REVIEW
|
doi:10.20944/preprints202307.0013.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
prostate cancer; PARP inhibitors; DDR gene; CRPC
Online: 3 July 2023 (08:22:22 CEST)
CASE REPORT
|
doi:10.20944/preprints202406.1688.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
epithelial ovarian cancer; brain metastases; PARP inhibitors; multimodal patient journey.
Online: 24 June 2024 (12:40:16 CEST)
ARTICLE
|
doi:10.20944/preprints202403.0717.v1
Subject:
Biology And Life Sciences,
Animal Science, Veterinary Science And Zoology
Keywords:
Lumpy skin disease; DNA polymerase; potential inhibitors; phytocompounds; antiviral drug compounds; molecular docking
Online: 13 March 2024 (07:58:39 CET)
REVIEW
|
doi:10.20944/preprints202304.0736.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
advanced breast cancer; germline BRCA1/2 mutations; pathogenic/likely pathogenic variants; CDK4/6 inhibitors; Pi3Ka inhibitors; HER2-low
Online: 23 April 2023 (03:12:48 CEST)
ARTICLE
|
doi:10.20944/preprints202102.0525.v1
Subject:
Chemistry And Materials Science,
Analytical Chemistry
Keywords:
HIV-RT; ribonuclease H; dual inhibitors; docking; putative binding
Online: 23 February 2021 (15:51:40 CET)
ARTICLE
|
doi:10.20944/preprints202407.0532.v1
Subject:
Medicine And Pharmacology,
Veterinary Medicine
Keywords:
FIP; Vitamin E; inhibitors; drug discovery
Online: 8 July 2024 (03:25:35 CEST)
REVIEW
|
doi:10.20944/preprints202407.1976.v1
Subject:
Medicine And Pharmacology,
Urology And Nephrology
Keywords:
erectile dysfunction; phosphodiesterase-5 inhibitors; sildenafil
Online: 24 July 2024 (14:17:23 CEST)
REVIEW
|
doi:10.20944/preprints202408.0330.v1
Subject:
Chemistry And Materials Science,
Physical Chemistry
Keywords:
self-healing; coatings; capsules; corrosion; inhibitors
Online: 6 August 2024 (12:22:47 CEST)
ARTICLE
|
doi:10.20944/preprints201611.0023.v1
Subject:
Biology And Life Sciences,
Immunology And Microbiology
Keywords:
anti-yeast; enzyme inhibitors; Terminalia mantaly; Combretaceae
Online: 3 November 2016 (09:35:17 CET)
REVIEW
|
doi:10.20944/preprints202405.0212.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
Hepatocellular carcinoma (HCC); systemic therapies; bridging; liver transplantation (LT); Tyrosine Kinase Inhibitors (TKIs); Immune Checkpoint Inhibitors (ICIs)
Online: 6 May 2024 (04:52:05 CEST)
ARTICLE
|
doi:10.20944/preprints202407.1061.v1
Subject:
Biology And Life Sciences,
Life Sciences
Keywords:
Deep learning; immune checkpoint inhibitors; Global self-attention mechanism
Online: 13 July 2024 (00:00:37 CEST)
REVIEW
|
doi:10.20944/preprints202402.0872.v1
Subject:
Biology And Life Sciences,
Life Sciences
Keywords:
Immunotherapy; Immune checkpoint inhibitors; Rechallenge therapy; Resistance; NSCLC
Online: 16 February 2024 (11:34:11 CET)
BRIEF REPORT
|
doi:10.20944/preprints202403.0928.v1
Subject:
Medicine And Pharmacology,
Immunology And Allergy
Keywords:
systemic sclerosis; pulmonary hypertension; Phosphodiesterase-5 inhibitors; endothelin receptor antagonist
Online: 15 March 2024 (13:15:50 CET)
REVIEW
|
doi:10.20944/preprints202405.1983.v1
Subject:
Medicine And Pharmacology,
Medicine And Pharmacology
Keywords:
MAFLD; THR-β Agonists; FGF-21 Agonists; SGLT2 Inhibitors
Online: 30 May 2024 (09:26:47 CEST)
REVIEW
|
doi:10.20944/preprints202407.1686.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
Melanoma; Immune checkpoint inhibitors; lymphoid subsets; biomarker; predictive biomarker; prognostic biomarker
Online: 22 July 2024 (09:53:07 CEST)
REVIEW
|
doi:10.20944/preprints202407.0700.v1
Subject:
Medicine And Pharmacology,
Dermatology
Keywords:
treatment; biologics; biological drugs; vitiligo; Janus kinase inhibitors (JAKs); cytokines
Online: 9 July 2024 (07:55:45 CEST)
REVIEW
|
doi:10.20944/preprints202309.0120.v1
Subject:
Biology And Life Sciences,
Cell And Developmental Biology
Keywords:
Melanoma; BRAF mutations; BRAF inhibitors; MEK inhibitors; Immunotherapy
Online: 4 September 2023 (15:46:20 CEST)
ARTICLE
|
doi:10.20944/preprints202404.0043.v1
Subject:
Medicine And Pharmacology,
Obstetrics And Gynaecology
Keywords:
KELIM score; Homologous recombination deficiency (HRD); Poly (ADP-ribose) polymerase inhibitors (PARPi).
Online: 1 April 2024 (11:12:26 CEST)
REVIEW
|
doi:10.20944/preprints202402.1496.v1
Subject:
Medicine And Pharmacology,
Pharmacy
Keywords:
Proton-pump inhibitors; eosinophilic esophagitis; pharmacogenetics; CYP219 gene; STAT6 gene.
Online: 26 February 2024 (23:53:49 CET)
ARTICLE
|
doi:10.20944/preprints202402.1288.v2
Subject:
Medicine And Pharmacology,
Endocrinology And Metabolism
Keywords:
SGLT2 Inhibitors; Empagliflozin; Renal fibrosis; Connective tissue growth factor; Epithelial-mesenchymal transition
Online: 23 February 2024 (13:25:01 CET)
REVIEW
|
doi:10.20944/preprints202404.0176.v1
Subject:
Biology And Life Sciences,
Biophysics
Keywords:
histone deacetylase inhibitors; radiosensitisation; heterochromatin; double strand break; DNA repair
Online: 2 April 2024 (10:09:33 CEST)
REVIEW
|
doi:10.20944/preprints201903.0288.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
Enhancers; BET inhibitors; CDK7 inhibitors; HDAC inhibitors; Transcription factors; eRNAs; cancer
Online: 30 March 2019 (08:33:07 CET)
ARTICLE
|
doi:10.20944/preprints202406.0034.v1
Subject:
Biology And Life Sciences,
Neuroscience And Neurology
Keywords:
voltage-gated sodium channels; fibroblast growth factors; split luciferase assay; kinase inhibitors
Online: 3 June 2024 (08:07:35 CEST)
REVIEW
|
doi:10.20944/preprints202307.0539.v3
Subject:
Medicine And Pharmacology,
Gastroenterology And Hepatology
Keywords:
Hepatocellular carcinoma; tyrosine kinase inhibitors; immune checkpoint inhibitors; biomarkers
Online: 17 July 2023 (13:22:33 CEST)
REVIEW
|
doi:10.20944/preprints202403.1203.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
rectal cancer; total neoadjuvant treatment; immunocheckpoint inhibitors; nonoperative management; ctDNA.
Online: 20 March 2024 (16:08:21 CET)
REVIEW
|
doi:10.20944/preprints201903.0256.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
immunocheckpoint inhibitors; chemotherapy; tirosin kinase inhibitors; angiogenesis
Online: 28 March 2019 (06:48:37 CET)
REVIEW
|
doi:10.20944/preprints202003.0251.v2
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
gastric acid suppressant; chemotherapy; tyrosine kinase inhibitors; proton pump inhibitors
Online: 31 March 2020 (03:40:46 CEST)
CASE REPORT
|
doi:10.20944/preprints202402.0658.v3
Subject:
Medicine And Pharmacology,
Medicine And Pharmacology
Keywords:
pharmacokinetic-pharmacodynamic interactions; low-dose methotrexate; proton pump inhibitors; analgesics; pancytopenia; hepatotoxicity
Online: 1 April 2024 (11:53:15 CEST)
ARTICLE
|
doi:10.20944/preprints202403.0239.v1
Subject:
Medicine And Pharmacology,
Clinical Medicine
Keywords:
JAK inhibitors; Psoriasis; Psoriatic arthitis
Online: 5 March 2024 (06:02:35 CET)
ARTICLE
|
doi:10.20944/preprints202405.1174.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
Gastric cancer; Proto-Oncogene Protein c-met; Tyrosine Kinase Inhibitors; Cell Line; Tumor
Online: 17 May 2024 (12:28:09 CEST)
REVIEW
|
doi:10.20944/preprints202306.0041.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
APE1; inhibitors; cancer.
Online: 1 June 2023 (07:05:48 CEST)
REVIEW
|
doi:10.20944/preprints202407.1744.v1
Subject:
Biology And Life Sciences,
Life Sciences
Keywords:
BRCA1; BRCA2; promoter methylation; breast cancer; ovarian; cancer; liquid biopsy; PARP inhibitors
Online: 23 July 2024 (07:30:06 CEST)
REVIEW
|
doi:10.20944/preprints202406.0356.v1
Subject:
Medicine And Pharmacology,
Gastroenterology And Hepatology
Keywords:
liver transplantation; hepatocellular carcinoma; Immune checkpoint inhibitors; allograft rejection
Online: 6 June 2024 (07:45:00 CEST)
ARTICLE
|
doi:10.20944/preprints202306.2038.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
Neurodegenerative diseases; cholinesterase inhibitors; monoaminoxidase inhibitors; photo-pharmacology
Online: 29 June 2023 (02:47:23 CEST)
REVIEW
|
doi:10.20944/preprints202401.0800.v1
Subject:
Medicine And Pharmacology,
Dermatology
Keywords:
psoriasis; oral therapies; topical therapies; biologics; Jak inhibitors; PDE4 inhibitors; systemic treatment; IL-17 inhibitors; IL-23 inhibitors; tapinarof; roflumilast
Online: 10 January 2024 (08:49:06 CET)
REVIEW
|
doi:10.20944/preprints202407.1534.v1
Subject:
Medicine And Pharmacology,
Hematology
Keywords:
lymphoma; B‐cell; hematologic neoplasms; bruton tyrosine kinase; protein kinase inhibitors; drug resistance; neoplasm; ibrutinib; pirtobrutinib; molecular targeted therapy; chronic lymphocytic leukemia; hematopoietic stem cell transplantation; covalent inhibitors; protein degradation
Online: 18 July 2024 (17:24:05 CEST)
REVIEW
|
doi:10.20944/preprints201905.0358.v1
Subject:
Medicine And Pharmacology,
Pharmacology And Toxicology
Keywords:
alloimmune response; immunosuppressants; calcineurin inhibitors; corticosteroids; mTOR inhibitors; neurotoxicity; neuroprotective effects
Online: 29 May 2019 (16:37:44 CEST)
REVIEW
|
doi:10.20944/preprints202405.0573.v1
Subject:
Medicine And Pharmacology,
Gastroenterology And Hepatology
Keywords:
Proton Pump Inhibitors (PPIs); Vonoprazan (VPZ); Intravenous infusion; Oral therapy; Bleeding peptic ulcers; Endoscopic therapy
Online: 9 May 2024 (09:15:54 CEST)
REVIEW
|
doi:10.20944/preprints202403.0902.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
NSCLC; lung cancer; gut microbiota; immunotherapy; immune checkpoint inhibitors
Online: 15 March 2024 (07:33:31 CET)
ARTICLE
|
doi:10.20944/preprints202404.1746.v1
Subject:
Biology And Life Sciences,
Life Sciences
Keywords:
Retinoblastoma; Epigenetic Reprogramming; Cancer Therapy; Epigenetic Therapy; DNA methyltransferase (DNMT) inhibitors
Online: 26 April 2024 (12:19:15 CEST)
REVIEW
|
doi:10.20944/preprints202407.2623.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
Tumor Mutational Burden (TMB); Immune Checkpoint Inhibitors (ICIs); Biomarkers; Cancer Immunotherapy; Cancer Treatment Outcomes; Personalized Medicine
Online: 2 August 2024 (11:50:44 CEST)
REVIEW
|
doi:10.20944/preprints202208.0008.v3
Subject:
Medicine And Pharmacology,
Pharmacology And Toxicology
Keywords:
adamantanes; antivirals; cap-dependent endonuclease inhibitors; influenza; neuraminidase inhibitors; umifenovir
Online: 19 September 2023 (04:16:16 CEST)
ARTICLE
|
doi:10.20944/preprints202405.0084.v1
Subject:
Biology And Life Sciences,
Virology
Keywords:
natural extracts; chitosan; liposomes; encapsulation; drug release; coronavirus HCoV-0C43; antiviral activity; natural inhibitors of viral replication; cytotoxicity; phototoxicity
Online: 2 May 2024 (12:03:47 CEST)
ARTICLE
|
doi:10.20944/preprints202307.1058.v1
Subject:
Medicine And Pharmacology,
Cardiac And Cardiovascular Systems
Keywords:
Heart Failure; Therapy; type-2 sodium-glucose cotransporters inhibitors; angiotensin receptor neprylisin inhibitors
Online: 17 July 2023 (15:07:48 CEST)
ARTICLE
|
doi:10.20944/preprints201801.0213.v1
Subject:
Chemistry And Materials Science,
Analytical Chemistry
Keywords:
bichalcones; sirtuin inhibitors; virtual screening
Online: 23 January 2018 (09:12:43 CET)
REVIEW
|
doi:10.20944/preprints202402.1593.v1
Subject:
Medicine And Pharmacology,
Endocrinology And Metabolism
Keywords:
type 2 diabetes; therapeutic inertia; clinical guidelines; sodium-glucose cotransporter-2 inhibitors; glucagon-like peptide-1 receptor agonists; primary health care
Online: 28 February 2024 (10:53:42 CET)
ARTICLE
|
doi:10.20944/preprints202309.1391.v1
Online: 21 September 2023 (03:32:12 CEST)
REVIEW
|
doi:10.20944/preprints202108.0364.v1
Subject:
Medicine And Pharmacology,
Tropical Medicine
Keywords:
dengue virus; antiviral targets; NS5; flavivirus; polymerase; nucleoside inhibitors; non-nucleoside inhibitors
Online: 17 August 2021 (14:07:29 CEST)
REVIEW
|
doi:10.20944/preprints202408.0401.v1
Subject:
Medicine And Pharmacology,
Other
Keywords:
Immunotherapy; Cancer Immunotherapy; Gut Microbiota; Microbiota Modulation; Immune checkpoint Inhibitors
Online: 6 August 2024 (08:35:02 CEST)
REVIEW
|
doi:10.20944/preprints202311.1805.v1
Subject:
Biology And Life Sciences,
Cell And Developmental Biology
Keywords:
HDAC6; histone deacetylases inhibitors; colorectal cancer
Online: 28 November 2023 (10:13:23 CET)
REVIEW
|
doi:10.20944/preprints202305.1789.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
PTK6; Colorectal cancer; Tyrosine Kinase Inhibitors
Online: 25 May 2023 (09:52:24 CEST)
REVIEW
|
doi:10.20944/preprints202204.0065.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
COVID-19; Main protease; Mpro; inhibitors
Online: 8 April 2022 (03:01:37 CEST)
ARTICLE
|
doi:10.20944/preprints202407.1422.v1
Subject:
Computer Science And Mathematics,
Mathematical And Computational Biology
Keywords:
Alzheimer's disease; structural flexibility; AChE inhibitors
Online: 17 July 2024 (11:27:37 CEST)
REVIEW
|
doi:10.20944/preprints202406.0880.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
Dendritic cells; DC based cancer vaccine; Immune checkpoint inhibitors; Cancer Therapy; Combinatorial therapy
Online: 13 June 2024 (11:51:42 CEST)
REVIEW
|
doi:10.20944/preprints201907.0286.v1
Subject:
Biology And Life Sciences,
Virology
Keywords:
HIV-1 Gag; Gag inhibitors; Protease; Protease inhibitors; drug resistance mutations; drug design
Online: 25 July 2019 (10:05:03 CEST)
ARTICLE
|
doi:10.20944/preprints202001.0279.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
NS3 inhibitors; allosteric inhibitors; NS4A; peptidomimetics; imidazole; hepatitis C virus; molecular dynamics; Flaviviridae; DSLS; binding assay
Online: 24 January 2020 (11:11:46 CET)
REVIEW
|
doi:10.20944/preprints201805.0129.v1
Subject:
Medicine And Pharmacology,
Gastroenterology And Hepatology
Keywords:
BET inhibitors; HDAC inhibitors; pancreatic cancer; aberrant transcription; enhancers; transcription factors; distal regulatory elements; MYC; FOXA1; BRD4
Online: 8 May 2018 (10:47:27 CEST)
ARTICLE
|
doi:10.20944/preprints202307.1626.v1
Subject:
Medicine And Pharmacology,
Medicine And Pharmacology
Keywords:
Proton pump inhibitors; Clopidogrel; Stroke; Myocardial infarction
Online: 25 July 2023 (07:26:31 CEST)
REVIEW
|
doi:10.20944/preprints202401.1747.v1
Subject:
Medicine And Pharmacology,
Hematology
Keywords:
chronic lymphocytic leukemia; BTK inhibitors; BCL-2 inhibitors; prognostic scores; predictive factors; TP53 abnormalities; IGHV; complex karyotype
Online: 24 January 2024 (13:39:51 CET)
ARTICLE
|
doi:10.20944/preprints202402.0503.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
HNSCC; PI3K inhibitors; ErbB inhibitor; targeted therapy
Online: 8 February 2024 (14:11:24 CET)
ARTICLE
|
doi:10.20944/preprints202212.0542.v2
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
safety analysis; targeted therapy; monoclonal antibody therapy; immune checkpoint inhibibitors; tyrosine kinase inhibitors; breast cancer; gynecological cancer; Helixor; Viscum album L.; PARP inhibitors; CDK 4/6 inhibitors
Online: 30 December 2022 (12:00:35 CET)
ARTICLE
|
doi:10.20944/preprints202304.0063.v1
Subject:
Medicine And Pharmacology,
Medicine And Pharmacology
Keywords:
Cx43; gap junctions; conductance; inhibitors; docking; IC50
Online: 5 April 2023 (12:30:58 CEST)
REVIEW
|
doi:10.20944/preprints202105.0140.v1
Subject:
Engineering,
Automotive Engineering
Keywords:
Adsorption; Scale Inhibitors; Fine sands; Colloids; Reservoir
Online: 7 May 2021 (10:42:36 CEST)
REVIEW
|
doi:10.20944/preprints202306.0128.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
PD-L1; CTCs; immunotherapy; immune checkpoint inhibitors
Online: 2 June 2023 (04:28:01 CEST)
ARTICLE
|
doi:10.20944/preprints202309.1065.v1
Subject:
Medicine And Pharmacology,
Dermatology
Keywords:
psoriasis; plasma cytokines; TNFα inhibitors; etanercept; infliximab; adalimumab
Online: 18 September 2023 (02:32:17 CEST)
REVIEW
|
doi:10.20944/preprints202310.2105.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
radiotherapy; CD8+ T cells; immune checkpoint inhibitors
Online: 31 October 2023 (17:22:30 CET)
REVIEW
|
doi:10.20944/preprints202306.0609.v1
Subject:
Medicine And Pharmacology,
Medicine And Pharmacology
Keywords:
Kinases; human diseases; macrocyclic inhibitors; drug discovery
Online: 8 June 2023 (08:54:08 CEST)
REVIEW
|
doi:10.20944/preprints202307.0043.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
Gliomas; Tumour Microenvironment; Immunotherapy; Immune Checkpoint Inhibitors; Vaccines
Online: 4 July 2023 (02:39:07 CEST)
ARTICLE
|
doi:10.20944/preprints202311.1799.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
usnic acid derivatives; TDP1 inhibitors; anticancer therapy; topotecan
Online: 28 November 2023 (10:06:47 CET)
ARTICLE
|
doi:10.20944/preprints202407.1916.v1
Subject:
Medicine And Pharmacology,
Gastroenterology And Hepatology
Keywords:
cardiovascular disease; hepatic fibrosis; metabolic dysfunction-associated steatotic liver disease; sodium-glucose cotransporter 2 inhibitors; serum lipids
Online: 24 July 2024 (08:27:35 CEST)
ARTICLE
|
doi:10.20944/preprints202405.1422.v1
Subject:
Medicine And Pharmacology,
Gastroenterology And Hepatology
Keywords:
eosinophilic esophagitis; esophagus; proton pump inhibitors
Online: 22 May 2024 (07:54:48 CEST)
REVIEW
|
doi:10.20944/preprints202404.0091.v1
Subject:
Medicine And Pharmacology,
Hematology
Keywords:
menin; menin inhibitors; leukemia; KMT2A; NPM1
Online: 2 April 2024 (02:51:43 CEST)
REVIEW
|
doi:10.20944/preprints202307.1892.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
Oncolytic virus; immune checkpoint inhibitors; immunotherapy
Online: 28 July 2023 (10:58:30 CEST)
ARTICLE
|
doi:10.20944/preprints202307.0031.v1
Subject:
Chemistry And Materials Science,
Applied Chemistry
Keywords:
Ionic Liquids; Corrosion Inhibitors; Bio-based
Online: 4 July 2023 (02:23:59 CEST)
ARTICLE
|
doi:10.20944/preprints201801.0027.v1
Subject:
Chemistry And Materials Science,
Organic Chemistry
Keywords:
microginins; cyanobacteria; Microcystis; aminopeptidase M inhibitors
Online: 5 January 2018 (04:16:23 CET)
ARTICLE
|
doi:10.20944/preprints202105.0638.v1
Subject:
Medicine And Pharmacology,
Immunology And Allergy
Keywords:
18F-FDG PET/CT; contrast-enhanced CT; melanoma; metastases; tyrosine kinase inhibitors; Immune checkpoint inhibitors; follow-up; therapy monitoring
Online: 26 May 2021 (13:14:06 CEST)
ARTICLE
Subject:
Medicine And Pharmacology,
Immunology And Allergy
Keywords:
18F-FDG PET/CT; contrast-enhanced CT; melanoma; metastases; tyrosine kinase inhibitors; Immune checkpoint inhibitors; follow-up; therapy monitoring
Online: 25 January 2021 (15:01:17 CET)
REVIEW
|
doi:10.20944/preprints202104.0679.v1
Subject:
Medicine And Pharmacology,
Immunology And Allergy
Keywords:
Sildenafil; phosphodiesterase 5 inhibitors; drug repurposing; cancer; chemoadjuvant
Online: 26 April 2021 (15:02:08 CEST)
REVIEW
|
doi:10.20944/preprints202312.1388.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
Rheb1; Rheb2; Cancer; mTOR; Hallmarks; Neurons; Rheb1 inhibitors
Online: 19 December 2023 (05:58:46 CET)
ARTICLE
|
doi:10.20944/preprints202308.0880.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
tyrosyl-DNA phosphodiesterase 1 (Tdp1); tyrosyl-DNA phosphodiesterase 2 (Tdp2); usnic acid; Tdp2 inhibitors; Tdp1 inhibitors
Online: 11 August 2023 (08:18:31 CEST)
ARTICLE
|
doi:10.20944/preprints202109.0520.v1
Subject:
Biology And Life Sciences,
Biology And Biotechnology
Keywords:
Phytoene, Dunaliella salina, mitosis inhibitors, herbicides, red light
Online: 30 September 2021 (14:18:55 CEST)
ARTICLE
|
doi:10.20944/preprints202407.0117.v1
Subject:
Biology And Life Sciences,
Immunology And Microbiology
Keywords:
Acral, mucosal, anti-PD-1 Abs, BRAF plus MEK inhibitors, adjuvant therapy
Online: 2 July 2024 (10:51:38 CEST)
REVIEW
|
doi:10.20944/preprints202011.0005.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
aminoacyl-tRNA synthetase, small molecule inhibitors, human diseases
Online: 2 November 2020 (09:09:37 CET)
REVIEW
|
doi:10.20944/preprints202405.1755.v1
Subject:
Medicine And Pharmacology,
Transplantation
Keywords:
Keywords. Sodium-glucose- cotransporters type 2 inhibitors, glucose reabsorption, sodium reabsorption, randomized clinical trials, diabetes, heart failure, chronic kidney disease, kidney transplantati
Online: 27 May 2024 (14:31:30 CEST)
REVIEW
|
doi:10.20944/preprints201809.0291.v1
Subject:
Biology And Life Sciences,
Immunology And Microbiology
Keywords:
CCR6, CCL20, Inhibitors, TH17, Treg, Inflammatory diseases, Cancer
Online: 17 September 2018 (09:31:43 CEST)
ARTICLE
|
doi:10.20944/preprints201807.0199.v1
Subject:
Biology And Life Sciences,
Agricultural Science And Agronomy
Keywords:
ALS-inhibitors; horseweed; multiple-resistance; alternative chemical control
Online: 11 July 2018 (11:56:59 CEST)
REVIEW
|
doi:10.20944/preprints202307.2046.v1
Subject:
Medicine And Pharmacology,
Pharmacy
Keywords:
CADD; SBDD; LBDD; kinase; small molecule kinase inhibitors
Online: 31 July 2023 (03:05:42 CEST)
ARTICLE
|
doi:10.20944/preprints202003.0425.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
cancer; immune checkpoint inhibitors; survival; antibiotic; meta-analysis
Online: 29 March 2020 (06:43:23 CEST)
REVIEW
|
doi:10.20944/preprints202112.0282.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
Acalabrutinib; Bruton’s tyrosine kinase; BTK; CLL; Covalent inhibitors; COVID-19; Ibrutinib; Non-covalent inhibitors; Fenebrutinib; MK1026; Pirtobrutinib; Spebrutinib; Tirabrutinib; Zanubrutinib
Online: 16 December 2021 (16:13:54 CET)
CASE REPORT
|
doi:10.20944/preprints202307.0658.v1
Subject:
Medicine And Pharmacology,
Endocrinology And Metabolism
Keywords:
hypertriglyceridemia; dyslipidemia; evinacumab; ANGPTL3-inhibitors; lipid-lowering drugs
Online: 11 July 2023 (10:45:58 CEST)
ARTICLE
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doi:10.20944/preprints201905.0046.v1
Subject:
Chemistry And Materials Science,
Medicinal Chemistry
Keywords:
aminopeptidases; inhibitors; aminophosphonate; phenylglycine analogues; fluorine substituted; molecular modeling
Online: 6 May 2019 (10:16:45 CEST)
ARTICLE
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
CYP3A5; androgen receptor; African American; CYP3A5 inhibitors/inducers
Online: 6 March 2020 (03:33:52 CET)
REVIEW
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doi:10.20944/preprints202309.0633.v1
Subject:
Medicine And Pharmacology,
Oncology And Oncogenics
Keywords:
metastatic hormone-sensitive prostate cancer; new hormonal agents; transcriptomic profiling; DNA damage repair genes; tumor suppressor genes; androgen receptor; immunotherapy; CDK4/6 inhibitors; PARP inhibitors; AKT inhibitors.
Online: 11 September 2023 (07:17:07 CEST)
REVIEW
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doi:10.20944/preprints202304.0843.v2
Subject:
Medicine And Pharmacology,
Hematology
Keywords:
CLL, Zanubrutinib, BTK inhibitors, efficacy, safety, chronic lymphocytic leukemia
Online: 22 May 2023 (16:15:16 CEST)
COMMUNICATION
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doi:10.20944/preprints202012.0365.v1
Subject:
Chemistry And Materials Science,
Analytical Chemistry
Keywords:
corrosion; amino acids; inhibitors; steel; iron; Monte Carlo simulation
Online: 15 December 2020 (10:09:29 CET)
ARTICLE
|
doi:10.20944/preprints201806.0131.v1
Subject:
Biology And Life Sciences,
Biochemistry And Molecular Biology
Keywords:
histone demethylase inhibitors; DNA damage; epigenetic drugs; breast cancer
Online: 8 June 2018 (12:29:10 CEST)
REVIEW
|
doi:10.20944/preprints201911.0264.v1
Subject:
Medicine And Pharmacology,
Endocrinology And Metabolism
Keywords:
cardiovascular risk; dipeptidyl peptidase-4 inhibitors; glucagon like peptide-1 receptor agonists; sodium glucose cotransporter-2 inhibitors; type 2 diabetes mellitus
Online: 24 November 2019 (04:26:47 CET)
CASE REPORT
|
doi:10.20944/preprints202312.1085.v1
Subject:
Medicine And Pharmacology,
Obstetrics And Gynaecology
Keywords:
Antiphospholipid syndrome; TNF-α Inhibitors; Dangerous pregnancy; gestational weeks
Online: 14 December 2023 (12:15:47 CET)
ARTICLE
|
doi:10.20944/preprints202403.1880.v1
Subject:
Public Health And Healthcare,
Other
Keywords:
Anti-interferon-γ autoantibodies; herpes zoster; monocyte chemoattractant protein-1; IFN-γ inducible protein-10; Janus kinas inhibitors; rheumatoid arthritis.
Online: 1 April 2024 (10:20:44 CEST)
REVIEW
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doi:10.20944/preprints202309.0229.v1
Subject:
Medicine And Pharmacology,
Hematology
Keywords:
acute myeloid leukemia; immunotherapy; checkpoint inhibitors; new therapeutic landscapes
Online: 6 September 2023 (14:36:13 CEST)