ARTICLE
|
doi:10.20944/preprints201905.0319.v1
Subject:
Biology And Life Sciences,
Immunology And Microbiology
Keywords:
cyanobacteria; protease inhibitors; digestive enzyme; daphnia; HPLC; UV/Vis
Online: 27 May 2019 (12:56:49 CEST)
ARTICLE
|
doi:10.20944/preprints201905.0046.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
aminopeptidases; inhibitors; aminophosphonate; phenylglycine analogues; fluorine substituted; molecular modeling
Online: 6 May 2019 (10:16:45 CEST)
ARTICLE
|
doi:10.20944/preprints201806.0131.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
histone demethylase inhibitors; DNA damage; epigenetic drugs; breast cancer
Online: 8 June 2018 (12:29:10 CEST)
REVIEW
|
doi:10.20944/preprints202004.0160.v2
Subject:
Biology And Life Sciences,
Virology
Keywords:
COVID-19; ACE; ACE2; Angiotensin II; Bradykinin; RAS inhibitors; ACE inhibitors; AT1 receptor blockers; Losartan; Bradykinin Antagonists; Ang II loading; Giapreza; Icatibant.
Online: 14 April 2020 (14:34:43 CEST)
REVIEW
|
doi:10.20944/preprints202407.0700.v1
Subject:
Medicine And Pharmacology,
Dermatology
Keywords:
treatment; biologics; biological drugs; vitiligo; Janus kinase inhibitors (JAKs); cytokines
Online: 9 July 2024 (07:55:45 CEST)
CASE REPORT
|
doi:10.20944/preprints202406.1688.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
epithelial ovarian cancer; brain metastases; PARP inhibitors; multimodal patient journey.
Online: 24 June 2024 (12:40:16 CEST)
ARTICLE
|
doi:10.20944/preprints202406.1311.v1
Subject:
Biology And Life Sciences,
Virology
Keywords:
Coronavirus; SARS-CoV-2; MERS-CoV; 3CLPro; antivirals; protease inhibitors
Online: 19 June 2024 (05:53:52 CEST)
REVIEW
|
doi:10.20944/preprints202404.0176.v1
Subject:
Biology And Life Sciences,
Biophysics
Keywords:
histone deacetylase inhibitors; radiosensitisation; heterochromatin; double strand break; DNA repair
Online: 2 April 2024 (10:09:33 CEST)
REVIEW
|
doi:10.20944/preprints202403.1203.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
rectal cancer; total neoadjuvant treatment; immunocheckpoint inhibitors; nonoperative management; ctDNA.
Online: 20 March 2024 (16:08:21 CET)
BRIEF REPORT
|
doi:10.20944/preprints202403.0928.v1
Subject:
Medicine And Pharmacology,
Immunology And Allergy
Keywords:
systemic sclerosis; pulmonary hypertension; Phosphodiesterase-5 inhibitors; endothelin receptor antagonist
Online: 15 March 2024 (13:15:50 CET)
REVIEW
|
doi:10.20944/preprints202402.1496.v1
Subject:
Medicine And Pharmacology,
Pharmacy
Keywords:
Proton-pump inhibitors; eosinophilic esophagitis; pharmacogenetics; CYP219 gene; STAT6 gene.
Online: 26 February 2024 (23:53:49 CET)
ARTICLE
|
doi:10.20944/preprints202402.0449.v1
Subject:
Medicine And Pharmacology,
Internal Medicine
Keywords:
herpes zoster; immune checkpoint inhibitors; standardized incidence ratio; cancer patients
Online: 7 February 2024 (14:34:28 CET)
ARTICLE
|
doi:10.20944/preprints202311.1938.v1
Subject:
Medicine And Pharmacology,
Pharmacology And Toxicology
Keywords:
drug-induced allergy; anaphylaxis; antibiotics; local anesthetics; cyclooxygenase (COX)-inhibitors
Online: 30 November 2023 (04:21:45 CET)
ARTICLE
|
doi:10.20944/preprints202307.1694.v1
Subject:
Medicine And Pharmacology,
Internal Medicine
Keywords:
Idiopathic Pulmonary Fibrosis; Lung Neoplasms; Hydroxymethylglutaryl-CoA Reductase Inhibitors; Database
Online: 25 July 2023 (10:01:14 CEST)
REVIEW
|
doi:10.20944/preprints202306.0143.v1
Subject:
Medicine And Pharmacology,
Immunology And Allergy
Keywords:
Systemic sclerosis; treatment; Janus kinase inhibitors; fibrosis; anti-cytokine treatment
Online: 2 June 2023 (07:07:00 CEST)
ARTICLE
|
doi:10.20944/preprints202305.1103.v1
Subject:
Engineering,
Bioengineering
Keywords:
mutate HIV protease inhibitors; carboxamides; heteroarenes; mammalian cells essay; ADME
Online: 16 May 2023 (05:32:28 CEST)
REVIEW
|
doi:10.20944/preprints202304.0564.v1
Subject:
Medicine And Pharmacology,
Psychiatry And Mental Health
Keywords:
serotonin antagonist/reuptake inhibitors; comorbidity; psychiatric disorders; trazodone; neurobiology; emotion
Online: 19 April 2023 (07:52:17 CEST)
ARTICLE
|
doi:10.20944/preprints202304.0327.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
Ovarian cancer; PARP inhibitors; epithelial to mesenchymal transition; drug response
Online: 13 April 2023 (14:30:07 CEST)
ARTICLE
|
doi:10.20944/preprints202203.0405.v1
Subject:
Biology And Life Sciences,
Immunology And Microbiology
Keywords:
α-amylase inhibitors; diabetes; hemi-pyocyanin; marine discards; microbial conversion
Online: 31 March 2022 (10:47:24 CEST)
REVIEW
|
doi:10.20944/preprints202111.0087.v1
Subject:
Biology And Life Sciences,
Virology
Keywords:
virome; microbiota; cancer; bacteriophages; fecal microbiota transplantation; checkpoint inhibitors; immunotherapy
Online: 3 November 2021 (14:30:14 CET)
ARTICLE
|
doi:10.20944/preprints202104.0174.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
Phosphodiesterase (PDE); natural products; inhibitors; Protein Kinase; selectivity; fluorescence polarization
Online: 6 April 2021 (12:07:58 CEST)
REVIEW
|
doi:10.20944/preprints202010.0338.v1
Subject:
Medicine And Pharmacology,
Immunology And Allergy
Keywords:
Urothelial carcinoma; immune checkpoint inhibitors; immunotherapy; tumor microenvironment; metabolic pathway
Online: 16 October 2020 (08:00:41 CEST)
ARTICLE
|
doi:10.20944/preprints202005.0016.v1
Subject:
Medicine And Pharmacology,
Epidemiology And Infectious Diseases
Keywords:
COVID-19; elderly; proton pump inhibitors; antipsychotics; metformin; oral antidiabetics
Online: 2 May 2020 (15:48:33 CEST)
REVIEW
|
doi:10.20944/preprints202004.0331.v1
Subject:
Medicine And Pharmacology,
Epidemiology And Infectious Diseases
Keywords:
COVID-19; associated comorbidities; treatment; ACE2 inhibitors; Type 2 diabetes
Online: 19 April 2020 (05:42:22 CEST)
ARTICLE
|
doi:10.20944/preprints202004.0003.v2
Subject:
Biology And Life Sciences,
Virology
Keywords:
SARS-CoV-2; protease; virtual screening; pharmacophore; inhibitors; natural compounds
Online: 17 April 2020 (11:00:55 CEST)
ARTICLE
|
doi:10.20944/preprints201811.0221.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
Fatty Acid Amide Hydrolase; cannabinoid; carboxamide inhibitors; 3D-QSAR; CoMSIA.
Online: 8 November 2018 (14:52:23 CET)
REVIEW
|
doi:10.20944/preprints202302.0030.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
angiogenesis inhibitors; VEGF inhibitors; ovarian cancer; progression-free survival; overall sur-vival; toxicity; systematic review; meta-analysis; randomized controlled trials; FDA approval of cancer drugs
Online: 2 February 2023 (05:26:47 CET)
ARTICLE
|
doi:10.20944/preprints202404.1746.v1
Subject:
Biology And Life Sciences,
Life Sciences
Keywords:
Retinoblastoma; Epigenetic Reprogramming; Cancer Therapy; Epigenetic Therapy; DNA methyltransferase (DNMT) inhibitors
Online: 26 April 2024 (12:19:15 CEST)
REVIEW
|
doi:10.20944/preprints202401.0407.v1
Subject:
Medicine And Pharmacology,
Urology And Nephrology
Keywords:
prostatic neoplasm; biochemical recurrence; androgen receptor signaling inhibitors; androgen deprivation therapy
Online: 4 January 2024 (11:22:30 CET)
SHORT NOTE
|
doi:10.20944/preprints202312.0899.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
monoamine oxidase; inhibitors; 1,3-oxazole; benzenesulfonamide; drug research; Parkinson’s disease; MAO
Online: 12 December 2023 (14:22:48 CET)
REVIEW
|
doi:10.20944/preprints202311.0295.v1
Subject:
Medicine And Pharmacology,
Cardiac And Cardiovascular Systems
Keywords:
Atrial fibrillation, SGLT2 inhibitors, cardiovascular outcomes, hemodynamic effects, AF risk reduction
Online: 6 November 2023 (08:13:49 CET)
REVIEW
|
doi:10.20944/preprints202310.1318.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
advanced melanoma; immunotherapy; target therapy; lysine histone methyl transferase inhibitors; UNC0642
Online: 20 October 2023 (08:35:45 CEST)
REVIEW
|
doi:10.20944/preprints202305.0751.v1
Subject:
Medicine And Pharmacology,
Medicine And Pharmacology
Keywords:
Skin pigmentation; melanin; Tyrosinase inhibitors; hypopigmentation; hyperpigmentation; Vitiligo; skin-lightening; Depigmentation
Online: 10 May 2023 (11:32:48 CEST)
REVIEW
|
doi:10.20944/preprints202304.1236.v1
Subject:
Medicine And Pharmacology,
Hematology
Keywords:
FLT3 mutations; resistant/relapsed acute myeloid leukemia; tyrosine kinase inhibitors; gilteritinib
Online: 29 April 2023 (10:55:21 CEST)
REVIEW
|
doi:10.20944/preprints202302.0205.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
breast cancer; ovarian cancer; PARP inhibitors; Alu repeats; protein-protein interactions
Online: 13 February 2023 (07:54:35 CET)
ARTICLE
|
doi:10.20944/preprints202301.0325.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
Immune checkpoint inhibitors; Anti-tumor immunity; Predictive biomarker; Malignant melanoma; NSCLC
Online: 18 January 2023 (08:39:18 CET)
REVIEW
|
doi:10.20944/preprints202201.0468.v1
Subject:
Biology And Life Sciences,
Virology
Keywords:
Flavivirus; NS2B-NS3; ZIKA Virus; Dengue Virus; West Nile Virus; Inhibitors
Online: 31 January 2022 (13:46:44 CET)
ARTICLE
|
doi:10.20944/preprints202106.0565.v1
Subject:
Biology And Life Sciences,
Virology
Keywords:
HIV-1 transcription; HIV-1 Tat; TAR RNA; small molecule inhibitors
Online: 23 June 2021 (11:04:21 CEST)
ARTICLE
|
doi:10.20944/preprints202105.0772.v1
Subject:
Medicine And Pharmacology,
Immunology And Allergy
Keywords:
Immune checkpoint inhibitors; immune-related endocrine dysfunction; hypothyroidism; targeted therapy; malignancy
Online: 31 May 2021 (12:49:40 CEST)
REVIEW
|
doi:10.20944/preprints202102.0150.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
CTLA-4; Treg cells: Immune checkpoint inhibitors; CD28; Antigen Presenting Cells
Online: 5 February 2021 (09:35:47 CET)
REVIEW
|
doi:10.20944/preprints202012.0343.v1
Subject:
Medicine And Pharmacology,
Immunology And Allergy
Keywords:
COVID-19; platelet activating factor; thrombosis; inflammation; Mediterranean diet; PAF-inhibitors
Online: 14 December 2020 (14:16:37 CET)
REVIEW
|
doi:10.20944/preprints202003.0378.v1
Subject:
Medicine And Pharmacology,
Epidemiology And Infectious Diseases
Keywords:
China's COVID-19 Guide; Remdesivir; Xuebijing; Hydroxychloroquine; IL6 inhibitors; COVID-19
Online: 26 March 2020 (01:48:42 CET)
ARTICLE
|
doi:10.20944/preprints201810.0133.v2
Subject:
Biology And Life Sciences,
Immunology And Microbiology
Keywords:
aging; angiotensin-converting enzyme inhibitors; nutrient metabolism; genetic background; nutritional stress
Online: 29 October 2018 (10:33:59 CET)
ARTICLE
|
doi:10.20944/preprints201706.0022.v1
Subject:
Chemistry And Materials Science,
Theoretical Chemistry
Keywords:
HPPD inhibitors; pharmacophore model; molecule docking; HipHop model; virtual screening; ChemDiv
Online: 5 June 2017 (05:16:39 CEST)
REVIEW
|
doi:10.20944/preprints202311.0529.v1
Subject:
Public Health And Healthcare,
Primary Health Care
Keywords:
SARS-CoV-2; Papain-like protease; COVID-19; Molecular modelling; Molecular dynamics simulations; Drug discovery; Antiviral drugs; Inhibitors; Therapeutic agents; therapeutic targets; Irreversible inhibitors; Repurposing drugs
Online: 8 November 2023 (16:11:55 CET)
ARTICLE
|
doi:10.20944/preprints202407.0117.v1
Subject:
Biology And Life Sciences,
Immunology And Microbiology
Keywords:
Acral, mucosal, anti-PD-1 Abs, BRAF plus MEK inhibitors, adjuvant therapy
Online: 2 July 2024 (10:51:38 CEST)
REVIEW
|
doi:10.20944/preprints202407.0073.v1
Subject:
Chemistry And Materials Science,
Polymers And Plastics
Keywords:
Natural gas hydrates; Kinetic inhibitors; Research history; Structure composition; Mechanisms of inhibition
Online: 1 July 2024 (15:03:18 CEST)
ARTICLE
|
doi:10.20944/preprints202406.0034.v1
Subject:
Biology And Life Sciences,
Neuroscience And Neurology
Keywords:
voltage-gated sodium channels; fibroblast growth factors; split luciferase assay; kinase inhibitors
Online: 3 June 2024 (08:07:35 CEST)
CASE REPORT
|
doi:10.20944/preprints202402.0658.v3
Subject:
Medicine And Pharmacology,
Medicine And Pharmacology
Keywords:
pharmacokinetic-pharmacodynamic interactions; low-dose methotrexate; proton pump inhibitors; analgesics; pancytopenia; hepatotoxicity
Online: 1 April 2024 (11:53:15 CEST)
ARTICLE
|
doi:10.20944/preprints202404.0043.v1
Subject:
Medicine And Pharmacology,
Obstetrics And Gynaecology
Keywords:
KELIM score; Homologous recombination deficiency (HRD); Poly (ADP-ribose) polymerase inhibitors (PARPi).
Online: 1 April 2024 (11:12:26 CEST)
ARTICLE
|
doi:10.20944/preprints202402.1288.v2
Subject:
Medicine And Pharmacology,
Endocrinology And Metabolism
Keywords:
SGLT2 Inhibitors; Empagliflozin; Renal fibrosis; Connective tissue growth factor; Epithelial-mesenchymal transition
Online: 23 February 2024 (13:25:01 CET)
REVIEW
|
doi:10.20944/preprints202401.2222.v1
Subject:
Medicine And Pharmacology,
Pediatrics, Perinatology And Child Health
Keywords:
gastroesophageal reflux disease; efficacy; safety; proton-pump inhibitors; pediatric patients; systematic review
Online: 31 January 2024 (14:59:40 CET)
REVIEW
|
doi:10.20944/preprints202401.0310.v1
Subject:
Medicine And Pharmacology,
Dentistry And Oral Surgery
Keywords:
inflammation; inflammasome; inhibitors of the inflammasome; nanomaterials; functionalized biomaterials; periodontitis; general pathology
Online: 4 January 2024 (09:25:17 CET)
ARTICLE
|
doi:10.20944/preprints202310.1726.v1
Subject:
Medicine And Pharmacology,
Medicine And Pharmacology
Keywords:
dacomitinib; EGFR inhibitor; overall survival; pharmacokinetics; progression-free survival; proton pump inhibitors
Online: 27 October 2023 (07:06:07 CEST)
HYPOTHESIS
|
doi:10.20944/preprints202309.0196.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
Neurodegenerative disorders; schizophremia; PDK1 inhibitors; Lipid replacement therapy; Aryl hydrocarbon receptor antagonists
Online: 4 September 2023 (14:29:13 CEST)
ARTICLE
|
doi:10.20944/preprints202308.0458.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
polyamine analogs; monoamine oxidases; antiproliferative activity; inhibitors; docking studies; LN-229 cells
Online: 7 August 2023 (11:57:36 CEST)
REVIEW
|
doi:10.20944/preprints202308.0055.v1
Subject:
Medicine And Pharmacology,
Medicine And Pharmacology
Keywords:
COVID-19; SARS-CoV-2 Mpro; protease inhibitors; coronavirus; peptidomimetics; Paxlovid; Nirmatrelvir
Online: 2 August 2023 (05:25:21 CEST)
ARTICLE
|
doi:10.20944/preprints202307.1905.v1
Subject:
Medicine And Pharmacology,
Pharmacology And Toxicology
Keywords:
Colorectal cancer; pharmacovigilance; BRAF inhibitors; regorafenib; encorafenib; adverse drug reactions; renal disorders
Online: 28 July 2023 (02:34:59 CEST)
CASE REPORT
|
doi:10.20944/preprints202307.0971.v1
Subject:
Medicine And Pharmacology,
Dermatology
Keywords:
atopic dermatitis; emollient plus cream; topical corticosteroids; topical calcineurin inhibitors; case report
Online: 14 July 2023 (09:18:55 CEST)
REVIEW
|
doi:10.20944/preprints202307.0979.v1
Subject:
Biology And Life Sciences,
Immunology And Microbiology
Keywords:
breast cancer; microbiota; estrobolome; β-glucuronidase; dysbiosis; inhibitors; metabolomics; personalized medicine; review
Online: 14 July 2023 (07:08:34 CEST)
REVIEW
|
doi:10.20944/preprints202306.1788.v1
Subject:
Medicine And Pharmacology,
Medicine And Pharmacology
Keywords:
Meningioma; Cabozantinib; VEGF; Targeted treatment Cabozantinib; METs; VEGFR2; Inhibitors; Angiogen-esis; Oncology
Online: 26 June 2023 (10:57:00 CEST)
ARTICLE
|
doi:10.20944/preprints202305.0742.v1
Subject:
Medicine And Pharmacology,
Urology And Nephrology
Keywords:
renal lithiasis; phytate; lower inositol phosphates; crystallization inhibitors; calcium oxalate; calcium phosphates
Online: 10 May 2023 (10:45:26 CEST)
REVIEW
|
doi:10.20944/preprints202305.0041.v1
Subject:
Biology And Life Sciences,
Endocrinology And Metabolism
Keywords:
endothelial dysfunction; chronic kidney disease; heart failure; sodium-glucose cotransporter 2 inhibitors
Online: 2 May 2023 (02:18:51 CEST)
ARTICLE
|
doi:10.20944/preprints202304.0530.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
Poly (ADP-Ribose) Polymerase-1; PARP inhibitors; neoplasm; cancer; animal disease models
Online: 19 April 2023 (03:30:59 CEST)
REVIEW
|
doi:10.20944/preprints202302.0380.v1
Subject:
Medicine And Pharmacology,
Psychiatry And Mental Health
Keywords:
serotonin antagonist/reuptake inhibitors; comorbidity; psychiatric disorders; neurological disorders; dementia; primary care
Online: 22 February 2023 (08:42:51 CET)
ARTICLE
|
doi:10.20944/preprints202212.0170.v1
Subject:
Medicine And Pharmacology,
Pharmacology And Toxicology
Keywords:
SonoCloud; GL261 mouse model; ultrasound-mediated drug delivery; glioblastoma; immune checkpoint inhibitors
Online: 9 December 2022 (02:59:28 CET)
REVIEW
|
doi:10.20944/preprints202212.0026.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
Advanced Hepatocellular carcinoma; Immune checkpoint inhibitors; Low middle-income countries; Financial Toxicity
Online: 1 December 2022 (10:33:14 CET)
ARTICLE
|
doi:10.20944/preprints202205.0142.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
glioblastoma; immunotherapy; radiotherapy; brain cancers; radioimmunotherapy; immune checkpoint inhibitors; temozolomide; durvalumab; immunoradiotherapy.
Online: 10 May 2022 (13:22:16 CEST)
REVIEW
|
doi:10.20944/preprints202110.0298.v1
Subject:
Medicine And Pharmacology,
Orthopedics And Sports Medicine
Keywords:
Osteoarthritis; LithoLexal; Lithothamnion; Disease-modifying adjunctive therapy; Anti-inflammatory agents; Cytokine inhibitors
Online: 20 October 2021 (22:49:47 CEST)
REVIEW
|
doi:10.20944/preprints202108.0037.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
ovarian cancer; checkpoint inhibitors; ICIs; immunotherapy; PARP; avelumab; pembrolizumab; nivolumab; bevacizumab; platinum
Online: 2 August 2021 (13:01:35 CEST)
ARTICLE
|
doi:10.20944/preprints202011.0395.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
TNBC; Ca2+-ATPase; SICE; HDAC inhibitors; EMT; WNT signaling; vorinostat; romidepsin; vimentin
Online: 13 November 2020 (20:50:48 CET)
ARTICLE
|
doi:10.20944/preprints202007.0221.v1
Subject:
Chemistry And Materials Science,
Food Chemistry
Keywords:
hCA IX and XII; dual inhibitors; molecular modeling studies; in vitro assays
Online: 11 July 2020 (02:30:03 CEST)
REVIEW
|
doi:10.20944/preprints201909.0140.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
hepatocellular carcinoma; immune checkpoint inhibitors; HCC; pembrolizumab; nivolumab; immune microenvironment; targeted therapies
Online: 14 September 2019 (18:37:29 CEST)
REVIEW
|
doi:10.20944/preprints202406.0880.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
Dendritic cells; DC based cancer vaccine; Immune checkpoint inhibitors; Cancer Therapy; Combinatorial therapy
Online: 13 June 2024 (11:51:42 CEST)
REVIEW
|
doi:10.20944/preprints202406.0356.v1
Subject:
Medicine And Pharmacology,
Gastroenterology And Hepatology
Keywords:
liver transplantation; hepatocellular carcinoma; Immune checkpoint inhibitors; allograft rejection
Online: 6 June 2024 (07:45:00 CEST)
ARTICLE
|
doi:10.20944/preprints202405.1174.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
Gastric cancer; Proto-Oncogene Protein c-met; Tyrosine Kinase Inhibitors; Cell Line; Tumor
Online: 17 May 2024 (12:28:09 CEST)
REVIEW
|
doi:10.20944/preprints202403.0902.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
NSCLC; lung cancer; gut microbiota; immunotherapy; immune checkpoint inhibitors
Online: 15 March 2024 (07:33:31 CET)
ARTICLE
|
doi:10.20944/preprints202403.0717.v1
Subject:
Biology And Life Sciences,
Animal Science, Veterinary Science And Zoology
Keywords:
Lumpy skin disease; DNA polymerase; potential inhibitors; phytocompounds; antiviral drug compounds; molecular docking
Online: 13 March 2024 (07:58:39 CET)
ARTICLE
|
doi:10.20944/preprints202310.0751.v1
Subject:
Biology And Life Sciences,
Cell And Developmental Biology
Keywords:
Drosophila; male meiosis; cyclin B; Cyclin-dependent kinase 1; Cyclin-dependent kinase inhibitors
Online: 12 October 2023 (05:32:28 CEST)
ARTICLE
|
doi:10.20944/preprints202307.1154.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
Uterine fibroids; BRD9 inhibitors; Cell proliferation; Extracellular Matrix; Transcriptome; Epigenome; m6A regulators; Epitranscriptome
Online: 18 July 2023 (04:30:08 CEST)
ARTICLE
|
doi:10.20944/preprints202307.0161.v1
Subject:
Biology And Life Sciences,
Immunology And Microbiology
Keywords:
Non-small cell lung cancer; Targeted Gene Therapy; Immune Checkpoint Inhibitors; Machine Learning
Online: 4 July 2023 (07:57:03 CEST)
SHORT NOTE
|
doi:10.20944/preprints202212.0230.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
monoamine oxidase; inhibitors; indole; 1,2,4-oxadiazole; drug research; neuroprotective drugs; Parkinson’s disease; MAO
Online: 13 December 2022 (07:12:01 CET)
CASE REPORT
|
doi:10.20944/preprints202201.0298.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
Checkpoint inhibitors; Immune related adverse events; Cholestasis; Severe ductopenia; Vanishing bile duct syndrome
Online: 20 January 2022 (11:07:21 CET)
ARTICLE
|
doi:10.20944/preprints202109.0375.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
HIV-protease inhibitors; pseudo-symmetric core; heteroaryl carboxyamides; synthesis; biological screening; molecular modeling
Online: 22 September 2021 (10:44:16 CEST)
REVIEW
|
doi:10.20944/preprints202105.0430.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
ethylene biosynthesis; ethylene inhibitors; in vitro culture; plant hormones; S-adenosylmethionine; stress responses
Online: 19 May 2021 (07:50:29 CEST)
ARTICLE
|
doi:10.20944/preprints202011.0292.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
Alzheimer's disease; BACE1; Molecular dynamics; MM/GBSA; Inhibitors; Drug likeness; Ligand efficiency, Kd.
Online: 10 November 2020 (09:10:50 CET)
ARTICLE
|
doi:10.20944/preprints202010.0032.v1
Subject:
Chemistry And Materials Science,
Biomaterials
Keywords:
Nanomedicine; human ferritin; gastrointestinal tumors; non-camptothecin topoisomerase I inhibitors; drug-delivery; CD71
Online: 2 October 2020 (09:21:53 CEST)
ARTICLE
|
doi:10.20944/preprints202004.0439.v1
Subject:
Biology And Life Sciences,
Biophysics
Keywords:
SARS-CoV-2; COVID-19; spike glycoprotein; variability; molecular docking; molecular dynamics; inhibitors
Online: 24 April 2020 (11:42:01 CEST)
REVIEW
|
doi:10.20944/preprints201910.0255.v1
Subject:
Biology And Life Sciences,
Immunology And Microbiology
Keywords:
antimicrobial resistance; biofilm; efflux pump inhibitors; antibiotic potentiation; eskapee pathogens; gram-negative bacteria
Online: 22 October 2019 (10:22:56 CEST)
ARTICLE
|
doi:10.20944/preprints201812.0362.v1
Subject:
Biology And Life Sciences,
Immunology And Microbiology
Keywords:
Antibiotic resistance, efflux pump inhibitors, Escherichia coli, efflux pumps, multidrug resistance, Staphylococcus aureus
Online: 31 December 2018 (09:55:32 CET)
ARTICLE
|
doi:10.20944/preprints202403.1433.v1
Subject:
Computer Science And Mathematics,
Artificial Intelligence And Machine Learning
Keywords:
FLT3 Inhibitors; Ligand-based Drug Design; Computer-Aided Drug Design; QSAR Modeling; AML Treatment
Online: 25 March 2024 (08:47:40 CET)
ARTICLE
|
doi:10.20944/preprints202401.0661.v1
Subject:
Medicine And Pharmacology,
Pharmacology And Toxicology
Keywords:
Protozoan diseases; Drug repurposing; Cytotoxicity; Dihydrofolate reductase inhibitors; Potassium (K+) channel blocker; ADME properties
Online: 9 January 2024 (10:30:36 CET)
REVIEW
|
doi:10.20944/preprints202311.1632.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
checkpoint inhibitors; esophageal cancer; gastric cancer; immunotherapy; PD-L1; HER2; clinical trials; history; disparities
Online: 28 November 2023 (01:45:08 CET)
REVIEW
|
doi:10.20944/preprints202309.1061.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
prodrugs; HIV; AIDS; Nucleoside Reverse Transcriptase Inhibitors (NRTI); co-drugs; new drugs; medicinal chemistry
Online: 18 September 2023 (05:47:07 CEST)
REVIEW
|
doi:10.20944/preprints202308.0688.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
Urothelial cell cancer; metastasis, drug resistance, immunotherapy; immune checkpoint inhibitors; tumorigenesis; antibody–drug conjugate.
Online: 9 August 2023 (08:23:29 CEST)
REVIEW
|
doi:10.20944/preprints202306.0994.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
hepatocellular carcinoma (HCC); LOXL2; tumor microenvironment (TME); extracellular matrix (ECM); LOXL2 inhibitors; target therapy
Online: 14 June 2023 (07:18:34 CEST)
ARTICLE
|
doi:10.20944/preprints202305.2226.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
melanoma; cutaneous melanoma; mucosal melanoma; uveal melanoma; immune-checkpoint inhibitors; metabolomics; tryptophan; kynurenine; spermine
Online: 31 May 2023 (10:45:46 CEST)
HYPOTHESIS
|
doi:10.20944/preprints202305.1129.v1
Subject:
Biology And Life Sciences,
Anatomy And Physiology
Keywords:
Lymphangiontrope; salt sensitivity; cardiorenal syndrome; SGLT2 inhibitors; Down’s syndrome; depression; schizophrenia; C Reactive Protein
Online: 16 May 2023 (08:51:13 CEST)
REVIEW
|
doi:10.20944/preprints202304.0516.v1
Subject:
Medicine And Pharmacology,
Internal Medicine
Keywords:
SGLT-2 Inhibitors; Inflammasome; NLRP3; reno-protective effects; Cardio-protective effects; neuro-protective effects.
Online: 18 April 2023 (10:33:39 CEST)
ARTICLE
|
doi:10.20944/preprints202211.0516.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
Antivirals; coronavirus; COVID-19; covalent drugs; dynamic light scattering; inhibitors; main protease; natural products
Online: 28 November 2022 (13:40:01 CET)