
Ligand-Receptor Binding Affinity; ziconotide; CaV2.2; Structural Biophysics; Peptide Design
Online: 11 September 2024 (10:58:35 CEST)
REVIEW
|
doi:10.20944/preprints202407.1270.v1
Subject:
Medicine And Pharmacology,
Epidemiology And Infectious Diseases
Keywords:
Enterovirus; Multi-target directed ligand; Clinical Trials; Combination; Drug design
Online: 16 July 2024 (08:27:11 CEST)
ARTICLE
|
doi:10.20944/preprints202401.0084.v1
Subject:
Chemistry And Materials Science,
Inorganic And Nuclear Chemistry
Keywords:
lanthanide oxygen cluster; magnetocaloric effect; magnetic refrigerant materials; rhodamine ligand
Online: 3 January 2024 (02:15:52 CET)
ARTICLE
|
doi:10.20944/preprints202305.1903.v1
Subject:
Chemistry And Materials Science,
Theoretical Chemistry
Keywords:
Analysis of magnetic shieldings; electronic mechanisms; LRESC-Loc; Ligand-dependent
Online: 26 May 2023 (09:41:54 CEST)
ARTICLE
|
doi:10.20944/preprints202405.2076.v1
Subject:
Engineering,
Civil Engineering
Keywords:
IGMM Algorithm; Endurance Time Method; Life-Cycle Cost Assessment (LCCA); Multi-Objective Optimization; Reinforced Concrete Structures; Performance-Based Design
Online: 30 May 2024 (15:50:18 CEST)
ARTICLE
|
doi:10.20944/preprints202406.0622.v1
Subject:
Engineering,
Aerospace Engineering
Keywords:
contra-rotating propulsor; CFD-based design tool; composite fan blades; electric fan engine
Online: 11 June 2024 (08:56:05 CEST)
ARTICLE
|
doi:10.20944/preprints202212.0556.v1
Subject:
Environmental And Earth Sciences,
Environmental Science
Keywords:
Three Lines One Permit; web-based interactive analysis; online environmental planning analysis platform; EIA approval; Web-GIS; geospatial data; Guangzhou
Online: 29 December 2022 (08:56:25 CET)
ARTICLE
|
doi:10.20944/preprints202407.2140.v1
Subject:
Engineering,
Electrical And Electronic Engineering
Keywords:
grid-based sparse MIMO arrays; array design and optimization; mitigation of mutual coupling; adaptive desirability function; grating-lobe free arrays; side lobe reduction; machine learning
Online: 26 July 2024 (06:49:32 CEST)
ARTICLE
|
doi:10.20944/preprints202009.0006.v2
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
COVID-19; SARS-CoV-2; protein design; complementarity; competitive inhibitor; homology-based threading in rational protein design
Online: 4 March 2021 (10:14:39 CET)
ARTICLE
|
doi:10.20944/preprints202404.1891.v1
Subject:
Chemistry And Materials Science,
Inorganic And Nuclear Chemistry
Keywords:
single-molecular nanomedicine; porphyrin ligand; chemodynamic therapy; ferroptosis; breast cancer therapy
Online: 29 April 2024 (09:55:51 CEST)
BRIEF REPORT
|
doi:10.20944/preprints202004.0476.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
androgen insensitivity syndrome; androgen receptor; ligand binding domain; pathogenic mutation; bioinformatics
Online: 27 April 2020 (03:59:38 CEST)
ARTICLE
|
doi:10.20944/preprints201911.0071.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
NMDAR; amantadine; dansyl; fluorescent ligand; energy minima; molecular modelling; fluorescent bioassay
Online: 7 November 2019 (04:17:07 CET)
ARTICLE
|
doi:10.20944/preprints201910.0281.v1
Subject:
Biology And Life Sciences,
Biophysics
Keywords:
protein structural dynamics; NQO1; ligand binding; protein stability; allostery; protein degradation
Online: 24 October 2019 (15:41:46 CEST)
DATASET
|
doi:10.20944/preprints202003.0011.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
antigen-antibody complex structure; interfacial electrostatic feature; Machine Learning-Based Antibody Design; Protein Data Bank
Online: 1 March 2020 (12:39:55 CET)
ARTICLE
|
doi:10.20944/preprints202111.0241.v1
Subject:
Engineering,
Marine Engineering
Keywords:
Collaborative robotics; Human-Robot Collaboration (HRC); Knowledge-Based Approach (KBA); collaborative workplace design; systematic layout planning; digital layout optimization; what-if analysis.
Online: 12 November 2021 (17:17:02 CET)
ARTICLE
|
doi:10.20944/preprints202408.1826.v1
Subject:
Chemistry And Materials Science,
Polymers And Plastics
Keywords:
titanium; catalyst; homogeneous catalyst; copolymerization; half-titanocene; ethylene; styrene; ligand effect; cyclopentadienyl
Online: 26 August 2024 (11:30:09 CEST)
REVIEW
|
doi:10.20944/preprints202406.1388.v1
Subject:
Medicine And Pharmacology,
Hematology
Keywords:
acute myeloid leukemia; NPM1 mutation; immunogenic subtype; Programmed Death Ligand 1; immunotherapy
Online: 20 June 2024 (08:30:47 CEST)
ARTICLE
|
doi:10.20944/preprints202401.1778.v1
Subject:
Chemistry And Materials Science,
Organic Chemistry
Keywords:
Rhodium; tridentate ligand; tandem reaction; allylic decarboxylation; cycloaddition; C−N Bond Formation
Online: 25 January 2024 (05:18:35 CET)
ARTICLE
|
doi:10.20944/preprints202309.1826.v1
Subject:
Chemistry And Materials Science,
Inorganic And Nuclear Chemistry
Keywords:
coordination polymers; coordination networks; triazole ligand; iron(II); self-assembly; hydrogen bonds
Online: 27 September 2023 (07:17:13 CEST)
ARTICLE
|
doi:10.20944/preprints202305.1131.v1
Subject:
Medicine And Pharmacology,
Pediatrics, Perinatology And Child Health
Keywords:
adipokine; chemokine (C-C motif) ligand 2; interleukin-6; leptin; neonatal; preeclampsia
Online: 16 May 2023 (09:00:30 CEST)
ARTICLE
|
doi:10.20944/preprints202303.0082.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
CENPA; cell cycle; pan-cancer; diagnostic; prognostic; glioma; immune; protein-ligand docking
Online: 6 March 2023 (02:38:13 CET)
REVIEW
|
doi:10.20944/preprints202211.0484.v1
Subject:
Biology And Life Sciences,
Immunology And Microbiology
Keywords:
G-quadruplex DNA; G4-ligand; class switch recombination; transcriptional regulation; B lymphocytes
Online: 28 November 2022 (01:20:40 CET)
ARTICLE
|
doi:10.20944/preprints202204.0053.v1
Subject:
Biology And Life Sciences,
Immunology And Microbiology
Keywords:
Programmed death ligand-1; Natural products; Immunotherapy; Neoenactin B1; Molecular dynamics simulation
Online: 7 April 2022 (04:08:19 CEST)
ARTICLE
|
doi:10.20944/preprints202011.0618.v1
Subject:
Medicine And Pharmacology,
Immunology And Allergy
Keywords:
Neprilisin; Docking; Molecular Dynamics Simulation; MM-PBSA; Ligand Efficiency Metrics; ADME-Tox
Online: 24 November 2020 (14:21:22 CET)
REVIEW
|
doi:10.20944/preprints202003.0285.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
HIF-1α; NQO1; hypoxia; angiogenesis; cancer; protein:protein interactions; ligand binding; proteasomal degradation
Online: 18 March 2020 (08:45:33 CET)
REVIEW
|
doi:10.20944/preprints201608.0054.v1
Subject:
Biology And Life Sciences,
Virology
Keywords:
influenza virus; antiviral agent; proteomics; phosphoproteomics; metabolomics; transcriptomics; genomics; virtual ligand screening
Online: 5 August 2016 (12:41:07 CEST)