ARTICLE
|
doi:10.20944/preprints202308.0506.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
cemiplimab; pembrolizumab; immune checkpoint inhibitor; PD-1; cutaneous squamous cell carcinoma
Online: 7 August 2023 (10:37:53 CEST)
ARTICLE
|
doi:10.20944/preprints202306.1177.v1
Subject:
Chemistry And Materials Science,
Electrochemistry
Keywords:
layered double hydroxides; corrosion inhibitor; hydrochloric acid; chemical pickling; mild steel
Online: 16 June 2023 (05:40:46 CEST)
ARTICLE
|
doi:10.20944/preprints202305.1839.v2
Subject:
Medicine And Pharmacology,
Medicine And Pharmacology
Keywords:
Anti-tubercular agents; DprE1 inhibitor; Structure activity relationship; in vivo activity
Online: 1 June 2023 (07:42:34 CEST)
REVIEW
|
doi:10.20944/preprints202304.1087.v1
Subject:
Medicine And Pharmacology,
Endocrinology And Metabolism
Keywords:
glucose transport; SGLT2 inhibitor; diabetic nephropathy; heart failure; chronic kidney disease
Online: 28 April 2023 (03:08:47 CEST)
REVIEW
|
doi:10.20944/preprints202107.0497.v1
Subject:
Medicine And Pharmacology,
Immunology And Allergy
Keywords:
lung cancer; immune checkpoint inhibitor; perioperative therapy; neoadjuvant therapy; adjuvant therapy
Online: 21 July 2021 (14:58:36 CEST)
ARTICLE
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
Azanucleoside; DMSO; DNA methylation, epigenetics; phosphorylation; restriction factor; triphosphohydrolase; methyltransferase inhibitor
Online: 4 January 2021 (08:19:38 CET)
ARTICLE
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
Kinase Inhibitor; NEK2; Chemoresistance; Avicennia marina; Marine compounds; Molecular docking; Cancer
Online: 7 June 2020 (11:16:35 CEST)
ARTICLE
|
doi:10.20944/preprints202003.0347.v1
Subject:
Medicine And Pharmacology,
Pulmonary And Respiratory Medicine
Keywords:
nsp12; RNA-dependent-RNA polymerase; SARS-CoV-2; inhibitor; vitamin B12
Online: 23 March 2020 (07:46:54 CET)
REVIEW
|
doi:10.20944/preprints201907.0256.v1
Subject:
Biology And Life Sciences,
Cell And Developmental Biology
Keywords:
PI 3-kinase; chromosomal instability; PI3K inhibitor; cancer; tumour evolution; centrosome
Online: 23 July 2019 (11:01:34 CEST)
REVIEW
|
doi:10.20944/preprints201810.0732.v1
Subject:
Social Sciences,
Behavior Sciences
Keywords:
depression; estrogenic endocrine disruptor; environmental factor; inhibitor of differentiation; mental disorder
Online: 31 October 2018 (04:51:16 CET)
ARTICLE
|
doi:10.20944/preprints201809.0591.v1
Subject:
Medicine And Pharmacology,
Neuroscience And Neurology
Keywords:
adverse events; immune checkpoint inhibitor; myasthenia gravis; myopathy; neuropathy; nivolumab; pembrolizumab
Online: 29 September 2018 (11:28:00 CEST)
ARTICLE
|
doi:10.20944/preprints201807.0131.v1
Subject:
Medicine And Pharmacology,
Ophthalmology
Keywords:
pigmentary glaucoma; ROCK kinase inhibitor; RKI-1447; trabecular meshwork; phagocytosis; cytoskeleton
Online: 9 July 2018 (11:27:28 CEST)
ARTICLE
|
doi:10.20944/preprints201805.0088.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
p53; proteasome inhibitor; endometrial cancer; ovarian cancer; gain-of-function mutation
Online: 4 May 2018 (09:03:27 CEST)
ARTICLE
|
doi:10.20944/preprints202409.1353.v1
Subject:
Computer Science And Mathematics,
Mathematical And Computational Biology
Keywords:
Interleukin(IL); Porcupine inhibitor ETC-1922159; Sensitivity analysis; Colorectal cancer
Online: 18 September 2024 (07:13:19 CEST)
ARTICLE
|
doi:10.20944/preprints202409.0885.v1
Subject:
Computer Science And Mathematics,
Mathematical And Computational Biology
Keywords:
DNA repair; Porcupine inhibitor ETC-1922159; Sensitivity analysis; Colorectal cancer
Online: 12 September 2024 (02:52:34 CEST)
REVIEW
|
doi:10.20944/preprints202408.0282.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
familial pancreatic cancer; BRCA2; BRCA1; PARP inhibitor; Pancreatic Ductal Adenocarcinoma; Homologous recombination
Online: 5 August 2024 (14:02:08 CEST)
ARTICLE
|
doi:10.20944/preprints202407.1251.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
α-glucosidase inhibitor; biaryl polyketides; molecular docking; molecular dynamics; nonaketide; setomimycin BGC
Online: 17 July 2024 (04:16:49 CEST)
ARTICLE
|
doi:10.20944/preprints202404.1047.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
Breast cancer; EMT; TWIST1; metastasis; immunosuppression; PD-L1; immune-checkpoint-inhibitor therapy
Online: 16 April 2024 (10:47:24 CEST)
ARTICLE
|
doi:10.20944/preprints202404.0867.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
Personalized medicine; genomic instability; Miliary disease; epithelial ovarian cancer; PARP inhibitor; staging
Online: 12 April 2024 (21:20:09 CEST)
ARTICLE
|
doi:10.20944/preprints202403.0938.v1
Subject:
Medicine And Pharmacology,
Medicine And Pharmacology
Keywords:
endoplasmic reticulum stress, unfolded protein response, ER-adaptosome, PERK inhibitor, rheumatoid arthritis.
Online: 15 March 2024 (14:59:49 CET)
ARTICLE
|
doi:10.20944/preprints202312.1162.v1
Subject:
Medicine And Pharmacology,
Gastroenterology And Hepatology
Keywords:
statin; multityrosine kinase inhibitor; sorafenib resistance; hepatocellular carcinoma; lipophilic statin; hydrophilic statin
Online: 15 December 2023 (12:14:20 CET)
ARTICLE
|
doi:10.20944/preprints202310.1726.v1
Subject:
Medicine And Pharmacology,
Medicine And Pharmacology
Keywords:
dacomitinib; EGFR inhibitor; overall survival; pharmacokinetics; progression-free survival; proton pump inhibitors
Online: 27 October 2023 (07:06:07 CEST)
REVIEW
|
doi:10.20944/preprints202310.1501.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
plant triterpenoid; structure modifier; antiviral activity; HIV-1; HSV-1; maturation inhibitor
Online: 24 October 2023 (07:33:45 CEST)
ARTICLE
|
doi:10.20944/preprints202309.0739.v1
Subject:
Environmental And Earth Sciences,
Soil Science
Keywords:
Slurry application method; silage maize; nitrous oxide emissions; mineral nitrogen; nitrification inhibitor
Online: 12 September 2023 (07:24:27 CEST)
SHORT NOTE
|
doi:10.20944/preprints202307.0049.v1
Subject:
Chemistry And Materials Science,
Organic Chemistry
Keywords:
furan carboxamide; organic synthesis; furoic acid; isoniazid; molecular docking; COX-2 inhibitor
Online: 3 July 2023 (10:19:42 CEST)
REVIEW
|
doi:10.20944/preprints202305.1507.v1
Subject:
Medicine And Pharmacology,
Medicine And Pharmacology
Keywords:
Radionuclide therapy; nuclear medicine; radiopharmaceutical; antibody; peptide; small molecule inhibitor; tumor; microenvironment
Online: 22 May 2023 (10:51:48 CEST)
ARTICLE
|
doi:10.20944/preprints202305.1300.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
Apoptosis; PD-L1; catalytic topo I inhibitor; cyclin D1 overexpression; ATR; p53
Online: 18 May 2023 (08:31:34 CEST)
ARTICLE
|
doi:10.20944/preprints202301.0585.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
glioblastoma; cancer stem cells; EMT; MGMT; temozolomide; doxorubicin; STAT3; EGFR inhibitor (AG1478)
Online: 31 January 2023 (12:01:04 CET)
ARTICLE
|
doi:10.20944/preprints202212.0512.v1
Subject:
Chemistry And Materials Science,
Physical Chemistry
Keywords:
Intelligent corrosion inhibitor; Oleate imidazoline; Polyacrylamide; pH-controlled release; L80 carbon steel.
Online: 27 December 2022 (07:49:22 CET)
ARTICLE
|
doi:10.20944/preprints202201.0243.v1
Subject:
Chemistry And Materials Science,
Food Chemistry
Keywords:
aqueous micellar system; trypsin inhibitor; isoflavone extraction; non-ionic surfactant; multifactorial optimization
Online: 17 January 2022 (16:01:53 CET)
REVIEW
|
doi:10.20944/preprints202112.0482.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
non-small-cell lung cancer; immune checkpoint inhibitor; Bayesian meta-analysis; Review
Online: 30 December 2021 (12:13:58 CET)
ARTICLE
|
doi:10.20944/preprints202003.0024.v1
Subject:
Medicine And Pharmacology,
Immunology And Allergy
Keywords:
SARS-CoV-2; nonstructural proteins (NSP); NSP12; NSP7; NSP8; virtual screening; inhibitor
Online: 2 March 2020 (03:11:33 CET)
REVIEW
|
doi:10.20944/preprints201807.0254.v1
Subject:
Biology And Life Sciences,
Cell And Developmental Biology
Keywords:
endocrine disruptor, environmental health sciences, gene-environment, inhibitor of differentiation, neurocognitive disorders
Online: 14 July 2018 (23:30:36 CEST)
REVIEW
|
doi:10.20944/preprints201804.0359.v1
Subject:
Biology And Life Sciences,
Immunology And Microbiology
Keywords:
oncolytic virus; in situ autovaccination; cytokine; immune checkpoint inhibitor; immune co-stimulator
Online: 27 April 2018 (09:18:37 CEST)
ARTICLE
|
doi:10.20944/preprints201801.0177.v1
Subject:
Biology And Life Sciences,
Virology
Keywords:
Ebola; influenza virus; HIV; envelope protein; membrane fusion inhibitor; HR2; pentacyclic triterpenoids
Online: 19 January 2018 (04:02:15 CET)
ARTICLE
|
doi:10.20944/preprints202405.1741.v1
Subject:
Medicine And Pharmacology,
Neuroscience And Neurology
Keywords:
Alzheimer’ s disease; vascular complications; monoclonal antibody therapy; Aducanumab; Lecanemab; epoxide of polyunsaturated fatty acid; soluble epoxide hydrolase inhibitor EC5026; EP4 inhibitor; monocyte/macrophage; amyloid-beta degradation
Online: 27 May 2024 (13:00:54 CEST)
ARTICLE
|
doi:10.20944/preprints202409.0696.v1
Subject:
Computer Science And Mathematics,
Mathematical And Computational Biology
Keywords:
NFκ B; Porcupine inhibitor ETC-1922159; Sensitivity analysis; Colorectal cancer
Online: 10 September 2024 (03:34:23 CEST)
REVIEW
|
doi:10.20944/preprints202402.0835.v3
Subject:
Biology And Life Sciences,
Life Sciences
Keywords:
Hypertension; calcium channel blocker; combination therapy; thiazide diuretics; Renin-angiotensin-aldosterone system inhibitor
Online: 25 July 2024 (00:11:59 CEST)
ARTICLE
|
doi:10.20944/preprints202407.1116.v1
Subject:
Biology And Life Sciences,
Life Sciences
Keywords:
Hepatitis C virus; MD Simulations; Covalent inhibitor; Drug resistance; Pharmacophore-based virtual screening
Online: 16 July 2024 (04:54:08 CEST)
ARTICLE
|
doi:10.20944/preprints202312.0595.v1
Subject:
Medicine And Pharmacology,
Hematology
Keywords:
chronic myeloid leukemia; tyrosine kinase inhibitor; very elderly; safety; efficacy; outcome; dose optimization
Online: 8 December 2023 (10:26:16 CET)
ARTICLE
|
doi:10.20944/preprints202212.0023.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
spinal cord injury; X-linked inhibitor of apoptosis protein; neuroprotection; apoptosis; transgenic mice
Online: 1 December 2022 (09:59:17 CET)
ARTICLE
|
doi:10.20944/preprints202208.0208.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
Plasma PD-L1; liquid biopsy; cfRNA; immune checkpoint inhibitor; predictive immune biomarker; NSCLC
Online: 11 August 2022 (06:10:34 CEST)
ARTICLE
|
doi:10.20944/preprints202206.0144.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
Molecular docking; molecular dynamics; pharmacophore; molecular modeling; XIAP protein; protein inhibitor; anticancer activity
Online: 9 June 2022 (11:08:29 CEST)
ARTICLE
|
doi:10.20944/preprints202111.0257.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
metastatic melanoma; targeted therapy; immune checkpoint inhibitor therapy; survival; statutory health insurance data
Online: 15 November 2021 (11:50:07 CET)
COMMUNICATION
|
doi:10.20944/preprints202103.0113.v1
Subject:
Medicine And Pharmacology,
Immunology And Allergy
Keywords:
blood-based mutation burden (bTMB); cancer immunotherapy; immune checkpoint inhibitor (ICI); biomarker; mutation
Online: 2 March 2021 (21:45:40 CET)
REVIEW
Subject:
Chemistry And Materials Science,
Analytical Chemistry
Keywords:
hyperoxaluria; oxalate; inhibitor; small molecule drug; glycolate oxidase; lactate dehydrogenase; liver selective distribution
Online: 31 December 2020 (08:59:47 CET)
ARTICLE
|
doi:10.20944/preprints202007.0581.v1
Subject:
Biology And Life Sciences,
Biology And Biotechnology
Keywords:
Wheat; RNAi silencing; amylase/trypsin inhibitor (ATI); allergy; Non Celiac Wheat Sensitivity (NCWS)
Online: 24 July 2020 (11:51:53 CEST)
ARTICLE
Subject:
Medicine And Pharmacology,
Pharmacology And Toxicology
Keywords:
COVID-19; SARS-CoV-2; 3CLpro; PLpro; RdRp; AAK1; inhibitor; dock; molecular dynamics
Online: 15 March 2020 (02:34:14 CET)
ARTICLE
|
doi:10.20944/preprints201810.0570.v1
Subject:
Medicine And Pharmacology,
Pharmacology And Toxicology
Keywords:
bone resorption; butyric acid; HDAC inhibitor; osteoblasts; osteoprotegerin/RANKL; periodontal/root canal pathogens
Online: 24 October 2018 (11:21:42 CEST)
ARTICLE
|
doi:10.20944/preprints201803.0144.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
sea anemone; drug discovery; cancer; antiangiogenic; endothelial cells; RGD motif; Kunitz type inhibitor
Online: 19 March 2018 (08:15:38 CET)
ARTICLE
|
doi:10.20944/preprints202404.1491.v1
Subject:
Biology And Life Sciences,
Virology
Keywords:
HIV-2; integrase strand transfer inhibitor (INSTIs); HIV; integrase; Lenacapavir; SARs-CoV-2
Online: 23 April 2024 (05:06:50 CEST)
ARTICLE
|
doi:10.20944/preprints202404.0994.v1
Subject:
Medicine And Pharmacology,
Clinical Medicine
Keywords:
plasminogen activator inhibitor-1; obstructive sleep apnea; continuous positive airway pressure; atherogenesis; fibrinolytic capacity
Online: 16 April 2024 (07:41:29 CEST)
ARTICLE
|
doi:10.20944/preprints202311.1678.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
erythropoietin; PHD inhibitor; hypoxia; deglycosylation; proximal tubules; distal tubules; renal erythropoietin-producing interstitial cells
Online: 27 November 2023 (08:44:10 CET)
REVIEW
|
doi:10.20944/preprints202209.0296.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
non-small-cell lung cancer; performance status; cytotoxic chemotherapy; immune checkpoint inhibitor; cancer cachexia
Online: 20 September 2022 (05:53:12 CEST)
REVIEW
|
doi:10.20944/preprints202110.0450.v1
Subject:
Medicine And Pharmacology,
Gastroenterology And Hepatology
Keywords:
Fibrosis; Integrin; TGFβ; Therapeutic target; Drug; Inhibitor; Monoclonal antibody; α8β1; α11β1; Hepatic stellate cell
Online: 29 October 2021 (10:16:13 CEST)
ARTICLE
|
doi:10.20944/preprints202108.0366.v2
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
Lung adenocarcinoma; PD-1 inhibitor; LASSO analysis and SVM-RFE; Immune cell infiltration; TCGA
Online: 25 August 2021 (09:22:41 CEST)
REVIEW
|
doi:10.20944/preprints202101.0393.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
Breast cancer; Angiogenesis; Lymphangiogenesis; Cancer Stem cells, microRNA; EP4 receptor; Immune check-point inhibitor
Online: 19 January 2021 (17:40:53 CET)
COMMUNICATION
|
doi:10.20944/preprints201908.0126.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
protein-protein interaction; protein-peptide interaction; triglycine; substrate binding site; peptide; inhibitor; Proteinase K
Online: 11 August 2019 (08:37:08 CEST)
ARTICLE
|
doi:10.20944/preprints201804.0374.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
STAT3 as a drug target; cyclic STAT3 decoy; oligodeoxynucleotide inhibitor; head and neck cancer
Online: 29 April 2018 (10:10:00 CEST)
CONCEPT PAPER
|
doi:10.20944/preprints201804.0358.v1
Subject:
Medicine And Pharmacology,
Pharmacology And Toxicology
Keywords:
snakebite; antidote; inhibitor; small molecule therapeutics; SMT; secretory phospholipase; sPLA2; Neglected Tropical Disease; NTD
Online: 27 April 2018 (09:00:55 CEST)
ARTICLE
|
doi:10.20944/preprints201802.0026.v1
Subject:
Medicine And Pharmacology,
Ophthalmology
Keywords:
pig eye perfusion model; pigmentary glaucoma; ocular hypertension; ocular hypotension; phagocytosis; rho-kinase inhibitor
Online: 5 February 2018 (03:39:57 CET)
ARTICLE
|
doi:10.20944/preprints201710.0180.v1
Subject:
Biology And Life Sciences,
Immunology And Microbiology
Keywords:
primary Sjögren's syndrome; alpha-1-antitrypsin; inhibitor; 4-hydroxy-2-nonenal; autoantibody isotypes; serum
Online: 30 October 2017 (04:30:59 CET)
REVIEW
|
doi:10.20944/preprints202409.1641.v1
Subject:
Medicine And Pharmacology,
Hematology
Keywords:
Chronic Myeloid Leukemia; Bone Mineral Density; Bone Turnover; Tyrosine Kinase Inhibitor; CTX-1; Osteocalcin; Imatinib
Online: 20 September 2024 (15:06:17 CEST)
ARTICLE
|
doi:10.20944/preprints202408.2198.v1
Subject:
Chemistry And Materials Science,
Materials Science And Technology
Keywords:
inhibitor; electrochemical impedance spectroscopy; polarization curves; Langmuir; adsorption isotherms; Al-Si alloys; low carbon steel
Online: 30 August 2024 (10:57:00 CEST)
ARTICLE
|
doi:10.20944/preprints202407.2128.v1
Subject:
Medicine And Pharmacology,
Urology And Nephrology
Keywords:
metastatic renal cell carcinoma; tyrosine kinase inhibitor sunitinib; nomogram; cancer-specific survival; prognosis; treatment response
Online: 26 July 2024 (06:23:32 CEST)
REVIEW
|
doi:10.20944/preprints202401.1750.v1
Subject:
Biology And Life Sciences,
Life Sciences
Keywords:
ATR; ATR inhibitor; ceralasertib (AZD6738); DNA damage response; immune system; synthetic lethality; ATR-ATM interplay
Online: 24 January 2024 (10:02:52 CET)
ARTICLE
|
doi:10.20944/preprints202401.0336.v1
Subject:
Medicine And Pharmacology,
Urology And Nephrology
Keywords:
circulating tumor cells (CTCs); enzalutamide; bone metastases; castration-resistant prostate cancer; androgen receptor signaling inhibitor
Online: 4 January 2024 (11:29:18 CET)
ARTICLE
|
doi:10.20944/preprints202311.0210.v1
Subject:
Biology And Life Sciences,
Immunology And Microbiology
Keywords:
Brucella abortus; 3-AT; catalase inhibitor; intracellular growth; immune response; RAW 264.7 cell; ICR mouse
Online: 3 November 2023 (05:07:39 CET)
ARTICLE
|
doi:10.20944/preprints202308.0250.v3
Subject:
Biology And Life Sciences,
Life Sciences
Keywords:
PCa; Synthetic lethality; TLK1 signaling; Homologous recombination repair; TLK1 inhibitor J54; CPT-based PCa therapy
Online: 21 September 2023 (08:46:22 CEST)
ARTICLE
|
doi:10.20944/preprints202309.1118.v1
Subject:
Biology And Life Sciences,
Cell And Developmental Biology
Keywords:
epithelial-to-mesenchymal transition; heat shock transcription factor 1; HSF1 inhibitor; human mammary epithelial cells
Online: 18 September 2023 (08:51:33 CEST)
REVIEW
|
doi:10.20944/preprints202307.1897.v1
Subject:
Biology And Life Sciences,
Biology And Biotechnology
Keywords:
Keywords: recurrent glioblastoma; immunotherapy; CAR-T therapy; immune checkpoint inhibitor; cancer vaccine; oncolytic viral therapy
Online: 27 July 2023 (09:30:30 CEST)
ARTICLE
|
doi:10.20944/preprints202104.0456.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
ethidium; tetraphenylphosphonium; multidrug resistance; outer membrane permeability; efflux inhibitor; phenylalanyl-arginyl-β-naphtylamide, Polymyxin B
Online: 18 April 2021 (10:14:56 CEST)
COMMENTARY
|
doi:10.3390/sci2030070
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
small molecule inhibitor; personalized medicine; precision medicine; oncology; targeted therapy; drug delivery; drug screening; chemotherapy
Online: 8 September 2020 (00:00:00 CEST)
REVIEW
|
doi:10.20944/preprints202004.0181.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
renal cell carcinoma; angiogenesis; immune-checkpoint inhibitor; tumor microenvironment; molecular subtypes; prognostic-biomarkers; predictive factors
Online: 12 April 2020 (04:48:44 CEST)
REVIEW
|
doi:10.20944/preprints202402.1049.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
malignant pleural mesothelioma; immune checkpoint inhibitor; orphan drug; good clinical practice; Pharmaceuticals and Medical Devices Agency
Online: 20 February 2024 (04:03:22 CET)
COMMUNICATION
|
doi:10.20944/preprints202305.0704.v2
Subject:
Chemistry And Materials Science,
Other
Keywords:
protein-protein interaction inhibitor; rule of five; rule of four; QEPPI; molecular generation; virtual chemical library
Online: 30 June 2023 (08:50:24 CEST)
ARTICLE
|
doi:10.20944/preprints202306.1387.v1
Subject:
Biology And Life Sciences,
Food Science And Technology
Keywords:
press cake; soy; extrusion; meat analogue; texture; water-holding capacity; oil-binding capacity; trypsin inhibitor activity
Online: 20 June 2023 (07:20:50 CEST)
ARTICLE
|
doi:10.20944/preprints202305.1403.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
Alzheimer’s Disease; Tauopathy; Cell penetrating peptide; Polyarginine; TAT; Liposomes; Nanoparticles; Tau pathology; Tau aggregation inhibitor; Endocytosis
Online: 19 May 2023 (08:06:10 CEST)
ARTICLE
|
doi:10.20944/preprints202111.0447.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
Immunotherapy; immune-checkpoint inhibitor; response prediction; men and women; pembrolizumab; nivolumab; atezolizumab; ECOG; CRP; chemo-immunotherapy
Online: 24 November 2021 (09:02:46 CET)
REVIEW
|
doi:10.20944/preprints202106.0609.v1
Subject:
Medicine And Pharmacology,
Immunology And Allergy
Keywords:
Chronic myeloid leukaemia; chronic phase; Tyrosine kinase inhibitor; Treatment free remission; deep molecular response; BCR-ABL.
Online: 25 June 2021 (08:13:40 CEST)
REVIEW
|
doi:10.20944/preprints202104.0742.v1
Subject:
Medicine And Pharmacology,
Endocrinology And Metabolism
Keywords:
Diabetes mellitus; Glucose metabolism; Histone deacetylase; HDACs; Histone deacetylase inhibitor; HDACi, Insulin release; Sirtuins, Sirtuin activation
Online: 28 April 2021 (10:23:12 CEST)
ARTICLE
|
doi:10.20944/preprints201905.0374.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
Keywords: Tumor microenvironment (TME), glioblastoma multiforme (GBM), GBM- associated macrophages (GAMs), exosomes, oncomiR-21, STAT3 inhibitor.
Online: 31 May 2019 (08:18:33 CEST)
ARTICLE
|
doi:10.20944/preprints202409.1240.v1
Subject:
Medicine And Pharmacology,
Hematology
Keywords:
tapering; sustained response; ITP; fostamatinib; thrombopoietin analogs; Syk inhibitor; Syk; remission; purpura; thrombocytopenic; idiopathic; diarrhea; hemorrhage; thrombocytopenia
Online: 18 September 2024 (05:14:38 CEST)
REVIEW
|
doi:10.20944/preprints202408.0744.v1
Subject:
Medicine And Pharmacology,
Hematology
Keywords:
Peripheral T-cell lymphoma; Histone deacetylase (HDAC); HDAC inhibitor (HDACi); targeted therapy; epigenetic; DNA mutation; TET2; DNMT3A
Online: 12 August 2024 (05:07:04 CEST)
ARTICLE
|
doi:10.20944/preprints202403.1780.v1
Subject:
Biology And Life Sciences,
Aging
Keywords:
cardiovascular dysfunction; metabolic syndrome; renin-angiotensin system; Kallikrein-kinin system; human telomerase reverse transcriptase; complex I inhibitor
Online: 28 March 2024 (14:24:12 CET)
REVIEW
|
doi:10.20944/preprints202311.0836.v1
Subject:
Medicine And Pharmacology,
Cardiac And Cardiovascular Systems
Keywords:
Acute Decompensated Heart failure; fluid overload; loop diuretics; diuretic resistance; mineralocorticoid; SGLT2 inhibitors; ultrafiltration; Carbonic Anhydrase Inhibitor
Online: 14 November 2023 (07:52:29 CET)
ARTICLE
|
doi:10.20944/preprints202308.1201.v1
Subject:
Medicine And Pharmacology,
Pharmacy
Keywords:
Methicillin-resistant Staphylococcus aureus; poly-amidoamine dendrimers (PAMAM); anti-virulence agent, accessory gene regulator; histidine kinase inhibitor.
Online: 16 August 2023 (20:32:54 CEST)
REVIEW
|
doi:10.20944/preprints202106.0176.v1
Subject:
Medicine And Pharmacology,
Gastroenterology And Hepatology
Keywords:
chronic hepatitis B; covalently closed circular DNA; viral integration; transcription factor; nuclear receptor; transcriptional inhibitor; RNA interference
Online: 7 June 2021 (12:43:06 CEST)
ARTICLE
|
doi:10.20944/preprints202104.0732.v1
Subject:
Medicine And Pharmacology,
Immunology And Allergy
Keywords:
Epidermal Growth Factor Receptor (EGFR); mutations, EGFR tyrosine kinase inhibitor; molecular epidemiology; Non-small-cell lung cancer
Online: 28 April 2021 (07:55:22 CEST)
ARTICLE
|
doi:10.20944/preprints202009.0006.v2
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
COVID-19; SARS-CoV-2; protein design; complementarity; competitive inhibitor; homology-based threading in rational protein design
Online: 4 March 2021 (10:14:39 CET)
REVIEW
|
doi:10.20944/preprints202001.0030.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
histone deacetylase 6 inhibitor; personalized treatment; heat shock protein 90α; leukemia stem cells; imatinib resistance; targeted therapy
Online: 4 January 2020 (06:18:22 CET)
REVIEW
|
doi:10.20944/preprints201806.0163.v2
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
SIRT6, Diabetes, Gluconeogenesis, Cancer, Aging, Heart Disease, Pharmacological SIRT6 Inhibitor, Cardiac Hypertrophy, Tumorigenesis, Neurodegeneration, Neurodegenerative Diseases, AD
Online: 29 August 2018 (13:04:23 CEST)
ARTICLE
|
doi:10.20944/preprints201807.0123.v1
Subject:
Biology And Life Sciences,
Virology
Keywords:
Snake venomics; Viperidae; Protobothrops flavoviridis; Habu pit viper; Bottom-Up; Top-Down; BPP; Tripeptide metalloprotease inhibitor; Cytotoxicity
Online: 6 July 2018 (16:34:48 CEST)
TECHNICAL NOTE
|
doi:10.20944/preprints201706.0085.v1
Subject:
Engineering,
Civil Engineering
Keywords:
finite element modeling; electrochemical chloride extraction (ECE); electrical injection of corrosion inhibitor (EICI); rebar corrosion; repair mortar
Online: 19 June 2017 (13:40:09 CEST)
REVIEW
|
doi:10.20944/preprints202409.1669.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
eIF4A; mTORC2-Akt pathway; β-catenin pathway; JNK pathway; paclitaxel; doxorubicin; fluorouracil; platinum-containing drug; IGF1R/IR inhibitor
Online: 23 September 2024 (11:53:36 CEST)
REVIEW
|
doi:10.20944/preprints202401.1219.v1
Subject:
Chemistry And Materials Science,
Nanotechnology
Keywords:
biofuel; insecticides; pesticides; catalytic reduction of CO2; green economy; sustainability; biodegradation; nanoparticles; corrosion inhibitor; nanofertilizer; heavy metal detection
Online: 16 January 2024 (13:35:19 CET)
ARTICLE
|
doi:10.20944/preprints202308.1173.v1
Subject:
Medicine And Pharmacology,
Neuroscience And Neurology
Keywords:
ACEI – Angiotensin converting enzyme inhibitor; HTN - Hypertension; mRS – Modified ranking scale; NIHSS – National institute of health stroke scale
Online: 16 August 2023 (07:09:24 CEST)
ARTICLE
|
doi:10.20944/preprints201608.0211.v1
Subject:
Biology And Life Sciences,
Cell And Developmental Biology
Keywords:
Metalloproteinase; phenanthroline; metalloproteinase inhibitor; zebrafish; aryl hydrocarbon receptor; poly aromatic hydrocarbon toxicity; angiogenesis; neural crest; in vivo study
Online: 26 August 2016 (11:19:51 CEST)
CASE REPORT
|
doi:10.20944/preprints202408.0349.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
Personalized immunotherapy; Precision oncology; Immune checkpoint inhibitor (ICI); Integrative therapies; Adenoid cystic carcinoma (ACC); Frameshift mutation; Splice site mutation
Online: 6 August 2024 (12:39:34 CEST)
REVIEW
|
doi:10.20944/preprints202310.0910.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
immune checkpoint inhibitor; resistance mechanism; melanoma; oral mucosal melanoma; immunotherapy; immune checkpoint blockade; anti-PD-1; anti-CTLA-4
Online: 17 October 2023 (03:37:34 CEST)