REVIEW
|
doi:10.20944/preprints202008.0273.v1
Subject:
Medicine And Pharmacology,
Pharmacology And Toxicology
Keywords:
Mycobacterium abscessus, drug treatment, experimental therapy, review,
Online: 12 August 2020 (08:01:41 CEST)
REVIEW
|
doi:10.20944/preprints202008.0100.v1
Subject:
Medicine And Pharmacology,
Pharmacology And Toxicology
Keywords:
adrenoceptor; constitutive activity; drug development; inverse agonism
Online: 4 August 2020 (16:01:12 CEST)
REVIEW
|
doi:10.20944/preprints202005.0408.v1
Subject:
Medicine And Pharmacology,
Pharmacology And Toxicology
Keywords:
drug discovery; machine learning; in silico; pharmacology
Online: 25 May 2020 (04:55:24 CEST)
ARTICLE
|
doi:10.20944/preprints202005.0057.v2
Subject:
Medicine And Pharmacology,
Epidemiology And Infectious Diseases
Keywords:
COVID-19; treatment; drug; survival; antiviral; hydroxychloroquine
Online: 9 May 2020 (04:45:37 CEST)
REVIEW
|
doi:10.20944/preprints201810.0512.v1
Subject:
Medicine And Pharmacology,
Pharmacology And Toxicology
Keywords:
nanotechnology; diatom; biosilica; drug delivery; hybrid devices
Online: 22 October 2018 (16:15:47 CEST)
ARTICLE
|
doi:10.20944/preprints201710.0143.v1
Subject:
Medicine And Pharmacology,
Pharmacology And Toxicology
Keywords:
cheminformatics; docking simulation; drug repositioning; thiopurine; tyrosinase
Online: 22 October 2017 (14:03:13 CEST)
CONCEPT PAPER
|
doi:10.20944/preprints202405.1739.v1
Subject:
Biology And Life Sciences,
Biophysics
Keywords:
Drug Discovery & Design; Synthetic Data Generation; Intermolecular Binding Affinity (Kd); GIBAC
Online: 27 May 2024 (10:49:40 CEST)
REVIEW
|
doi:10.20944/preprints202311.1051.v1
Subject:
Biology And Life Sciences,
Parasitology
Keywords:
Toxoplasma gondii; proteomics; host-parasite interactions; PTMs; drug discovery
Online: 16 November 2023 (07:46:09 CET)
ARTICLE
|
doi:10.20944/preprints202311.0140.v1
Subject:
Medicine And Pharmacology,
Medicine And Pharmacology
Keywords:
Electrospinning; Polysaccharides; Antibacterial; Cancer treatment; Core-shell nanofibers, Drug delivery systems
Online: 2 November 2023 (09:12:20 CET)
REVIEW
|
doi:10.20944/preprints202310.0962.v1
Subject:
Medicine And Pharmacology,
Medicine And Pharmacology
Keywords:
oxygen; nanobubbles; hypoxia; mitochondria; metabolism, molecular; drug delivery; cancer, stress; innovation
Online: 16 October 2023 (11:09:22 CEST)
REVIEW
|
doi:10.20944/preprints202110.0069.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
biology; drug resistance; gene expression profiling; mRNA; multiple myeloma; prognosis; treatment
Online: 5 October 2021 (08:20:44 CEST)
REVIEW
|
doi:10.20944/preprints202311.0246.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
bladder cancer; non-muscle-invasive cancer; local intravesical drug delivery; colloidal drug delivery systems; indwelling devices; sustained delivery
Online: 3 November 2023 (11:26:53 CET)
ARTICLE
|
doi:10.20944/preprints202004.0448.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
acetyleugenol; Acacia nilotica; anti-tuberculosis; Serine/Threonine kinases; multi-drug resistant TB
Online: 24 April 2020 (14:12:33 CEST)
REVIEW
|
doi:10.20944/preprints202208.0180.v1
Subject:
Medicine And Pharmacology,
Psychiatry And Mental Health
Keywords:
Nitrous Oxid; N₂O; nangs; systematic review; harm reduction; drug use
Online: 9 August 2022 (11:29:40 CEST)
REVIEW
|
doi:10.20944/preprints202005.0342.v1
Subject:
Medicine And Pharmacology,
Pharmacology And Toxicology
Keywords:
seaweed; metabolites; neuroprotection; Alzheimer’s disease; Parkinson’s disease; ischemic stroke; computer-aided drug discovery
Online: 21 May 2020 (09:49:29 CEST)
REVIEW
|
doi:10.20944/preprints202208.0230.v1
Subject:
Chemistry And Materials Science,
Theoretical Chemistry
Keywords:
chemoinformatics; compound databases; chemical space; diversity; drug discovery; openscience; pseudo-natural product
Online: 12 August 2022 (08:39:40 CEST)
ARTICLE
|
doi:10.20944/preprints202308.2113.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
herbs; spices; flavonoids; antioxidants; diabetes; volatile compounds; drug discovery; phytochemicals; human health
Online: 31 August 2023 (10:12:18 CEST)
ARTICLE
|
doi:10.20944/preprints202105.0308.v1
Subject:
Biology And Life Sciences,
Anatomy And Physiology
Keywords:
Indonesia; biodiversity; novel antibiotics; drug screening; bioactivity; gene cluster networking; GNPS
Online: 13 May 2021 (14:05:00 CEST)
REVIEW
|
doi:10.20944/preprints202012.0242.v1
Subject:
Medicine And Pharmacology,
Immunology And Allergy
Keywords:
COVID-19; SARS-CoV-2; long-haul; inflammation; tissue damage; drug repurposing
Online: 10 December 2020 (09:42:20 CET)
ARTICLE
|
doi:10.20944/preprints202312.0574.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
DOCK program; GOLD program; Grb14; insulin receptor (IR); structure-based drug screening (SBDS)
Online: 8 December 2023 (08:24:15 CET)
REVIEW
|
doi:10.20944/preprints202408.1827.v1
Subject:
Computer Science And Mathematics,
Mathematical And Computational Biology
Keywords:
Predictive Toxicology; Omics Technologies; Machine Learning; Structure-Activity Relationship; Fragment-Based Drug Design; Microphysiological Systems; Physiologically Based Pharmacokinetic Modeling; Virtual Screening; Biochemical Targets; Automated De Novo Drug Design
Online: 26 August 2024 (11:31:51 CEST)
ARTICLE
|
doi:10.20944/preprints202308.2094.v1
Subject:
Medicine And Pharmacology,
Gastroenterology And Hepatology
Keywords:
biosimilars; bio-originators; biologic drug; ulcerative colitis; Crohn’s disease; interchangeability; economics
Online: 31 August 2023 (02:41:46 CEST)
REVIEW
|
doi:10.20944/preprints202210.0142.v1
Subject:
Medicine And Pharmacology,
Pharmacology And Toxicology
Keywords:
bioactive compounds; anthocyanins; drug delivery system; nanoparticles; chronic diseases; health benefits
Online: 11 October 2022 (05:04:19 CEST)
REVIEW
|
doi:10.20944/preprints202206.0333.v1
Subject:
Medicine And Pharmacology,
Medicine And Pharmacology
Keywords:
hPSCs derived-organoids; Culture strategy; Disease modeling; Drug screening; Regenerative therapy
Online: 24 June 2022 (08:11:15 CEST)
ARTICLE
|
doi:10.20944/preprints202106.0279.v1
Subject:
Biology And Life Sciences,
Animal Science, Veterinary Science And Zoology
Keywords:
Blood-Brain Barrier, Penetrating Peptides, Machine learning techniques, Drug delivery, Therapeutic peptides
Online: 10 June 2021 (08:13:15 CEST)
DATA DESCRIPTOR
|
doi:10.20944/preprints202209.0323.v1
Subject:
Computer Science And Mathematics,
Information Systems
Keywords:
COVID-19; Open-source dataset; Drug Repurposing; Database system; Web application devel-opment; software development; Drug fingerprints; Bulk upload
Online: 21 September 2022 (10:14:11 CEST)
ARTICLE
|
doi:10.20944/preprints202402.0537.v1
Subject:
Social Sciences,
Sociology
Keywords:
Family environment, Family interventions, Statistical test, and Extent of drug addiction.
Online: 9 February 2024 (09:59:43 CET)
REVIEW
|
doi:10.20944/preprints202407.1682.v1
Subject:
Medicine And Pharmacology,
Medicine And Pharmacology
Keywords:
pharmacogenetics; blood-brain barrier; drug discovery; personalised medicine; precision medicine; clinical translation
Online: 22 July 2024 (09:54:15 CEST)
ARTICLE
|
doi:10.20944/preprints202309.0467.v1
Subject:
Biology And Life Sciences,
Life Sciences
Keywords:
pan-cancer analysis; RKIP; YY1; gene expression; mutations; immune infiltration; drug resistance
Online: 7 September 2023 (13:33:14 CEST)
CONCEPT PAPER
|
doi:10.20944/preprints202004.0213.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
covid-19; rlmE MTase; new drug target; corona diagnosis; corona pandemic
Online: 13 April 2020 (12:33:22 CEST)
ARTICLE
|
doi:10.20944/preprints201804.0310.v1
Subject:
Medicine And Pharmacology,
Ophthalmology
Keywords:
primary open angle glaucoma; dorzolamide/timolol fixed combination; drug efficacy; safety
Online: 24 April 2018 (08:36:58 CEST)
REVIEW
|
doi:10.20944/preprints202211.0070.v1
Subject:
Biology And Life Sciences,
Food Science And Technology
Keywords:
Nutraceuticals; Personalized Medicine; Precision Medicine; Probiotics; Vitamins; Covid; Dietary Supplements; Adverse Drug Effects
Online: 3 November 2022 (06:27:25 CET)
ARTICLE
|
doi:10.20944/preprints202403.0918.v1
Subject:
Chemistry And Materials Science,
Biomaterials
Keywords:
Raman technology; recovery and resource utilization technology; process control; biogenic carbonate waste; chitin; calcium acetate drug; carotenoids.
Online: 15 March 2024 (12:01:12 CET)
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
oleanolic acid derivatives; synthesis; anti-tumor activity; molecular docking; computer-aided drug design
Online: 24 April 2017 (12:08:36 CEST)
ARTICLE
|
doi:10.20944/preprints202403.0750.v1
Subject:
Biology And Life Sciences,
Virology
Keywords:
Hepatitis B virus; drug resistance; people living with HIV; Botswana; Africa
Online: 13 March 2024 (11:38:15 CET)
COMMUNICATION
|
doi:10.20944/preprints202007.0709.v1
Subject:
Biology And Life Sciences,
Cell And Developmental Biology
Keywords:
intrinsic multi-drug resistance; acquired multi-drug resistance; circulating tumor cells; single cells; cell clusters; cell monolayer; multi-cellular spheroids; cytometry of reaction rate constant; ovarian cancer
Online: 30 July 2020 (09:01:50 CEST)
ARTICLE
|
doi:10.20944/preprints202407.1758.v1
Subject:
Medicine And Pharmacology,
Medicine And Pharmacology
Keywords:
oxaliplatin; hepatic arterial infusion chemotherapy; adverse drug reactions
Online: 23 July 2024 (11:25:24 CEST)
CASE REPORT
|
doi:10.20944/preprints202407.0750.v1
Subject:
Medicine And Pharmacology,
Epidemiology And Infectious Diseases
Keywords:
carbapenem-resistant enterobacteriaceae; drug resistance; microbial; public health
Online: 9 July 2024 (13:50:48 CEST)
ARTICLE
|
doi:10.20944/preprints202407.0490.v1
Subject:
Biology And Life Sciences,
Life Sciences
Keywords:
Gait disorders; Stroke; Muscle synergies; EMG; Drug traitment
Online: 8 July 2024 (13:16:43 CEST)
ARTICLE
|
doi:10.20944/preprints202401.0907.v1
Subject:
Biology And Life Sciences,
Life Sciences
Keywords:
cancer; protein degradation; degraders; drug discovery; PROTAC; CDK9
Online: 11 January 2024 (10:20:13 CET)
REVIEW
|
doi:10.20944/preprints202312.1293.v1
Subject:
Biology And Life Sciences,
Life Sciences
Keywords:
Topoisomerases; Drug resistance; Molecular heterogeneity; Neoplasms; Combinatorial approaches
Online: 18 December 2023 (13:52:10 CET)
REVIEW
|
doi:10.20944/preprints202310.0881.v1
Subject:
Biology And Life Sciences,
Immunology And Microbiology
Keywords:
Biofilm; proteins; drug target; essential; non-host homologous
Online: 13 October 2023 (11:34:33 CEST)
CASE REPORT
|
doi:10.20944/preprints202309.1048.v1
Subject:
Medicine And Pharmacology,
Clinical Medicine
Keywords:
drug induced autoimmune hepatitis; AIH; DILI; acute hepatitis
Online: 15 September 2023 (10:56:37 CEST)
ARTICLE
|
doi:10.20944/preprints202308.0037.v1
Subject:
Medicine And Pharmacology,
Pharmacology And Toxicology
Keywords:
NONMEM; covariate analysis; PopPK; therapeutic drug monitoring; children.
Online: 1 August 2023 (10:00:25 CEST)
ARTICLE
|
doi:10.20944/preprints202306.1769.v1
Subject:
Medicine And Pharmacology,
Epidemiology And Infectious Diseases
Keywords:
Multi-drug resistance; Gram-negative bacteria; Enterobacterales; carbapenemases
Online: 26 June 2023 (09:40:12 CEST)
ARTICLE
|
doi:10.20944/preprints202209.0288.v1
Subject:
Biology And Life Sciences,
Virology
Keywords:
COVID-19; Therapeutics; Drug Repurposing; 3D Tissue Models
Online: 20 September 2022 (03:24:22 CEST)
ARTICLE
|
doi:10.20944/preprints202209.0126.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
liposome; tumor-targeted; radiation; tumor; drug delivery; chemotherapy
Online: 8 September 2022 (14:06:26 CEST)
ARTICLE
|
doi:10.20944/preprints202208.0331.v1
Subject:
Computer Science And Mathematics,
Information Systems
Keywords:
Drug-Target Binding Affinity; Multi-Instance Learning; Transformer
Online: 18 August 2022 (03:58:34 CEST)
REVIEW
|
doi:10.20944/preprints202204.0093.v1
Subject:
Biology And Life Sciences,
Immunology And Microbiology
Keywords:
Electrophile signaling; drug mechanism; immunology; antioxidant response; apoptosis
Online: 11 April 2022 (10:39:31 CEST)
ARTICLE
|
doi:10.20944/preprints202201.0263.v1
Subject:
Biology And Life Sciences,
Immunology And Microbiology
Keywords:
drug resistance; ABC transporter; efflux pump; cryptococcosis; aging
Online: 18 January 2022 (15:56:02 CET)
ARTICLE
|
doi:10.20944/preprints202106.0675.v1
Subject:
Biology And Life Sciences,
Anatomy And Physiology
Keywords:
pharmacogenes; transcripts; sex-bias; drug metabolism; sex differences
Online: 28 June 2021 (15:08:38 CEST)
ARTICLE
|
doi:10.20944/preprints202105.0746.v1
Subject:
Biology And Life Sciences,
Anatomy And Physiology
Keywords:
ABC transporter; ABCB1; P-glycoprotein; taxol; drug recognition
Online: 31 May 2021 (11:27:14 CEST)
REVIEW
|
doi:10.20944/preprints202104.0679.v1
Subject:
Medicine And Pharmacology,
Immunology And Allergy
Keywords:
Sildenafil; phosphodiesterase 5 inhibitors; drug repurposing; cancer; chemoadjuvant
Online: 26 April 2021 (15:02:08 CEST)
ARTICLE
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
K-Ras; Hsp90; Cdc37; nanoclustering; cancer; drug development
Online: 31 March 2021 (15:30:27 CEST)
REVIEW
|
doi:10.20944/preprints202103.0771.v1
Subject:
Medicine And Pharmacology,
Immunology And Allergy
Keywords:
cancer; gold nanoparticles; marine; drug delivery; imaging; detection
Online: 31 March 2021 (14:44:42 CEST)
REVIEW
|
doi:10.20944/preprints202101.0503.v1
Subject:
Medicine And Pharmacology,
Neuroscience And Neurology
Keywords:
CNS; Drug receptors; GABA; Cannabinoid; Opioid; Serotonin; Dopamine
Online: 25 January 2021 (14:15:20 CET)
ARTICLE
|
doi:10.20944/preprints202004.0466.v1
Subject:
Biology And Life Sciences,
Endocrinology And Metabolism
Keywords:
COVID-19; coronavirus; ACE2; bioinformatics analysis; drug prediction
Online: 26 April 2020 (03:14:50 CEST)
REVIEW
|
doi:10.20944/preprints202003.0345.v2
Subject:
Medicine And Pharmacology,
Pharmacology And Toxicology
Keywords:
COVID-19; lysosomotropic agents; endosome; antiviral; drug repurposing
Online: 24 March 2020 (06:26:54 CET)
ARTICLE
|
doi:10.20944/preprints202003.0060.v1
Subject:
Medicine And Pharmacology,
Dietetics And Nutrition
Keywords:
Alcaligenes faecalis; Diabetic foot ulcer; extensive-drug resistant
Online: 4 March 2020 (10:34:23 CET)
CONCEPT PAPER
|
doi:10.20944/preprints202001.0040.v1
Subject:
Medicine And Pharmacology,
Pharmacology And Toxicology
Keywords:
cybernetics; complex systems; new drug development; human system
Online: 5 January 2020 (15:38:27 CET)
REVIEW
|
doi:10.20944/preprints201912.0342.v1
Subject:
Biology And Life Sciences,
Immunology And Microbiology
Keywords:
Anti-MDR strategies; anti-persistent treatments; drug repurposing
Online: 25 December 2019 (09:33:57 CET)
ARTICLE
|
doi:10.20944/preprints201811.0608.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
spheroids; concentration gradient generator; drug screening; high-throughput
Online: 28 November 2018 (10:08:05 CET)
ARTICLE
|
doi:10.20944/preprints201809.0587.v1
Subject:
Biology And Life Sciences,
Biology And Biotechnology
Keywords:
machine learning; conotoxins; cone snails; venom; drug discovery
Online: 29 September 2018 (07:39:42 CEST)
REVIEW
|
doi:10.20944/preprints201805.0319.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
annexins; inflammation; wound healing; drug target; translational research
Online: 23 May 2018 (08:19:42 CEST)
ARTICLE
|
doi:10.20944/preprints201802.0012.v3
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
chitosan; self-assembled; polyelectrolyte complex; nanoparticle; drug delivery
Online: 21 February 2018 (16:00:38 CET)
ARTICLE
|
doi:10.20944/preprints202311.0766.v1
Subject:
Medicine And Pharmacology,
Neuroscience And Neurology
Keywords:
Alzheimer's disease; neural networks; Training and learning; early diagnosis; drug discovery; brain diseases
Online: 13 November 2023 (08:41:42 CET)
REVIEW
|
doi:10.20944/preprints202402.0148.v1
Subject:
Medicine And Pharmacology,
Dentistry And Oral Surgery
Keywords:
medication-related osteonecrosis of the jaw; drug holiday; treatment; tooth extraction; incidence
Online: 2 February 2024 (11:48:46 CET)
ARTICLE
|
doi:10.20944/preprints202111.0364.v1
Subject:
Medicine And Pharmacology,
Ophthalmology
Keywords:
Polymeric micelles; cannabidiol (CBD); spray-drying; ocular drug delivery; corneal epithelial cells
Online: 19 November 2021 (14:48:27 CET)
ARTICLE
|
doi:10.20944/preprints202405.0360.v1
Subject:
Medicine And Pharmacology,
Neuroscience And Neurology
Keywords:
Traumatic brain injury; TBI; secondary injury; peptide therapeutics; cell penetrating peptide; pro-inflammatory cytokines; intranasal drug delivery; blood brain barrier
Online: 7 May 2024 (11:13:30 CEST)
ARTICLE
|
doi:10.20944/preprints202403.1775.v1
Subject:
Biology And Life Sciences,
Virology
Keywords:
Hepatitis B virus; Antivirals; Flavonoid; Drug discovery; Pharmacophore; Quantitative structure-activity relationship
Online: 28 March 2024 (13:31:24 CET)
REVIEW
|
doi:10.20944/preprints202107.0650.v1
Subject:
Medicine And Pharmacology,
Immunology And Allergy
Keywords:
chronic disorders; inflammation; human superorganism; holobiont; microbiome; multimorbidity; microimmunosome; polypharmacy; drug safety; sustainable healthcare
Online: 29 July 2021 (11:37:20 CEST)
ARTICLE
|
doi:10.20944/preprints202105.0158.v1
Subject:
Medicine And Pharmacology,
Immunology And Allergy
Keywords:
Imatinib; NLC; Tween 80; SLS; MTT Assay; Release study; Drug delivery; Breast cancer
Online: 10 May 2021 (10:13:02 CEST)
REVIEW
Subject:
Biology And Life Sciences,
Cell And Developmental Biology
Keywords:
nucleoid-associated proteins (NAPs); moonlighting proteins; drug target; biofilm; specificity determination; phylogenetic analysis
Online: 7 June 2020 (09:07:56 CEST)
ARTICLE
|
doi:10.20944/preprints202311.1816.v1
Subject:
Medicine And Pharmacology,
Pharmacology And Toxicology
Keywords:
essential antimicrobials; essential medicine list; drug procurement; gap analysis; paediatric antibiotic formulations
Online: 29 November 2023 (11:04:15 CET)
ARTICLE
|
doi:10.20944/preprints202311.1179.v1
Subject:
Public Health And Healthcare,
Public Health And Health Services
Keywords:
reporting; system; chemical; drug overdose; poisoning; surveillance; Makkah Almukarramah; Saudi Arabia
Online: 17 November 2023 (15:04:33 CET)
ARTICLE
|
doi:10.20944/preprints202111.0072.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
antimalarial drugs; artemisinins; ACTs; resistance; amino-artemisinins, pharmacokinetics; metabolism; Cmax; drug efficacy
Online: 3 November 2021 (09:10:50 CET)
ARTICLE
|
doi:10.20944/preprints202003.0393.v1
Subject:
Biology And Life Sciences,
Biophysics
Keywords:
SARS-CoV2; RNA depended RNA polymerase; Valproic acid Co-A; drug repurposing
Online: 26 March 2020 (15:04:22 CET)
ARTICLE
|
doi:10.20944/preprints202309.0417.v1
Subject:
Medicine And Pharmacology,
Pharmacology And Toxicology
Keywords:
adenylosuccinic acid; Duchenne muscular dystrophy; myopathy; metabolic disease; skeletal muscle; toxicology; drug development
Online: 7 September 2023 (05:09:43 CEST)
ARTICLE
|
doi:10.20944/preprints202301.0076.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
COVID-19; drug repurposing; long COVID; molecular docking; molecular dynamics; SARS-CoV-2
Online: 4 January 2023 (09:38:47 CET)
ARTICLE
|
doi:10.20944/preprints202311.0653.v1
Subject:
Medicine And Pharmacology,
Pharmacology And Toxicology
Keywords:
Cytochrome P450 oxidoreductase; POR; gnomAD, CAH; drug metabolism, steroid hormones; SNV; bioinformatics
Online: 9 November 2023 (15:09:12 CET)
ARTICLE
|
doi:10.20944/preprints202212.0170.v1
Subject:
Medicine And Pharmacology,
Pharmacology And Toxicology
Keywords:
SonoCloud; GL261 mouse model; ultrasound-mediated drug delivery; glioblastoma; immune checkpoint inhibitors
Online: 9 December 2022 (02:59:28 CET)
ARTICLE
|
doi:10.20944/preprints202405.1100.v1
Subject:
Medicine And Pharmacology,
Anesthesiology And Pain Medicine
Keywords:
ibuprofen; diclofenac; celecoxib; membrane interaction; lipid composition; medium pH; drug concentration; analgesic activity; gastrointestinal toxicity
Online: 17 May 2024 (03:10:22 CEST)
ARTICLE
|
doi:10.20944/preprints202208.0317.v1
Subject:
Biology And Life Sciences,
Endocrinology And Metabolism
Keywords:
Cytochrome P450; POR; Congenital adrenal hyperplasia; metabolic disorders; CYP3A4; protein stability; drug metabolism
Online: 17 August 2022 (10:02:51 CEST)
ARTICLE
|
doi:10.20944/preprints202310.1539.v1
Subject:
Computer Science And Mathematics,
Mathematical And Computational Biology
Keywords:
graph neural network; convolutional neural network; drug-target affinity; sequence and structural knowledge; heterogeneous models
Online: 25 October 2023 (08:23:34 CEST)
ARTICLE
|
doi:10.20944/preprints202306.0038.v1
Subject:
Medicine And Pharmacology,
Pharmacy
Keywords:
Lagenaria siceraria; In silico study; Drug design; Diabetes mellitus; Molecular docking; ADMET
Online: 1 June 2023 (05:41:13 CEST)
ARTICLE
|
doi:10.20944/preprints202310.0980.v1
Subject:
Chemistry And Materials Science,
Surfaces, Coatings And Films
Keywords:
microparticles; scalable manufacturing; laser cutting; drug delivery; complex structures; composites; core-shell; defined size
Online: 16 October 2023 (16:53:55 CEST)
ARTICLE
|
doi:10.20944/preprints202011.0292.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
Alzheimer's disease; BACE1; Molecular dynamics; MM/GBSA; Inhibitors; Drug likeness; Ligand efficiency, Kd.
Online: 10 November 2020 (09:10:50 CET)
ARTICLE
|
doi:10.20944/preprints202209.0090.v1
Subject:
Computer Science And Mathematics,
Computational Mathematics
Keywords:
epithelial cell; antibody response; basic reproduction number; transcritical bifurcation; impulsive control; drug holidays
Online: 6 September 2022 (10:25:07 CEST)
COMMUNICATION
|
doi:10.20944/preprints202012.0823.v1
Subject:
Medicine And Pharmacology,
Immunology And Allergy
Keywords:
neuroscience; rheumatology; osteoarthritis; pain; peripheral nerve; biological drug; growth factor; peptide; monoclonal antibody; ion channel
Online: 31 December 2020 (15:41:05 CET)
REVIEW
|
doi:10.20944/preprints202210.0347.v1
Subject:
Medicine And Pharmacology,
Pharmacology And Toxicology
Keywords:
monkeypox virus; infection; treatment; antiviral; drug; management; public health emergency; tecovirimat; cidofovir; bibliometric analysis
Online: 24 October 2022 (03:38:12 CEST)
REVIEW
|
doi:10.20944/preprints202207.0031.v1
Subject:
Biology And Life Sciences,
Biophysics
Keywords:
Cell-state transitions; Phenotypic plasticity; Cancer Stem Cells; Intratumoral heterogeneity; Lamarckian Induction; Drug resistance
Online: 4 July 2022 (04:56:00 CEST)
ARTICLE
|
doi:10.20944/preprints202307.1492.v1
Subject:
Medicine And Pharmacology,
Neuroscience And Neurology
Keywords:
HIV; antiretroviral drug; combination antiretroviral therapy; mitochondrial dysfunction; human microglia; iron; neural cell; metabolic reprogramming
Online: 21 July 2023 (09:50:45 CEST)
ARTICLE
|
doi:10.20944/preprints202403.1579.v2
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
Multiple Drug Resistant breast cancer; Anaphase Promoting Complex; cell culture; PDX mouse model
Online: 28 March 2024 (13:34:15 CET)
ARTICLE
|
doi:10.20944/preprints202308.0025.v1
Subject:
Chemistry And Materials Science,
Biomaterials
Keywords:
cells culture; drug delivery; FT-IR; mice skin; thermal analysis; UV-Vis; Zetasizer
Online: 1 August 2023 (09:47:56 CEST)
REVIEW
|
doi:10.20944/preprints202408.0057.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
antibody-drug conjugates; urothelial cancer; enfortumab vedotin; bystander effect
Online: 2 August 2024 (03:52:03 CEST)
ARTICLE
|
doi:10.20944/preprints202407.1965.v1
Subject:
Biology And Life Sciences,
Biology And Biotechnology
Keywords:
curcumin; breast cancer; chitosan; nanoparticle; drug delivery; cancer therapy
Online: 24 July 2024 (17:43:03 CEST)
ARTICLE
|
doi:10.20944/preprints202404.1974.v1
Subject:
Medicine And Pharmacology,
Other
Keywords:
Respiratory virus; Long COVID; Nasal drug; EGCG-palmitate; Nanoformulations
Online: 30 April 2024 (11:45:40 CEST)
ARTICLE
|
doi:10.20944/preprints202402.0808.v1
Subject:
Medicine And Pharmacology,
Pharmacology And Toxicology
Keywords:
drug-induced hiccups; FAERS; nuclear receptor; stress response pathways
Online: 15 February 2024 (01:25:14 CET)
ARTICLE
|
doi:10.20944/preprints202401.1525.v1
Subject:
Medicine And Pharmacology,
Pharmacy
Keywords:
Fingolimod; nanoemulsion; ocular drug delivery; sterilization; stability; physicochemical characterization
Online: 22 January 2024 (10:08:55 CET)
ARTICLE
|
doi:10.20944/preprints202312.1368.v1
Subject:
Physical Sciences,
Condensed Matter Physics
Keywords:
porous composites; corona treatment; polyelectrolyte multilayers, drug delivery systems.
Online: 19 December 2023 (09:38:56 CET)