ARTICLE
|
doi:10.20944/preprints202004.0161.v2
Subject:
Medicine And Pharmacology,
Pharmacology And Toxicology
Keywords:
COVID-19; docking; drug repurposing; natural products; in silico drug design; viral replication inhibition
Online: 1 June 2020 (02:42:54 CEST)
ARTICLE
|
doi:10.20944/preprints202106.0528.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
ACE-inhibition; antioxidant potential; processed cheddar cheese; water soluble extract; ethanol soluble extract
Online: 22 June 2021 (07:45:25 CEST)
ARTICLE
|
doi:10.20944/preprints201901.0062.v1
Subject:
Medicine And Pharmacology,
Pharmacology And Toxicology
Keywords:
small molecule; ligand; receptor; docking; molecular dynamics; DNA repair; inhibition; PCNA; ADME; toxicology
Online: 8 January 2019 (11:10:26 CET)
REVIEW
|
doi:10.20944/preprints202301.0532.v2
Subject:
Biology And Life Sciences,
Plant Sciences
Keywords:
natural products; plant extracts; Myrtus communis; medicinal plants; antimicrobial; antioxidants; antiviral; biofilm inhibition
Online: 7 February 2023 (03:33:29 CET)
ARTICLE
|
doi:10.20944/preprints202311.1460.v1
Subject:
Biology And Life Sciences,
Parasitology
Keywords:
Onchocerciasis; drug discovery; anthelmintics; O. gutturosa; motility and MTT inhibition; FDA approved drugs
Online: 23 November 2023 (09:31:11 CET)
ARTICLE
|
doi:10.20944/preprints202308.1475.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
acetylcholinesterase inhibitory test; molecular docking; blood-brain barrier permeation; memory impairment; AChE inhibition kinetics
Online: 21 August 2023 (13:46:47 CEST)
ARTICLE
|
doi:10.20944/preprints202305.0738.v1
Subject:
Environmental And Earth Sciences,
Pollution
Keywords:
carbon nanomaterials; graphene family materials; bioassay; nanotoxicology; ecotoxicology; flow cytometry; growth rate inhibition
Online: 10 May 2023 (10:36:24 CEST)
ARTICLE
|
doi:10.20944/preprints202405.0380.v1
Subject:
Medicine And Pharmacology,
Pharmacy
Keywords:
thiocarbohydrazones; Schiff base; moleculer docking; urease inhibition; pharmacokinetic properties; drug combinations
Online: 8 May 2024 (02:40:50 CEST)
ARTICLE
|
doi:10.20944/preprints202305.1006.v1
Subject:
Medicine And Pharmacology,
Pharmacology And Toxicology
Keywords:
Melanoma; drug discovery; spliceosomal inhibition; BRAF; cell line xenograft; organ histopathology
Online: 15 May 2023 (09:19:54 CEST)
ARTICLE
|
doi:10.20944/preprints201807.0351.v1
Subject:
Chemistry And Materials Science,
Materials Science And Technology
Keywords:
electrochemical sensor; inhibition bacteria sensor array; immobilization of bacteria; water pollution; pattern recognition
Online: 19 July 2018 (11:51:41 CEST)
ARTICLE
|
doi:10.20944/preprints202401.0265.v1
Subject:
Medicine And Pharmacology,
Hematology
Keywords:
Myeloproliferative neoplasms; JAK2-V617F mediated resistance; ruxolitinib; JAK2-STAT5 signaling; HSP90 inhibition
Online: 3 January 2024 (14:39:52 CET)
ARTICLE
|
doi:10.20944/preprints202309.1869.v1
Subject:
Biology And Life Sciences,
Immunology And Microbiology
Keywords:
Enterocins; Enterococcus; breast-fed infants; bacterial infection; Listeria monocytogenes; selective inhibition; probiotic
Online: 27 September 2023 (09:17:31 CEST)
ARTICLE
|
doi:10.20944/preprints202304.0914.v1
Subject:
Biology And Life Sciences,
Immunology And Microbiology
Keywords:
Metformin; Quorum sensing; Quorum quenching; Pseudomonas aeruginosa; Virulence; Drug repurposing; Anti-virulence therapy; Biofilm inhibition
Online: 25 April 2023 (09:54:20 CEST)
ARTICLE
|
doi:10.20944/preprints201711.0196.v1
Subject:
Biology And Life Sciences,
Agricultural Science And Agronomy
Keywords:
carbohydrate starvation; non-structural carbohydrate; photosynthesis; photosynthesis inhibition; respiration; relative growth rate; structure; diurnal variation
Online: 30 November 2017 (08:48:58 CET)
ARTICLE
|
doi:10.20944/preprints202111.0184.v2
Subject:
Biology And Life Sciences,
Virology
Keywords:
baloxavir marboxil; H5N1 highly pathogenic avian influenza virus; viral replication; inhibition; lung inflammation; combination therapy; oseltamivir
Online: 12 January 2022 (13:18:58 CET)
ARTICLE
|
doi:10.20944/preprints201911.0039.v1
Subject:
Medicine And Pharmacology,
Cardiac And Cardiovascular Systems
Keywords:
heart failure; Sacubitril/valsartan; Neprilysin inhibition; reduced ejection fraction; echocardiography; Nt-Pro-BNP; hemodynamic; remodeling
Online: 4 November 2019 (11:20:22 CET)
ARTICLE
|
doi:10.20944/preprints202303.0539.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
Antibiotic resistance; metallo-β-lactamases; metal-dependent enzymes; broad-spectrum inhibitors; inhibition assays; enzyme kinetics
Online: 31 March 2023 (03:35:02 CEST)
REVIEW
|
doi:10.20944/preprints202407.1216.v1
Subject:
Social Sciences,
Psychology
Keywords:
BRIEF-P; flexibility; Executive Functions; inhibition; Miyake model; working memory; Autism Spectrum Disorder
Online: 15 July 2024 (17:09:37 CEST)
ARTICLE
|
doi:10.20944/preprints202401.1958.v1
Subject:
Medicine And Pharmacology,
Neuroscience And Neurology
Keywords:
electric stimulation; H-reflex; spinal excitability; multiple sclerosis; soleus; GABA; presynaptic inhibition; rehabilitation
Online: 29 January 2024 (03:59:03 CET)
ARTICLE
|
doi:10.20944/preprints202401.1633.v1
Subject:
Biology And Life Sciences,
Neuroscience And Neurology
Keywords:
Mesencephalic locomotor region; Anticipatory Postural Adjustment; Presynaptic inhibition; Freezers; Step initiation; H-reflex
Online: 23 January 2024 (13:44:14 CET)
ARTICLE
|
doi:10.20944/preprints202103.0596.v1
Subject:
Biology And Life Sciences,
Anatomy And Physiology
Keywords:
postharvest treatment; jasmonate; metabolite profiling; lipid metabolism; Solanum lycopersicum; ethylene inhibition; fruit quality
Online: 24 March 2021 (16:12:21 CET)
ARTICLE
|
doi:10.20944/preprints202012.0289.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
remdesivir; perturbation of nucleotide pools; inhibition of RNA and DNA synthesis; CTP synthase
Online: 11 December 2020 (15:57:14 CET)
ARTICLE
|
doi:10.20944/preprints202012.0032.v1
Subject:
Biology And Life Sciences,
Anatomy And Physiology
Keywords:
Colorectal cancer; Dehydrodiisoeugenol (DEH); Autophagy inhibition; Endoplasmic reticulum (ER) stress; anti-cancer agent
Online: 1 December 2020 (14:57:00 CET)
ARTICLE
|
doi:10.20944/preprints202305.0769.v1
Subject:
Environmental And Earth Sciences,
Pollution
Keywords:
carbon nanotubes; graphene; fullerene; nanotoxicology; bioassay; growth rate inhibition; flow cytometry; nanoparticles; oxidative stress; environmental fate
Online: 10 May 2023 (14:49:02 CEST)
ARTICLE
|
doi:10.20944/preprints202307.0569.v1
Subject:
Medicine And Pharmacology,
Medicine And Pharmacology
Keywords:
Porphyromonas gingivalis; Symphytum Officinale; Panax Ginseng; Metronidazole; Biofilm Inhibition; Acylated Homoserine Lactones; Periodontal Diseases.
Online: 10 July 2023 (09:51:35 CEST)
REVIEW
Subject:
Medicine And Pharmacology,
Neuroscience And Neurology
Keywords:
hearing loss; aging; hyperactivity; excitability; loss of inhibition; neurophysiology; auditory perception; neural plasticity; speech processing
Online: 15 April 2021 (13:34:54 CEST)
ARTICLE
|
doi:10.20944/preprints201811.0330.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
hyperpigmentation; tyrosinase inhibitors; 3-(2,4-dihydroxyphenyl)propionic acid; structure-activity relationship study; B16-F10 cellular melanogenesis inhibition
Online: 14 November 2018 (09:59:45 CET)
ARTICLE
|
doi:10.20944/preprints202308.1845.v1
Subject:
Engineering,
Metallurgy And Metallurgical Engineering
Keywords:
Localised corrosion and inhibition; wire beam electrode (WBE); scanning vibrating electrode technique (SVET); scanning electrochemical microscopy (SECM)
Online: 28 August 2023 (09:54:49 CEST)
ARTICLE
|
doi:10.20944/preprints202402.1747.v1
Subject:
Medicine And Pharmacology,
Epidemiology And Infectious Diseases
Keywords:
ZIKV; NS5; aberrant MTs; MT acetylation; autophagic p62; HDAC6; tubulin deacetylase; BUZ domain; NS5 clearance; inhibition of IFN production
Online: 29 February 2024 (20:03:44 CET)
REVIEW
|
doi:10.20944/preprints202306.0051.v1
Subject:
Biology And Life Sciences,
Biology And Biotechnology
Keywords:
green synthesis; MOFs; amyloid proteins; prionase; mycotoxins; growth inhibition; quorum sensing; quorum quenching; lactamases; biofilms; chitinases; lactonases; His6-OPH
Online: 1 June 2023 (07:31:58 CEST)
ARTICLE
|
doi:10.20944/preprints202310.0589.v1
Subject:
Biology And Life Sciences,
Immunology And Microbiology
Keywords:
Daptomycin; PMMA cement; mechanical properties; elution; antimicrobial effectiveness; inhibition zone test; Vancomycin-resistant germs; PMMA spacer
Online: 10 October 2023 (07:17:42 CEST)
REVIEW
|
doi:10.20944/preprints202308.1824.v1
Subject:
Biology And Life Sciences,
Life Sciences
Keywords:
antifungal peptides; enzyme-like activity; growth inhibition; antifungal activity; fungal metabolites; quorum response molecules; combined antifungals
Online: 28 August 2023 (09:44:34 CEST)
ARTICLE
|
doi:10.20944/preprints201906.0301.v1
Subject:
Medicine And Pharmacology,
Pathology And Pathobiology
Keywords:
tumor blood vessel; Tumor Angiogenic Inhibition Triggered Necrosis (TAITN); CXCR4 antagonist; oral squamous cell carcinoma; hypoxia
Online: 28 June 2019 (15:18:43 CEST)
ARTICLE
|
doi:10.20944/preprints201806.0092.v1
Subject:
Biology And Life Sciences,
Neuroscience And Neurology
Keywords:
Neuroscience; basal ganglia; cortical layers; cerebellum; habenula; inhibition; predictions; dopamine; serotonin; acetylcholine; opioids; mirror neurons; place cells; language; imagery; working memory
Online: 7 June 2018 (06:02:29 CEST)
ARTICLE
|
doi:10.20944/preprints202301.0421.v3
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
Oncology; Immune Checkpoint Inhibition; PD-1; PD-L1; CTLA-4; Immune Related Adverse Events; Immunotherapy; Tumor Plasticity; Tumor Microenvironment; Optimum Therapy Duration
Online: 6 March 2023 (01:53:16 CET)
REVIEW
|
doi:10.20944/preprints202309.0860.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
gastrointestinal cancer; immunotherapy; cancer vaccines; dendritic cell vaccine; adoptive cell treatment; cytokine-induced killer cells; immune checkpoint inhibitors; angiogenesis inhibition
Online: 13 September 2023 (10:07:21 CEST)
REVIEW
|
doi:10.20944/preprints201707.0019.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
affective disorders; alzheimer’s disease; l-Deprenyl (Selegiline); donepezil; galantamine; value; inhibitor constant; mechanism-based inhibition; multitarget-directed ligand (MTDL); rasagiline; rivastigmine
Online: 11 July 2017 (05:58:53 CEST)
ARTICLE
|
doi:10.20944/preprints201912.0184.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
sponge; quorum sensing; quorum sensing inhibition; N-acyl homoserine lactone; Sarcotragus spinosulus; 3-Br-N-methyltyramine; 5,6-dibromo-N,N-dimethyltryptamine
Online: 13 December 2019 (12:12:54 CET)
REVIEW
|
doi:10.20944/preprints201802.0070.v1
Subject:
Environmental And Earth Sciences,
Environmental Science
Keywords:
microbial sulphide oxidation, corrosion, mine waste and water remediation, biofilm development, inhibition of Acid mine and rock draiange
Online: 8 February 2018 (15:35:56 CET)
ARTICLE
|
doi:10.20944/preprints202010.0274.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
protein aggregation; inhibition of amyloid fibril formation; antioxidants; polyphenols; cystatin C; NAC and vitamin C; amyloid fibrils; stefin B aggregation; TEM
Online: 13 October 2020 (10:49:14 CEST)
ARTICLE
|
doi:10.20944/preprints202408.1170.v1
Subject:
Chemistry And Materials Science,
Nanotechnology
Keywords:
SiO2 NPs; superhydrophobic coatings; SH-SiO2 coating; PFDTES modification; antibacterial and bacteriostatic evaluation; biofilm prevention; nanotechnology; growth inhibition
Online: 20 August 2024 (03:58:03 CEST)
ARTICLE
|
doi:10.20944/preprints202002.0134.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
autophagy; autophagonizer; target identification of label-free compound; target validation; autophagic flux; autophagy inhibition; lysosomal integrity function of Hsp70
Online: 11 February 2020 (09:03:51 CET)
ARTICLE
|
doi:10.20944/preprints202012.0414.v1
Subject:
Medicine And Pharmacology,
Pharmacology And Toxicology
Keywords:
galantamine; curcumin; in vivo AChE inhibition; acute toxicity in mice; antioxidant activity; malondialdehide levels; glutathione levels; brain homogenate; complete blood count; biochemical serum parameters
Online: 16 December 2020 (13:45:10 CET)
REVIEW
|
doi:10.20944/preprints202402.1384.v1
Subject:
Biology And Life Sciences,
Immunology And Microbiology
Keywords:
Cystic fibrosis; Pseudomonas aeruginosa; Antivirulence therapy; Quorum quenching and biofilm inhibition; Lectin and efflux pump inhibitors; Iron chelation
Online: 23 February 2024 (15:01:30 CET)
ARTICLE
|
doi:10.20944/preprints201912.0399.v1
Subject:
Biology And Life Sciences,
Immunology And Microbiology
Keywords:
natural product; actinobacteria; quorum sensing inhibition (QSI); biosynthetic gene clusters (BGCs); global natural product social networking (GNPS); cyclic dipeptides (2,5-diketopiperazines, DKPs); LC-HRMS
Online: 31 December 2019 (02:59:59 CET)
ARTICLE
|
doi:10.20944/preprints202309.0963.v1
Subject:
Physical Sciences,
Biophysics
Keywords:
edge of chaos; intermittency; difference mapping; Lyapunov exponent; consciousness; thesaurus; memristor; forth phase of water; proton; Grotthuss mechanism; gap junctions; excitation; inhibition; neuron; brain; fields of hippocampus
Online: 14 September 2023 (11:16:53 CEST)
ARTICLE
|
doi:10.20944/preprints201805.0137.v1
Subject:
Biology And Life Sciences,
Neuroscience And Neurology
Keywords:
neuroscience; thalamus; basal ganglia; cortical layers; hippocampus; cerebellum; habenula; claustrum; amygdala; inhibition; predictions; automaticity; dopamine; serotonin; acetylcholine; opioids; oxytocin; crh; glucocorticoids; cannabinoids; orexin; melanin-concentrating hormone; mirror neuron; place cells; grid cells; language; imagery; working memory; attention; consciousness; emotions
Online: 9 May 2018 (05:35:51 CEST)