ARTICLE
|
doi:10.20944/preprints202005.0397.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
SARS-CoV-2; Drug repurposing; N-acetyl-D-glucosamine; ORF1ab; Biodata mining; Protein modelling
Online: 24 May 2020 (18:49:41 CEST)
ARTICLE
|
doi:10.20944/preprints202306.0723.v1
Subject:
Medicine And Pharmacology,
Complementary And Alternative Medicine
Keywords:
Synergistic effect; Antibiotic resistance; Medicinal Plants; Penicillin G; Sutherlandia Frutescens; Microbial sensitivity tests; Drug combinations
Online: 9 June 2023 (13:09:26 CEST)
COMMUNICATION
|
doi:10.20944/preprints202212.0060.v1
Subject:
Chemistry And Materials Science,
Nanotechnology
Keywords:
exosomes; extrusion; proteolipid nanoparticles; drug delivery; nanomedicine; doxorubicin; ex-truded nanoparticles; hydroxychloroquine; endolysosomal escape; lysosomotropic
Online: 5 December 2022 (06:04:21 CET)
ARTICLE
|
doi:10.20944/preprints201901.0046.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
Keywords: methotrexate, cubic phase, magnetocubosomes, monoolein, liquid crystalline phase, drug delivery system, alternating magnetic field
Online: 4 January 2019 (14:32:38 CET)
COMMUNICATION
|
doi:10.20944/preprints202002.0421.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
De novo transcriptome assembly; brushtail possums; liver; brain cerebral cortex; drug and xenobiotic metabolism; chemical toxicants
Online: 28 February 2020 (11:49:29 CET)
ARTICLE
|
doi:10.20944/preprints202205.0256.v1
Subject:
Biology And Life Sciences,
Cell And Developmental Biology
Keywords:
Extracellular matrices; Macromolecular crowding; human iPSC derived astrocytes; human iPSC derived dopaminergic neurons; drug testing
Online: 19 May 2022 (08:50:28 CEST)
ARTICLE
|
doi:10.20944/preprints202203.0117.v3
Subject:
Medicine And Pharmacology,
Pharmacology And Toxicology
Keywords:
active pharmaceutical ingredient; compounded drug; compounding; extemporaneous formulation; manufactured material; medication; monograph; pediatric; reference standards
Online: 5 April 2022 (10:17:10 CEST)
ARTICLE
|
doi:10.20944/preprints202112.0122.v1
Subject:
Medicine And Pharmacology,
Immunology And Allergy
Keywords:
hepatitis B virus; besifovir dipivoxil maleate (BSV); nucleos(t)ide analog; drug resistance; reverse transcription
Online: 8 December 2021 (12:06:52 CET)
REVIEW
|
doi:10.20944/preprints202207.0141.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
review; real -world evidence; real -world data; randomized controlled trials; registry; digital health technology; early drug approval
Online: 8 July 2022 (11:09:58 CEST)
REVIEW
|
doi:10.20944/preprints202407.0821.v1
Subject:
Chemistry And Materials Science,
Nanotechnology
Keywords:
Nanogels; nanoparticle synthesis; hydrogels and microgels; batch chemistry; flow chemistry; microfluidics; nanomedicine; theranostics; cross-linking; drug delivery
Online: 10 July 2024 (05:08:20 CEST)
ARTICLE
|
doi:10.20944/preprints202308.0141.v1
Subject:
Chemistry And Materials Science,
Materials Science And Technology
Keywords:
A549 lung cancer; nanoparticles; cell-penetration, drug affinity, dissociation constants; molecular docking; antibacterial; hydroxychloroquine
Online: 2 August 2023 (04:54:14 CEST)
ARTICLE
|
doi:10.20944/preprints202403.0565.v1
Subject:
Chemistry And Materials Science,
Analytical Chemistry
Keywords:
Two-dimensional liquid chromatography; heart-cutting 2D-LC; veterinary drug residue; nucleotides monophosphate; sheep’s milk
Online: 11 March 2024 (08:59:00 CET)
REVIEW
|
doi:10.20944/preprints202401.0524.v1
Subject:
Biology And Life Sciences,
Life Sciences
Keywords:
transdermal drug delivery system; skin permeation; permeation enhancers; quality by design ap-proach; therapeutic applications
Online: 8 January 2024 (06:41:04 CET)
REVIEW
|
doi:10.20944/preprints202309.0207.v1
Subject:
Biology And Life Sciences,
Biology And Biotechnology
Keywords:
Neglected tropic diseases; Parasites; Chagas disease; Leishmaniasis; Life cycle; Drug target; Biochemical mechanisms; Pharmacological therapeutics; Peptides
Online: 6 September 2023 (14:52:33 CEST)
ARTICLE
|
doi:10.20944/preprints202111.0395.v1
Subject:
Chemistry And Materials Science,
Physical Chemistry
Keywords:
Tamarind Gum; Hydrogels; Semi-IPNs; Green synthesis; Silver Nanoparticles; Drug Delivery; Chemotherapeutics; HCT116 Cell; Anti-microbial
Online: 22 November 2021 (13:46:47 CET)
ARTICLE
|
doi:10.20944/preprints202402.0156.v1
Subject:
Biology And Life Sciences,
Animal Science, Veterinary Science And Zoology
Keywords:
antimicrobial resistance; biosecurity; dairy calves; ESBL E. coli; multi-drug resistant; waste milk
Online: 2 February 2024 (14:20:05 CET)
ARTICLE
|
doi:10.20944/preprints201809.0513.v1
Subject:
Medicine And Pharmacology,
Tropical Medicine
Keywords:
Malawi, HIV, tuberculosis, anti-retroviral therapy, surveillance, patient monitoring, epidemic trends, drug supply, unique patient identifiers, data analysis
Online: 27 September 2018 (15:29:43 CEST)
ARTICLE
|
doi:10.20944/preprints201809.0544.v1
Subject:
Biology And Life Sciences,
Food Science And Technology
Keywords:
Bodybuilding; Drug Free; Competing; Peaking; Carbohydrate Loading; Water Loading; Sodium Loading; Fat Loading: Vitamin C; Fibre Restriction
Online: 27 September 2018 (12:58:34 CEST)
ARTICLE
|
doi:10.20944/preprints202307.1647.v1
Subject:
Medicine And Pharmacology,
Cardiac And Cardiovascular Systems
Keywords:
non-steroidal anti-inflammatory drug; stroke; acute coronary syndrome; myocardial infarction; mortality; readmission; Arabian Gulf
Online: 25 July 2023 (08:26:22 CEST)
ARTICLE
|
doi:10.20944/preprints202105.0492.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
Drug resistance; nsp12; protein design; fitness; RNA-dependent RNA polymerase; resistance mutations; SARS-CoV-2.
Online: 20 May 2021 (13:18:14 CEST)
REVIEW
|
doi:10.20944/preprints201910.0296.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
nasal delivery; glioblastoma multiforme; drug delivery; nanoparticles; nose-to-brain delivery; pre-clinical studies; clinical evaluation
Online: 27 October 2019 (09:36:27 CET)
REVIEW
Subject:
Medicine And Pharmacology,
Pharmacology And Toxicology
Keywords:
metabolic functionalization of alkyl moieties in drug molecules; structure influence on metabolic functionalization of alkyl moieties; mechanism of alkyl free radical hydroxy functionalization; pharmacologic activity of hydroxy and carboxy functionalized alkyl moieties in drug molecules; primary and auxiliary pharmacophores; auxophores
Online: 11 March 2020 (03:20:58 CET)
REVIEW
|
doi:10.20944/preprints202407.1534.v1
Subject:
Medicine And Pharmacology,
Hematology
Keywords:
lymphoma; B‐cell; hematologic neoplasms; bruton tyrosine kinase; protein kinase inhibitors; drug resistance; neoplasm; ibrutinib; pirtobrutinib; molecular targeted therapy; chronic lymphocytic leukemia; hematopoietic stem cell transplantation; covalent inhibitors; protein degradation
Online: 18 July 2024 (17:24:05 CEST)
REVIEW
|
doi:10.20944/preprints202305.0289.v1
Subject:
Chemistry And Materials Science,
Nanotechnology
Keywords:
cancer therapy; nanomedicine; drug delivery; pH-responsiveness; EPR; intratumoral delivery; intracellular delivery; nanoparticles; metal-organic frameworks
Online: 5 May 2023 (03:45:54 CEST)
ARTICLE
|
doi:10.20944/preprints202205.0392.v1
Subject:
Biology And Life Sciences,
Biophysics
Keywords:
atrial-fibrillation; multi-target; drug promiscuity; druggable binding site; flecainide; Nav1.5; Kv1.5; binding site comparison; polypharmacology
Online: 30 May 2022 (10:10:41 CEST)
REVIEW
|
doi:10.20944/preprints202102.0619.v1
Subject:
Biology And Life Sciences,
Anatomy And Physiology
Keywords:
Nanotechnology 1; Nanomedicine 2; organic and inorganic nanoparticles 3; drug delivery 4; antitumour therapy5; tissue engineering 6.
Online: 26 February 2021 (13:31:45 CET)
ARTICLE
|
doi:10.20944/preprints202101.0490.v1
Subject:
Biology And Life Sciences,
Anatomy And Physiology
Keywords:
CD44; Cancer Stem Cells; Tumorigenesis; Drug Resistance; Immune Markers; Epithelial to Mesenchymal Transition; Therapeutic Targeting
Online: 25 January 2021 (12:23:49 CET)
ARTICLE
|
doi:10.20944/preprints202407.1336.v2
Subject:
Public Health And Healthcare,
Health Policy And Services
Keywords:
GMP, cGMP, Quality Control, Quality Assurance, EMA, DGDA, Drug regulatory authorities, Quality Medicine, Pharmacists
Online: 18 July 2024 (07:18:16 CEST)
ARTICLE
|
doi:10.20944/preprints202402.0233.v1
Subject:
Public Health And Healthcare,
Public Health And Health Services
Keywords:
depression; adolescent girls; National Survey on Drug Use and Health; pandemic
Online: 5 February 2024 (07:56:24 CET)
REVIEW
|
doi:10.20944/preprints202402.0117.v1
Subject:
Biology And Life Sciences,
Biology And Biotechnology
Keywords:
nanomedicine; biomimicry; biomimetic nanoparticle; targeted drug delivery; homotypic targeting; nanoparticle coating
Online: 2 February 2024 (07:25:29 CET)
SHORT NOTE
|
doi:10.20944/preprints202312.0899.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
monoamine oxidase; inhibitors; 1,3-oxazole; benzenesulfonamide; drug research; Parkinson’s disease; MAO
Online: 12 December 2023 (14:22:48 CET)
ARTICLE
|
doi:10.20944/preprints202312.0540.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
c-FLIP; TRAIL; apoptosis; protein-protein interaction; drug resistance; cancer treatment
Online: 7 December 2023 (14:37:18 CET)
ARTICLE
|
doi:10.20944/preprints202310.0918.v1
Subject:
Medicine And Pharmacology,
Hematology
Keywords:
drug sensitivity scores; molecular modeling; molecular docking; four-parameter logistic curve
Online: 16 October 2023 (11:38:46 CEST)
ARTICLE
|
doi:10.20944/preprints202309.1049.v1
Subject:
Medicine And Pharmacology,
Medicine And Pharmacology
Keywords:
adverse drug reactions; anaphylactic reactions; arthralgia; hip synovitis; central precocious puberty
Online: 15 September 2023 (07:09:15 CEST)
ARTICLE
|
doi:10.20944/preprints202308.2158.v1
Subject:
Biology And Life Sciences,
Virology
Keywords:
Ebola virus; measles virus; VP35; PKR; PACT; RIG-I; drug screen.
Online: 31 August 2023 (08:42:45 CEST)
ARTICLE
|
doi:10.20944/preprints202306.1076.v1
Subject:
Medicine And Pharmacology,
Hematology
Keywords:
Thymoquinone; SBE-β-CD; Leukemia; Drug delivery system; Telomerase inhibition; Apoptosis
Online: 15 June 2023 (05:37:50 CEST)
ARTICLE
|
doi:10.20944/preprints202306.0257.v1
Subject:
Medicine And Pharmacology,
Dermatology
Keywords:
wound dressing; drug delivery; organ culture, infection models, ciprofloxacin, infected wounds
Online: 5 June 2023 (08:09:29 CEST)
ARTICLE
|
doi:10.20944/preprints202306.0109.v1
Subject:
Biology And Life Sciences,
Cell And Developmental Biology
Keywords:
triple negative breast cancer; MCAK/KIF2C; aneuploidy; chromosomal instability; drug discovery
Online: 1 June 2023 (15:47:29 CEST)
ARTICLE
|
doi:10.20944/preprints202305.1693.v1
Subject:
Computer Science And Mathematics,
Artificial Intelligence And Machine Learning
Keywords:
Digital twin; Clinical trials; Quality by Design; Blockchain technology; Drug development
Online: 24 May 2023 (04:46:13 CEST)
ARTICLE
|
doi:10.20944/preprints202305.1006.v1
Subject:
Medicine And Pharmacology,
Pharmacology And Toxicology
Keywords:
Melanoma; drug discovery; spliceosomal inhibition; BRAF; cell line xenograft; organ histopathology
Online: 15 May 2023 (09:19:54 CEST)
ARTICLE
|
doi:10.20944/preprints202305.0332.v1
Subject:
Medicine And Pharmacology,
Ophthalmology
Keywords:
Ophthalmology; Toxicology Pharmacology and therapeutics; Drug interactions; Pharma-cology and therapeutics
Online: 5 May 2023 (08:56:37 CEST)
REVIEW
|
doi:10.20944/preprints202212.0581.v1
Subject:
Biology And Life Sciences,
Virology
Keywords:
Japanese encephalitis (JE); Japanese Encephalitis Virus (JEV); Therapeutics; Vaccine; Antiviral; Drug
Online: 30 December 2022 (09:57:27 CET)
BRIEF REPORT
|
doi:10.20944/preprints202211.0063.v1
Subject:
Medicine And Pharmacology,
Pharmacology And Toxicology
Keywords:
melanoma; drug discovery; spliceosomal inhibition; acute toxicity; blood chemistry; organ histopathology
Online: 3 November 2022 (01:43:05 CET)
ARTICLE
|
doi:10.20944/preprints202210.0219.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
Endometriosis; Orbignya speciosa; Copaifera lansgdorffii nanoemulsion; self-nanoemulsifying drug delivery system
Online: 17 October 2022 (02:07:50 CEST)
COMMUNICATION
|
doi:10.20944/preprints202208.0039.v1
Subject:
Biology And Life Sciences,
Virology
Keywords:
Echovirus; enterovirus; broad-spectrum antiviral agent; antiviral drug combination; antiviral strategy
Online: 2 August 2022 (05:01:21 CEST)
REVIEW
|
doi:10.20944/preprints202201.0117.v1
Subject:
Biology And Life Sciences,
Cell And Developmental Biology
Keywords:
G protein-coupled receptor; mouse models; skin cancer; UVR; drug; network
Online: 10 January 2022 (13:41:08 CET)
ARTICLE
|
doi:10.20944/preprints202110.0021.v1
Subject:
Medicine And Pharmacology,
Medicine And Pharmacology
Keywords:
chitosan; dexketoprofen trometamol; drug delivery; gelatin; NSAIDs; personalized medicine; smart polymers
Online: 1 October 2021 (13:53:53 CEST)
ARTICLE
Subject:
Medicine And Pharmacology,
Otolaryngology
Keywords:
Drug-induced hearing loss; cochlea; outer hair cells; hearing protection; SIRT3
Online: 9 August 2021 (07:50:36 CEST)
ARTICLE
|
doi:10.20944/preprints202108.0031.v1
Subject:
Medicine And Pharmacology,
Immunology And Allergy
Keywords:
antibiotics; antimicrobial resistance; antimicrobial stewardship; AWaRe; Pharmacovigilance; Lareb; adverse drug reactions
Online: 2 August 2021 (12:27:02 CEST)
ARTICLE
|
doi:10.20944/preprints202107.0246.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
influenza virus; virus-host interaction; commonly prescribed drugs; drug adverse reaction
Online: 12 July 2021 (11:37:07 CEST)
ARTICLE
|
doi:10.20944/preprints202104.0385.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
antibiotic resistance; antimicrobial susceptibility testing; novel diagnostics; polymicrobial; sputum; drug resistant
Online: 14 April 2021 (14:21:15 CEST)
ARTICLE
|
doi:10.20944/preprints202012.0534.v1
Subject:
Medicine And Pharmacology,
Immunology And Allergy
Keywords:
creatinine; vancomycin; amikacin; renal impairment; acute kidney injury; adverse drug reaction
Online: 21 December 2020 (15:42:59 CET)
ARTICLE
|
doi:10.20944/preprints202012.0358.v1
Subject:
Chemistry And Materials Science,
Analytical Chemistry
Keywords:
Antitumor agents; Fluorescence lifetime imaging; Medicinal chemistry; Metabolic drug; Mitochondrial carrier
Online: 15 December 2020 (08:35:30 CET)
ARTICLE
|
doi:10.20944/preprints202009.0205.v1
Subject:
Medicine And Pharmacology,
Pharmacology And Toxicology
Keywords:
Franz-Bampa; BCS drugs; biomimetic membrane; Franz cell; passive drug transport
Online: 9 September 2020 (10:25:54 CEST)
REVIEW
|
doi:10.20944/preprints202008.0729.v2
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
p53; p73; MDM2; MDMX; tumor suppressor; drug repurposing; aspirin; protoporphyrin IX; verteporfin
Online: 17 September 2020 (07:23:37 CEST)
REVIEW
|
doi:10.20944/preprints202007.0478.v2
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
Bioinformatics; Drug Design; Small Organic Molecule; Target identification; Web-based Server
Online: 25 July 2020 (17:50:30 CEST)
ARTICLE
|
doi:10.20944/preprints202006.0358.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
Enzyme inhibition; Secondary Metabolites; In-silico Analysis; Molecular docking; Drug candidates
Online: 30 June 2020 (08:11:28 CEST)
HYPOTHESIS
|
doi:10.20944/preprints202004.0215.v1
Subject:
Medicine And Pharmacology,
Neuroscience And Neurology
Keywords:
endocanabinoid system; sleep deprivation; animal models; psychosis-like symptoms; drug development
Online: 14 April 2020 (06:28:23 CEST)
REVIEW
|
doi:10.20944/preprints202004.0012.v1
Subject:
Chemistry And Materials Science,
Theoretical Chemistry
Keywords:
chemoinformatics; chemical space; database; LANaPD; molecular diversity; drug discovery; natural sources
Online: 2 April 2020 (04:47:13 CEST)
ARTICLE
Subject:
Medicine And Pharmacology,
Clinical Medicine
Keywords:
humans; infection control; therapy; coronavirus; immunoglobulins; drug therapy; therapeutic use; corticosteroid
Online: 8 March 2020 (17:04:19 CET)
REVIEW
Subject:
Medicine And Pharmacology,
Anesthesiology And Pain Medicine
Keywords:
pharmacology; drug development; sodium channel; potassium channel; TRP channel; HCN channels
Online: 8 August 2019 (12:31:26 CEST)
ARTICLE
|
doi:10.20944/preprints201810.0236.v1
Subject:
Biology And Life Sciences,
Immunology And Microbiology
Keywords:
essential oils; drug resistant microorganisms; antimicrobial activity; antifungal activity; medicinal plants
Online: 11 October 2018 (11:51:16 CEST)
ARTICLE
|
doi:10.20944/preprints201809.0558.v1
Subject:
Chemistry And Materials Science,
Nanotechnology
Keywords:
Alginate, Chitosan, Layer-by-layer, Magnetic nanoparticles, Drug delivery, Cancer, Curcumin
Online: 28 September 2018 (09:26:48 CEST)
HYPOTHESIS
|
doi:10.20944/preprints201808.0127.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
Big Data, Systems Models, Cancer metabolism, Cancer personalized treatment, Drug Discovery.
Online: 6 August 2018 (15:09:15 CEST)
ARTICLE
|
doi:10.20944/preprints201806.0192.v1
Subject:
Biology And Life Sciences,
Biology And Biotechnology
Keywords:
β4-galactosyltransferase 4; transcriptional mechanism; sensor cells; colon cancer; drug screening
Online: 12 June 2018 (12:51:07 CEST)
REVIEW
|
doi:10.20944/preprints201805.0378.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
annexins; inflammation; wound healing; host-pathogen interplay; drug target; translational research
Online: 27 May 2018 (11:32:34 CEST)
ARTICLE
|
doi:10.20944/preprints201711.0090.v1
Subject:
Medicine And Pharmacology,
Dentistry And Oral Surgery
Keywords:
drug delivery; dentine; diffusion; bio-active molecules; CFD; μ-LIF; microfluidics
Online: 14 November 2017 (10:15:29 CET)
REVIEW
|
doi:10.20944/preprints202209.0201.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
ligand-based pharmacophores; structure-based pharmacophores; virtual screening; drug design; machine learning; molecular dynamics; de novo design
Online: 14 September 2022 (09:10:58 CEST)
ARTICLE
|
doi:10.20944/preprints202308.1963.v1
Subject:
Chemistry And Materials Science,
Biomaterials
Keywords:
Core-shell nanogels; nonlinear PEG; anisole; biocompatible; thermo-responsive; curcumin stability, high loading capacity; drug delivery
Online: 30 August 2023 (04:08:45 CEST)
REVIEW
|
doi:10.20944/preprints202108.0447.v1
Subject:
Medicine And Pharmacology,
Pharmacology And Toxicology
Keywords:
Interferons; IFNα; IFNß; IFNγ; antiviral; antiproliferative; immunomodulator; PEGylation; formulation; encapsulate IFNs; drug delivery system; liposomes; polymeric micelles; microparticles; nanoparticles
Online: 23 August 2021 (13:51:44 CEST)
ARTICLE
|
doi:10.20944/preprints202209.0417.v1
Subject:
Medicine And Pharmacology,
Cardiac And Cardiovascular Systems
Keywords:
Recreational substance abuse; drug abuse; marijuana; amphetamine; acute ischemic stroke; risk factors; young adult; NIS; Stroke; Sudden Cardiac Death
Online: 27 September 2022 (09:41:00 CEST)
ARTICLE
|
doi:10.20944/preprints202004.0198.v1
Subject:
Medicine And Pharmacology,
Gastroenterology And Hepatology
Keywords:
mathematical modelling; peristalsis; smoothed particle hydrodynamics (SPH); fluid dynamics; large intestine; colonl proximal colon; fluid-structure interactions; drug delivery
Online: 12 April 2020 (15:57:17 CEST)
REVIEW
|
doi:10.20944/preprints202406.0054.v1
Subject:
Medicine And Pharmacology,
Dermatology
Keywords:
melanoma; cancer vaccine; mRNA vaccine; renin-angiotensin system; drug repurposing; immunotherapy; embryonic stem cells; cancer stem cells
Online: 3 June 2024 (09:54:04 CEST)
REVIEW
|
doi:10.20944/preprints201812.0170.v1
Subject:
Biology And Life Sciences,
Biology And Biotechnology
Keywords:
bacterial nanocellulose; nanofibrillated nanocellulose; animal nanocellulose; algal nanocellulose; tissue engineering; tissue repair; wound dressing; cell delivery; drug delivery; antimicrobial properties
Online: 14 December 2018 (06:44:53 CET)
ARTICLE
|
doi:10.20944/preprints201811.0574.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
activity cliff; activity landscape plotter; epigenetics; docking; drug discovery; D-tools; molecular dynamics; Epi-polypharmacology; SmART; structure-activity relationships
Online: 26 November 2018 (07:14:05 CET)
ARTICLE
Subject:
Biology And Life Sciences,
Anatomy And Physiology
Keywords:
COVID-19; SARS-CoV-2; in silico drug discovery; gene expression profile; tensor decomposition; feature extraction
Online: 8 December 2020 (10:17:05 CET)
ARTICLE
|
doi:10.20944/preprints201812.0018.v2
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
colorectal cancer; differentially expressed genes; biomarkers; protein-protein interaction; reporter biomolecules; candidate drugs; systems biology; drug repositioning
Online: 29 December 2018 (07:05:05 CET)
ARTICLE
Subject:
Medicine And Pharmacology,
Pharmacology And Toxicology
Keywords:
Covid-19; proteins; normal-modes; protein-drug interactions; chloroquine; ivermectin; remdesivir; sofosbuvir; boceprevir; α-difluoromethylornithine (DMFO)
Online: 11 August 2020 (04:09:43 CEST)
ARTICLE
|
doi:10.20944/preprints202405.1908.v1
Subject:
Biology And Life Sciences,
Life Sciences
Keywords:
Breast cancer; Target Identification; Protein-Protein Interaction; Network Pharmacology; Drug Discovery; KEEG; Enrichment analysis; Text Mining; Cytoscape
Online: 29 May 2024 (08:33:40 CEST)
ARTICLE
|
doi:10.20944/preprints202109.0052.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
RNAi; drug delivery; siRNA delivery; DsiRNA delivery; RNAi delivery; Chol-DsiRNA polymer micelles; Chol-siRNA polymer micelles
Online: 3 September 2021 (08:56:48 CEST)
ARTICLE
|
doi:10.20944/preprints202305.1334.v1
Subject:
Public Health And Healthcare,
Public Health And Health Services
Keywords:
victimizing and perpetrating violence; interpersonal and intimate violence; harmful alcohol and drug use; mental health symptoms; paths of violence; gender
Online: 18 May 2023 (10:46:13 CEST)
ARTICLE
|
doi:10.20944/preprints202408.1941.v1
Subject:
Mathematical And Computational Biology,
Computer Science And Mathematics
Keywords:
Drug Response Prediction; Graph Neural Network; Graph Attention Networks; Heterogeneous Graph; Interpretability
Online: 27 August 2024 (12:44:15 CEST)
ARTICLE
|
doi:10.20944/preprints202407.1667.v1
Subject:
Biology And Life Sciences,
Biology And Biotechnology
Keywords:
active targeting; CRT peptide; drug delivery; cancer; nanoemulsion
Online: 22 July 2024 (07:50:13 CEST)
ARTICLE
|
doi:10.20944/preprints202406.1032.v1
Subject:
Medicine And Pharmacology,
Endocrinology And Metabolism
Keywords:
Semaglutide Analogues; GLP-1 Receptor Agonists; Binding Affinity Optimization; Computational Drug Design;
Online: 17 June 2024 (09:12:54 CEST)
REVIEW
|
doi:10.20944/preprints202312.2253.v1
Subject:
Medicine And Pharmacology,
Medicine And Pharmacology
Keywords:
Ganoderma lucidum; Nanotechnology; Nanoparticles; Triterpenoids; Polysaccharides; Bioactive compounds; Drug delivery; Cancer therapy
Online: 29 December 2023 (11:31:12 CET)
ARTICLE
|
doi:10.20944/preprints202307.1905.v1
Subject:
Medicine And Pharmacology,
Pharmacology And Toxicology
Keywords:
Colorectal cancer; pharmacovigilance; BRAF inhibitors; regorafenib; encorafenib; adverse drug reactions; renal disorders
Online: 28 July 2023 (02:34:59 CEST)
ARTICLE
|
doi:10.20944/preprints202307.1577.v1
Subject:
Computer Science And Mathematics,
Artificial Intelligence And Machine Learning
Keywords:
deep learning, transformer, drug use detection, exploratory data analysis, natural language processing.
Online: 24 July 2023 (10:57:47 CEST)
REVIEW
|
doi:10.20944/preprints202306.0220.v1
Subject:
Chemistry And Materials Science,
Biomaterials
Keywords:
hydrogel-forming microneedles; transdermal drug delivery; controlled release; permeation pathway; environmental response
Online: 2 June 2023 (15:57:01 CEST)
REVIEW
|
doi:10.20944/preprints202305.1084.v1
Subject:
Medicine And Pharmacology,
Medicine And Pharmacology
Keywords:
antibody-drug conjugate; lysosome; cathepsin; legumain; self-immolation; payload release; peptidomimetic; linker
Online: 16 May 2023 (04:51:34 CEST)
REVIEW
|
doi:10.20944/preprints202212.0207.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
Blood-Brain Barrier; Brain Drug Delivery; Carbon Nanomaterials; Cerebral Gliomas; Glioblastoma; Nanoparticles.
Online: 12 December 2022 (14:56:45 CET)
ARTICLE
|
doi:10.20944/preprints202211.0296.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
antimicrobial resistance; broad-spectrum antibiotics; antibacterial drug discovery; gram-negative bacteria; pyrrolobenzodiazepines
Online: 16 November 2022 (04:20:55 CET)
REVIEW
|
doi:10.20944/preprints202211.0062.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
membrane transporter; SLC; solute carrier; drug design; pharmacokinetics; prodrug; nanoparticle; bile acids
Online: 3 November 2022 (01:09:54 CET)
ARTICLE
|
doi:10.20944/preprints202210.0141.v1
Subject:
Biology And Life Sciences,
Immunology And Microbiology
Keywords:
AtbFinder; antibiotic susceptibility testing; cystic fibrosis; Pseudomonas aeruginosa; multi-drug re-sistant
Online: 11 October 2022 (04:56:32 CEST)
REVIEW
|
doi:10.20944/preprints202104.0652.v1
Subject:
Chemistry And Materials Science,
Biomaterials
Keywords:
Enzymatic reaction; crosslinking; Hydrogel; Biomedical application; Tissue engineering; Wound healing; Drug delivery
Online: 26 April 2021 (10:52:24 CEST)
ARTICLE
|
doi:10.20944/preprints202103.0621.v1
Subject:
Medicine And Pharmacology,
Immunology And Allergy
Keywords:
Auger electron; cisplatin; 191Pt; 189Pt; radio-drug; DNA double-strand break; γH2AX
Online: 25 March 2021 (14:30:14 CET)
CASE REPORT
|
doi:10.20944/preprints202103.0054.v1
Subject:
Medicine And Pharmacology,
Immunology And Allergy
Keywords:
DRESS syndrome, Eosinophilia, Adverse drug reaction, HHV-6 reactivation, Bactrim adverse reaction
Online: 2 March 2021 (09:26:48 CET)
REVIEW
|
doi:10.20944/preprints202102.0449.v1
Subject:
Chemistry And Materials Science,
Materials Science And Technology
Keywords:
multifunctional; hydrogel nanocomposties; tissue engineering; drug delivery; wound healing; bioprinting; biowearable devices
Online: 22 February 2021 (08:48:20 CET)
ARTICLE
|
doi:10.20944/preprints202012.0513.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
apoferritin nanocarriers; controlled drug delivery; idarubicin; ferritin receptor targeting; folate receptor targeting
Online: 21 December 2020 (11:28:08 CET)
COMMUNICATION
|
doi:10.20944/preprints202011.0441.v1
Subject:
Biology And Life Sciences,
Anatomy And Physiology
Keywords:
Sars-Cov-2; Proteomic,; Ghost proteome,; Alternative proteins,; AltOrf.; interactomic; drug repurposing
Online: 16 November 2020 (17:50:19 CET)
ARTICLE
|
doi:10.20944/preprints202004.0524.v2
Subject:
Biology And Life Sciences,
Virology
Keywords:
unsupervised learning; tensor decomposition; feature selection; COVID-19; drug discovery; gene expression
Online: 3 June 2020 (05:29:09 CEST)