ARTICLE
|
doi:10.20944/preprints202304.0625.v1
Subject:
Medicine And Pharmacology,
Pharmacology And Toxicology
Keywords:
adverse drug reaction; cisplatin liposomes; circulating tumor cells; enhanced permeability and retention effect; nephrotoxicity; pulmonary metastasis of pancreatic cancer; quality of life; recurrent liver metastases from primary nasal cancer
Online: 20 April 2023 (07:52:10 CEST)
REVIEW
|
doi:10.20944/preprints202407.1682.v1
Subject:
Medicine And Pharmacology,
Medicine And Pharmacology
Keywords:
pharmacogenetics; blood-brain barrier; drug discovery; personalised medicine; precision medicine; clinical translation
Online: 22 July 2024 (09:54:15 CEST)
ARTICLE
|
doi:10.20944/preprints202406.1032.v1
Subject:
Medicine And Pharmacology,
Endocrinology And Metabolism
Keywords:
Semaglutide Analogues; GLP-1 Receptor Agonists; Binding Affinity Optimization; Computational Drug Design;
Online: 17 June 2024 (09:12:54 CEST)
CONCEPT PAPER
|
doi:10.20944/preprints202405.1739.v1
Subject:
Biology And Life Sciences,
Biophysics
Keywords:
Drug Discovery & Design; Synthetic Data Generation; Intermolecular Binding Affinity (Kd); GIBAC
Online: 27 May 2024 (10:49:40 CEST)
REVIEW
|
doi:10.20944/preprints202404.1013.v3
Subject:
Medicine And Pharmacology,
Pharmacy
Keywords:
computational pharmaceutics; AI; multi-scale modeling; quantum computing; drug discovery; blockchain frameworks
Online: 22 April 2024 (18:38:54 CEST)
REVIEW
|
doi:10.20944/preprints202404.0674.v1
Subject:
Environmental And Earth Sciences,
Other
Keywords:
Microneedles; Bioactive molecules; Transdermal drug delivery system; Design parameters; Manufacturing techniques; Usage
Online: 9 April 2024 (14:52:30 CEST)
ARTICLE
|
doi:10.20944/preprints202403.1775.v1
Subject:
Biology And Life Sciences,
Virology
Keywords:
Hepatitis B virus; Antivirals; Flavonoid; Drug discovery; Pharmacophore; Quantitative structure-activity relationship
Online: 28 March 2024 (13:31:24 CET)
REVIEW
|
doi:10.20944/preprints202403.0140.v1
Subject:
Medicine And Pharmacology,
Complementary And Alternative Medicine
Keywords:
Cancer Pharmacotherapy; Drug development; Kinesin motor proteins; Microtubules; Mitotic kinases; Mitotic poisons
Online: 4 March 2024 (11:17:25 CET)
REVIEW
|
doi:10.20944/preprints202402.0148.v1
Subject:
Medicine And Pharmacology,
Dentistry And Oral Surgery
Keywords:
medication-related osteonecrosis of the jaw; drug holiday; treatment; tooth extraction; incidence
Online: 2 February 2024 (11:48:46 CET)
ARTICLE
|
doi:10.20944/preprints202311.1816.v1
Subject:
Medicine And Pharmacology,
Pharmacology And Toxicology
Keywords:
essential antimicrobials; essential medicine list; drug procurement; gap analysis; paediatric antibiotic formulations
Online: 29 November 2023 (11:04:15 CET)
ARTICLE
|
doi:10.20944/preprints202311.1179.v1
Subject:
Public Health And Healthcare,
Public Health And Health Services
Keywords:
reporting; system; chemical; drug overdose; poisoning; surveillance; Makkah Almukarramah; Saudi Arabia
Online: 17 November 2023 (15:04:33 CET)
ARTICLE
|
doi:10.20944/preprints202311.0653.v1
Subject:
Medicine And Pharmacology,
Pharmacology And Toxicology
Keywords:
Cytochrome P450 oxidoreductase; POR; gnomAD, CAH; drug metabolism, steroid hormones; SNV; bioinformatics
Online: 9 November 2023 (15:09:12 CET)
ARTICLE
|
doi:10.20944/preprints202309.0467.v1
Subject:
Biology And Life Sciences,
Life Sciences
Keywords:
pan-cancer analysis; RKIP; YY1; gene expression; mutations; immune infiltration; drug resistance
Online: 7 September 2023 (13:33:14 CEST)
ARTICLE
|
doi:10.20944/preprints202308.2113.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
herbs; spices; flavonoids; antioxidants; diabetes; volatile compounds; drug discovery; phytochemicals; human health
Online: 31 August 2023 (10:12:18 CEST)
ARTICLE
|
doi:10.20944/preprints202307.1905.v1
Subject:
Medicine And Pharmacology,
Pharmacology And Toxicology
Keywords:
Colorectal cancer; pharmacovigilance; BRAF inhibitors; regorafenib; encorafenib; adverse drug reactions; renal disorders
Online: 28 July 2023 (02:34:59 CEST)
REVIEW
|
doi:10.20944/preprints202305.1084.v1
Subject:
Medicine And Pharmacology,
Medicine And Pharmacology
Keywords:
antibody-drug conjugate; lysosome; cathepsin; legumain; self-immolation; payload release; peptidomimetic; linker
Online: 16 May 2023 (04:51:34 CEST)
REVIEW
|
doi:10.20944/preprints202212.0207.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
Blood-Brain Barrier; Brain Drug Delivery; Carbon Nanomaterials; Cerebral Gliomas; Glioblastoma; Nanoparticles.
Online: 12 December 2022 (14:56:45 CET)
ARTICLE
|
doi:10.20944/preprints202212.0170.v1
Subject:
Medicine And Pharmacology,
Pharmacology And Toxicology
Keywords:
SonoCloud; GL261 mouse model; ultrasound-mediated drug delivery; glioblastoma; immune checkpoint inhibitors
Online: 9 December 2022 (02:59:28 CET)
REVIEW
|
doi:10.20944/preprints202211.0062.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
membrane transporter; SLC; solute carrier; drug design; pharmacokinetics; prodrug; nanoparticle; bile acids
Online: 3 November 2022 (01:09:54 CET)
ARTICLE
|
doi:10.20944/preprints202210.0141.v1
Subject:
Biology And Life Sciences,
Immunology And Microbiology
Keywords:
AtbFinder; antibiotic susceptibility testing; cystic fibrosis; Pseudomonas aeruginosa; multi-drug re-sistant
Online: 11 October 2022 (04:56:32 CEST)
REVIEW
|
doi:10.20944/preprints202208.0230.v1
Subject:
Chemistry And Materials Science,
Theoretical Chemistry
Keywords:
chemoinformatics; compound databases; chemical space; diversity; drug discovery; openscience; pseudo-natural product
Online: 12 August 2022 (08:39:40 CEST)
ARTICLE
|
doi:10.20944/preprints202206.0183.v1
Subject:
Chemistry And Materials Science,
Biomaterials
Keywords:
Biomarkers; Drug Signature Identification; Key pathways; Oral Cancer; Oral Squamous Cell Carcinoma
Online: 13 June 2022 (10:14:58 CEST)
ARTICLE
|
doi:10.20944/preprints202103.0621.v1
Subject:
Medicine And Pharmacology,
Immunology And Allergy
Keywords:
Auger electron; cisplatin; 191Pt; 189Pt; radio-drug; DNA double-strand break; γH2AX
Online: 25 March 2021 (14:30:14 CET)
CASE REPORT
|
doi:10.20944/preprints202103.0054.v1
Subject:
Medicine And Pharmacology,
Immunology And Allergy
Keywords:
DRESS syndrome, Eosinophilia, Adverse drug reaction, HHV-6 reactivation, Bactrim adverse reaction
Online: 2 March 2021 (09:26:48 CET)
ARTICLE
|
doi:10.20944/preprints202012.0513.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
apoferritin nanocarriers; controlled drug delivery; idarubicin; ferritin receptor targeting; folate receptor targeting
Online: 21 December 2020 (11:28:08 CET)
REVIEW
|
doi:10.20944/preprints202012.0242.v1
Subject:
Medicine And Pharmacology,
Immunology And Allergy
Keywords:
COVID-19; SARS-CoV-2; long-haul; inflammation; tissue damage; drug repurposing
Online: 10 December 2020 (09:42:20 CET)
COMMUNICATION
|
doi:10.20944/preprints202011.0441.v1
Subject:
Biology And Life Sciences,
Anatomy And Physiology
Keywords:
Sars-Cov-2; Proteomic,; Ghost proteome,; Alternative proteins,; AltOrf.; interactomic; drug repurposing
Online: 16 November 2020 (17:50:19 CET)
ARTICLE
|
doi:10.20944/preprints202004.0448.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
acetyleugenol; Acacia nilotica; anti-tuberculosis; Serine/Threonine kinases; multi-drug resistant TB
Online: 24 April 2020 (14:12:33 CEST)
ARTICLE
|
doi:10.20944/preprints202003.0393.v1
Subject:
Biology And Life Sciences,
Biophysics
Keywords:
SARS-CoV2; RNA depended RNA polymerase; Valproic acid Co-A; drug repurposing
Online: 26 March 2020 (15:04:22 CET)
ARTICLE
|
doi:10.20944/preprints201810.0381.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
Biginelli reaction; dihydropyrimidin-2-thiones; synthesis, virtual screening, drug design; LaSOM 282
Online: 17 October 2018 (09:34:06 CEST)
ARTICLE
|
doi:10.20944/preprints201712.0024.v1
Subject:
Biology And Life Sciences,
Virology
Keywords:
HIV-1; quasispecies; minority resistance mutations; HAART; drug resistance; undetectable viral load
Online: 4 December 2017 (09:34:16 CET)
ARTICLE
|
doi:10.20944/preprints202105.0480.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
camptothecin; drug distribution; drug-membrane interaction; biophysical profiling; biomimetic models; partition coefficient; ADMET/PK prediction; small and wide-angle X-ray diffraction; fluorescence spectroscopy; human serum albumin (HSA)
Online: 20 May 2021 (10:52:33 CEST)
ARTICLE
|
doi:10.20944/preprints202407.1733.v1
Subject:
Chemistry And Materials Science,
Biomaterials
Keywords:
Berberine hydrochloride; Chitosan/Carboxymethyl-β-Cyclodextrin; Hydrogel formulation; Solubility enhancement; Oral drug delivery.
Online: 22 July 2024 (17:36:55 CEST)
ARTICLE
|
doi:10.20944/preprints202407.0129.v1
Subject:
Medicine And Pharmacology,
Gastroenterology And Hepatology
Keywords:
Atypical antipsychotics (AAPs), secondary drug effects, schizophrenia, liver, mitochondria, oxidative stress (OS), MAPK.
Online: 2 July 2024 (13:23:11 CEST)
ARTICLE
|
doi:10.20944/preprints202406.0953.v1
Subject:
Biology And Life Sciences,
Biophysics
Keywords:
GIBAC; Intermolecular binding affinity (Kd); Structural biophysics; Synthetic data; Drug discovery \& design;
Online: 14 June 2024 (05:04:28 CEST)
ARTICLE
|
doi:10.20944/preprints202406.0085.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
precision medicine; drug response prediction; cell-free mRNA; transcriptomic profiling; gene expression signature
Online: 6 June 2024 (03:09:40 CEST)
ARTICLE
|
doi:10.20944/preprints202403.1579.v2
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
Multiple Drug Resistant breast cancer; Anaphase Promoting Complex; cell culture; PDX mouse model
Online: 28 March 2024 (13:34:15 CET)
ARTICLE
|
doi:10.20944/preprints202403.0717.v1
Subject:
Biology And Life Sciences,
Animal Science, Veterinary Science And Zoology
Keywords:
Lumpy skin disease; DNA polymerase; potential inhibitors; phytocompounds; antiviral drug compounds; molecular docking
Online: 13 March 2024 (07:58:39 CET)
ARTICLE
|
doi:10.20944/preprints202401.1398.v1
Subject:
Medicine And Pharmacology,
Pharmacology And Toxicology
Keywords:
Nosocomial infections; Antibacterial activity; Drug resistance; Clausena anisata; GC-MS analysis; Essential oil
Online: 18 January 2024 (11:05:38 CET)
ARTICLE
|
doi:10.20944/preprints202401.1186.v1
Subject:
Medicine And Pharmacology,
Urology And Nephrology
Keywords:
kidney replacement therapy; medication review; drug-related problems; negative outcomes associated with medication.
Online: 16 January 2024 (13:57:35 CET)
ARTICLE
|
doi:10.20944/preprints202312.0574.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
DOCK program; GOLD program; Grb14; insulin receptor (IR); structure-based drug screening (SBDS)
Online: 8 December 2023 (08:24:15 CET)
ARTICLE
|
doi:10.20944/preprints202311.1460.v1
Subject:
Biology And Life Sciences,
Parasitology
Keywords:
Onchocerciasis; drug discovery; anthelmintics; O. gutturosa; motility and MTT inhibition; FDA approved drugs
Online: 23 November 2023 (09:31:11 CET)
ARTICLE
|
doi:10.20944/preprints202311.0766.v1
Subject:
Medicine And Pharmacology,
Neuroscience And Neurology
Keywords:
Alzheimer's disease; neural networks; Training and learning; early diagnosis; drug discovery; brain diseases
Online: 13 November 2023 (08:41:42 CET)
ARTICLE
|
doi:10.20944/preprints202309.0417.v1
Subject:
Medicine And Pharmacology,
Pharmacology And Toxicology
Keywords:
adenylosuccinic acid; Duchenne muscular dystrophy; myopathy; metabolic disease; skeletal muscle; toxicology; drug development
Online: 7 September 2023 (05:09:43 CEST)
ARTICLE
|
doi:10.20944/preprints202308.1966.v1
Subject:
Chemistry And Materials Science,
Theoretical Chemistry
Keywords:
Drug discovery; computational chemistry; conceptual DFT; marine cyclopeptides; chemical reactivity properties; bioavailability scores
Online: 29 August 2023 (09:36:49 CEST)
ARTICLE
|
doi:10.20944/preprints202308.0533.v1
Subject:
Medicine And Pharmacology,
Pharmacology And Toxicology
Keywords:
therapeutic drug monitoring (TDM); extracorporeal therapies; CKRT; hemoadsorption; cytosorb; antimicrobials; clearance; mass removal
Online: 7 August 2023 (10:46:18 CEST)
ARTICLE
|
doi:10.20944/preprints202307.1535.v1
Subject:
Chemistry And Materials Science,
Analytical Chemistry
Keywords:
Boswellia Serrata extract; layered double hydroxides; composite; drug delivery system; antimicrobial; anti-inflammatory
Online: 24 July 2023 (10:38:38 CEST)
ARTICLE
|
doi:10.20944/preprints202306.1793.v1
Subject:
Computer Science And Mathematics,
Artificial Intelligence And Machine Learning
Keywords:
bioactive compounds; black sea cucumbers; cancer; drug-target interactions; machine learning; molecular docking
Online: 26 June 2023 (10:36:43 CEST)
ARTICLE
|
doi:10.20944/preprints202304.0800.v1
Subject:
Biology And Life Sciences,
Toxicology
Keywords:
Brushtail possum; Trichosurus vulpecula; fertility control; and drug-metabolising enzymes (CYP3A and UGT2B)
Online: 23 April 2023 (13:11:28 CEST)
SHORT NOTE
|
doi:10.20944/preprints202212.0230.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
monoamine oxidase; inhibitors; indole; 1,2,4-oxadiazole; drug research; neuroprotective drugs; Parkinson’s disease; MAO
Online: 13 December 2022 (07:12:01 CET)
ARTICLE
|
doi:10.20944/preprints202210.0302.v1
Subject:
Biology And Life Sciences,
Virology
Keywords:
poxviruses; monkeypox virus; envelope proteins; drug repurposing; bioactive phytochemicals; molecular docking, molecular simulation
Online: 20 October 2022 (09:32:02 CEST)
ARTICLE
|
doi:10.20944/preprints202209.0090.v1
Subject:
Computer Science And Mathematics,
Computational Mathematics
Keywords:
epithelial cell; antibody response; basic reproduction number; transcritical bifurcation; impulsive control; drug holidays
Online: 6 September 2022 (10:25:07 CEST)
ARTICLE
|
doi:10.20944/preprints202208.0317.v1
Subject:
Biology And Life Sciences,
Endocrinology And Metabolism
Keywords:
Cytochrome P450; POR; Congenital adrenal hyperplasia; metabolic disorders; CYP3A4; protein stability; drug metabolism
Online: 17 August 2022 (10:02:51 CEST)
ARTICLE
|
doi:10.20944/preprints202112.0203.v1
Subject:
Biology And Life Sciences,
Virology
Keywords:
enterovirus; antidepressant sertraline; drug repurposing; viral entry; host-cell targets; broad-spectrum antiviral
Online: 13 December 2021 (12:55:13 CET)
ARTICLE
|
doi:10.20944/preprints202105.0158.v1
Subject:
Medicine And Pharmacology,
Immunology And Allergy
Keywords:
Imatinib; NLC; Tween 80; SLS; MTT Assay; Release study; Drug delivery; Breast cancer
Online: 10 May 2021 (10:13:02 CEST)
REVIEW
|
doi:10.20944/preprints202104.0574.v1
Subject:
Chemistry And Materials Science,
Analytical Chemistry
Keywords:
smart materials; drug delivery systems; flame retardant; industrial coatings; filtration membranes; antifouling coatings.
Online: 21 April 2021 (11:47:42 CEST)
REVIEW
Subject:
Chemistry And Materials Science,
Analytical Chemistry
Keywords:
hyperoxaluria; oxalate; inhibitor; small molecule drug; glycolate oxidase; lactate dehydrogenase; liver selective distribution
Online: 31 December 2020 (08:59:47 CET)
ARTICLE
|
doi:10.20944/preprints202012.0588.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
Trazodone; drug design; dissolution; crystal structure; solid-state NMR (SSNMR) spectroscopy; GIPAW calculation
Online: 23 December 2020 (13:42:36 CET)
ARTICLE
|
doi:10.20944/preprints202011.0512.v1
Subject:
Medicine And Pharmacology,
Immunology And Allergy
Keywords:
antimicrobials; meropenem; generic drug; real-life studies; product surveillance, postmarketing; treatment outcome; pharmacovigilance
Online: 19 November 2020 (13:34:26 CET)
ARTICLE
|
doi:10.20944/preprints202011.0292.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
Alzheimer's disease; BACE1; Molecular dynamics; MM/GBSA; Inhibitors; Drug likeness; Ligand efficiency, Kd.
Online: 10 November 2020 (09:10:50 CET)
REVIEW
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
apoptosis; antitumor; antimetastasis; anti-angiogenesis; NK-1 receptor; substance P; drug repositioning; Emend
Online: 31 August 2020 (10:11:13 CEST)
ARTICLE
|
doi:10.20944/preprints202007.0424.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
4-Phenylbutyric acid; Colon-targeted drug delivery; Colitis; Prodrug; ER stress; Chemical chaperone
Online: 19 July 2020 (19:15:20 CEST)
REVIEW
Subject:
Biology And Life Sciences,
Cell And Developmental Biology
Keywords:
nucleoid-associated proteins (NAPs); moonlighting proteins; drug target; biofilm; specificity determination; phylogenetic analysis
Online: 7 June 2020 (09:07:56 CEST)
REVIEW
|
doi:10.20944/preprints202005.0342.v1
Subject:
Medicine And Pharmacology,
Pharmacology And Toxicology
Keywords:
seaweed; metabolites; neuroprotection; Alzheimer’s disease; Parkinson’s disease; ischemic stroke; computer-aided drug discovery
Online: 21 May 2020 (09:49:29 CEST)
REVIEW
|
doi:10.20944/preprints201912.0179.v1
Subject:
Biology And Life Sciences,
Biophysics
Keywords:
globular set; category theory; multidimensional; visual recognition; drug-resistant epilepsy; transcranial magnetic stimulation.
Online: 13 December 2019 (10:37:03 CET)
ARTICLE
|
doi:10.20944/preprints201911.0024.v1
Subject:
Computer Science And Mathematics,
Information Systems
Keywords:
Iranian traditional medicine; Persian medicine; ontology; knowledge-base; Mizaj; temperament; new drug discovery
Online: 3 November 2019 (17:07:50 CET)
ARTICLE
|
doi:10.20944/preprints201908.0253.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
halogen bonding; fluorine; iodine; pentafluorosulfanyl; titration; ab initio calculation; NMR study; drug design
Online: 25 August 2019 (15:41:59 CEST)
ARTICLE
|
doi:10.20944/preprints201803.0144.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
sea anemone; drug discovery; cancer; antiangiogenic; endothelial cells; RGD motif; Kunitz type inhibitor
Online: 19 March 2018 (08:15:38 CET)
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
oleanolic acid derivatives; synthesis; anti-tumor activity; molecular docking; computer-aided drug design
Online: 24 April 2017 (12:08:36 CEST)
CASE REPORT
|
doi:10.20944/preprints202308.1373.v1
Subject:
Medicine And Pharmacology,
Hematology
Keywords:
Large B-cell lymphoma (LBCL); Immunohistochemical (IHC) staining; Glucoseregulated protein 94 (GRP94); CYP3A4; Multidrug resistance protein 1 (MDR1); Aldo-keto reductase family 1 member C3 (AKR1C3); Multi-drug resistance-associated protein 1 (MRP1); P53
Online: 18 August 2023 (11:42:22 CEST)
ARTICLE
|
doi:10.20944/preprints202405.0380.v1
Subject:
Medicine And Pharmacology,
Pharmacy
Keywords:
thiocarbohydrazones; Schiff base; moleculer docking; urease inhibition; pharmacokinetic properties; drug combinations
Online: 8 May 2024 (02:40:50 CEST)
REVIEW
|
doi:10.20944/preprints202404.1839.v1
Subject:
Medicine And Pharmacology,
Cardiac And Cardiovascular Systems
Keywords:
Omega-3 fatty acids; cardiovascular disease; Nanoparticle encapsulation; Metal-organic framework; Drug delivery systems
Online: 28 April 2024 (08:33:48 CEST)
ARTICLE
|
doi:10.20944/preprints202404.1209.v1
Subject:
Biology And Life Sciences,
Immunology And Microbiology
Keywords:
Mycobacterium tuberculosis; Drug Resistance; Whole Genome Sequencing; Genetic Diversity; Brazil; Novel Mutations
Online: 18 April 2024 (07:51:01 CEST)
ARTICLE
|
doi:10.20944/preprints202404.0426.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
CDK8; Cyclin C; Protein-protein interaction; Molecular dynamic simulation; Free energy calculation; Drug design
Online: 5 April 2024 (10:12:16 CEST)
REVIEW
|
doi:10.20944/preprints202403.1716.v1
Subject:
Biology And Life Sciences,
Other
Keywords:
Adjuvant; Archaeal carriers; Lipid-based drug delivery; Vaccine delivery; Gene therapy; Immune modulators; Tocosome
Online: 28 March 2024 (09:47:09 CET)
REVIEW
|
doi:10.20944/preprints202401.0079.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
NF-E2-related factor 2; Drug resistance; Reactive oxygen species; Autophagy; Unfolded protein response
Online: 3 January 2024 (02:26:23 CET)
ARTICLE
|
doi:10.20944/preprints202311.1667.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
α-MSH; melanoma; peptide-drug conjugates; in vitro antiproliferative effect; in vivo antitumor activity
Online: 27 November 2023 (08:49:52 CET)
ARTICLE
|
doi:10.20944/preprints202311.1319.v1
Subject:
Public Health And Healthcare,
Public Health And Health Services
Keywords:
HIV; AIDS; drug use; sexually transmitted diseases; alcohol; female sex workers; FSWs
Online: 21 November 2023 (13:17:51 CET)
COMMUNICATION
|
doi:10.20944/preprints202311.1268.v1
Subject:
Biology And Life Sciences,
Life Sciences
Keywords:
SARS-CoV-2; COVID-19; RdRp; m1A triphosphate; Antiviral Drug
Online: 21 November 2023 (07:19:23 CET)
ARTICLE
|
doi:10.20944/preprints202310.0980.v1
Subject:
Chemistry And Materials Science,
Surfaces, Coatings And Films
Keywords:
microparticles; scalable manufacturing; laser cutting; drug delivery; complex structures; composites; core-shell; defined size
Online: 16 October 2023 (16:53:55 CEST)
ARTICLE
|
doi:10.20944/preprints202309.0069.v1
Subject:
Public Health And Healthcare,
Health Policy And Services
Keywords:
MSM; trends; high-risk sexual behaviors; HIV; sexualized drug use; chemsex; sexually transmitted infections
Online: 4 September 2023 (02:43:27 CEST)
ARTICLE
|
doi:10.20944/preprints202309.0011.v1
Subject:
Medicine And Pharmacology,
Anesthesiology And Pain Medicine
Keywords:
immunoassay; urine drug test; opioid; nonmedical; cancer pain; safety-net hospital; palliative medicine; education
Online: 1 September 2023 (04:02:26 CEST)
REVIEW
|
doi:10.20944/preprints202308.1747.v1
Subject:
Medicine And Pharmacology,
Transplantation
Keywords:
kidney transplantation; immunosuppression; adverse drug event; nephrotoxicity; NODAT; anemia; leukopenia; viral reactivation; hypertension; dyslipidemia
Online: 24 August 2023 (13:34:38 CEST)
ARTICLE
|
doi:10.20944/preprints202308.0468.v1
Subject:
Medicine And Pharmacology,
Pharmacology And Toxicology
Keywords:
dasatinib; imatinib; nilotibin; ponatinib; children; therapeutic drug monitoring; sex and gender pharmacology; personalized medicine.
Online: 7 August 2023 (11:53:12 CEST)
REVIEW
|
doi:10.20944/preprints202308.0109.v1
Subject:
Biology And Life Sciences,
Biology And Biotechnology
Keywords:
preclinical; oncology; 3D culture; organ-on-a-chip; spheroid; organoid; 3D bioprinting; drug screening
Online: 2 August 2023 (02:48:00 CEST)
REVIEW
|
doi:10.20944/preprints202305.0945.v1
Subject:
Medicine And Pharmacology,
Medicine And Pharmacology
Keywords:
Systems Pharmacology; Polypharmacology; Adverse Events; Drug Discovery; Functional genomics; Disease Modeling; Network analysis; Innovation
Online: 12 May 2023 (12:18:59 CEST)
ARTICLE
|
doi:10.20944/preprints202301.0221.v1
Subject:
Computer Science And Mathematics,
Artificial Intelligence And Machine Learning
Keywords:
Ion channels; Membrane proteins; Transmembrane proteins; Drug discovery; Protein language models; Convolutional Neural Network
Online: 12 January 2023 (09:21:08 CET)
REVIEW
|
doi:10.20944/preprints202210.0347.v1
Subject:
Medicine And Pharmacology,
Pharmacology And Toxicology
Keywords:
monkeypox virus; infection; treatment; antiviral; drug; management; public health emergency; tecovirimat; cidofovir; bibliometric analysis
Online: 24 October 2022 (03:38:12 CEST)
REVIEW
|
doi:10.20944/preprints202207.0031.v1
Subject:
Biology And Life Sciences,
Biophysics
Keywords:
Cell-state transitions; Phenotypic plasticity; Cancer Stem Cells; Intratumoral heterogeneity; Lamarckian Induction; Drug resistance
Online: 4 July 2022 (04:56:00 CEST)
ARTICLE
|
doi:10.20944/preprints202201.0082.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
breast cancer; cancer stem cell; therapy resistance; cationic amphiphilic drug; lysosome-dependent cell death
Online: 6 January 2022 (11:51:28 CET)
ARTICLE
|
doi:10.20944/preprints202108.0512.v1
Subject:
Medicine And Pharmacology,
Pharmacy
Keywords:
oyster mushroom (Pleurotus sp.); PARP protein; 4UND protein; molecular docking; PyRx; BIOVIA drug discovery
Online: 26 August 2021 (16:15:06 CEST)
REVIEW
|
doi:10.20944/preprints202107.0650.v1
Subject:
Medicine And Pharmacology,
Immunology And Allergy
Keywords:
chronic disorders; inflammation; human superorganism; holobiont; microbiome; multimorbidity; microimmunosome; polypharmacy; drug safety; sustainable healthcare
Online: 29 July 2021 (11:37:20 CEST)
ARTICLE
|
doi:10.20944/preprints202008.0667.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
Ovarian cancer; drug resistance; apoptosis; proteomics; combination; cytotoxicity; artemisinin; oleanolic acid; platinum drugs; cisplatin
Online: 30 August 2020 (12:06:32 CEST)
ARTICLE
|
doi:10.20944/preprints202004.0369.v2
Subject:
Biology And Life Sciences,
Virology
Keywords:
COVID-19; SARS-CoV-2; spike protein; ACE1; ACE2; host-virus interaction; drug repurposing
Online: 2 August 2020 (09:23:18 CEST)
REVIEW
|
doi:10.20944/preprints202002.0451.v1
Subject:
Medicine And Pharmacology,
Clinical Medicine
Keywords:
systematic review; ADR assessment; elderly; aged-care facilities; medications monitoring; nursing home; drug review
Online: 29 February 2020 (03:41:22 CET)
ARTICLE
|
doi:10.20944/preprints201909.0063.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
FABP4; A-FABP; aP2; antidiabetes; antiobesity; antiatherosclerosis; anticancer; computational tools; computer-aided drug discovery
Online: 5 September 2019 (15:39:58 CEST)
ARTICLE
|
doi:10.20944/preprints201811.0627.v1
Subject:
Chemistry And Materials Science,
Theoretical Chemistry
Keywords:
chemical space; chemical data set; chemoinformatics; consensus diversity plot; drug discovery; molecular diversity; visualization
Online: 30 November 2018 (10:06:15 CET)
ARTICLE
|
doi:10.20944/preprints201804.0374.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
STAT3 as a drug target; cyclic STAT3 decoy; oligodeoxynucleotide inhibitor; head and neck cancer
Online: 29 April 2018 (10:10:00 CEST)
ARTICLE
|
doi:10.20944/preprints201801.0136.v1
Subject:
Chemistry And Materials Science,
Nanotechnology
Keywords:
polymer-drug association; inclusion nano-complex; an amphiphilic polymer; polysoaps; antibiotic resistance; ampicillin trihydrate
Online: 16 January 2018 (07:56:15 CET)
REVIEW
|
doi:10.20944/preprints201705.0129.v1
Subject:
Biology And Life Sciences,
Biophysics
Keywords:
cell fate decision; cancer attractors; gene network dynamics; EMT; drug resistance; intrinsically disordered proteins
Online: 17 May 2017 (06:25:17 CEST)